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Cat. No. Product Name Target Signaling Pathways
T27205 DPI 201-106

DPI-201-106

Sodium Channel Membrane transporter/Ion channel
DPI 201-106对电压门控钠通道的有心脏选择性调节活性,从而产生正性肌力作用。DPI 201-106 具有协同肌膜和细胞内作用机制。
T7191 Diphenyleneiodonium chloride

二苯基氯化碘盐,DPI

NOS; Reactive Oxygen Species; NADPH; TRP/TRPV Channel Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB
Diphenyleneiodonium chloride (DPI) 是 NADPH 氧化酶抑制剂,也是 TRPA1激活剂,EC50为 1 - 3 μM 。它选择性抑制胞内活性氧。
T15165 DPI-3290

Org 41793

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potent antinociceptive activity. DPI-3290 is one of a series of novel centrally acting agents.
T10700 (+)-CBI-CDPI1

Others Others
(+)-CBI-CDPI1 is an enhanced functional analog of CC-1065. It is a DNA alkylating agent and an antibody-drug conjugates (ADCs) toxin.
T10701 (+)-CBI-CDPI2

Others Others
(+)-CBI-CDPI2 is an enhanced functional analog of CC-1065.
TQ0095 Brincidofovir

CMX001,HDP-CDV

Others; Antiviral; HSV Immunology/Inflammation; Microbiology/Virology; Others
Brincidofovir (HDP-CDV) 是 Cidofovir 的一种具有口服活性的亲脂性形式的前体药物,是一种口服长效的抗病毒药物,有广泛的抗 DNA 病毒活性。

化合物

DPI 201-106
Cat.No: T27205
Synonym: DPI-201-106
Target: Sodium Channel
Diphenyleneiodonium chloride
Cat.No: T7191
Synonym: 二苯基氯化碘盐,DPI
Target: NOS, Reactive Oxygen Species, NADPH, TRP/TRPV Channel
DPI-3290
Cat.No: T15165
Synonym: Org 41793
Target: Opioid Receptor
(+)-CBI-CDPI1
Cat.No: T10700
Synonym:
Target: Others
(+)-CBI-CDPI2
Cat.No: T10701
Synonym:
Target: Others
Brincidofovir
Cat.No: TQ0095
Synonym: CMX001,HDP-CDV
Target: Others, Antiviral, HSV
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