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Search Results for " cyclosporine "

7

抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T6459 Cyclosporine

Phosphatase Metabolism
Cyclosporine 是一种钙调神经磷酸酶通路抑制剂,用作免疫抑制剂以防止器官移植中的排斥反应。
T9936 ZX-J-19J

N-(2,3-Diphenyl-6-quinoxalinyl)octanamide

Others Others
ZX-J-19J (N-(2,3-Diphenyl-6-quinoxalinyl)octanamide) 是 Cyclophilin J 的抑制剂,对肿瘤细胞生长有显着的抑制作用,与环孢素 A 相当,但比 5-氟尿嘧啶强得多。
T70889 Oxeclosporin

Oxeclosporin is a hydroxyethyl derivative of serine(8)-cyclosporine; inhibits proliferation and functions of lymphocytes.
T32020 Gusperimus

Deoxyspergualin,15-Deoxyspergualin

Gusperimus was synthesized by chemical modification of spergualin and in combination with cyclosporine A to prevent diabetes in susceptible NOD mice.
T28080 Mocravimod

KRP 203 free base,KRP-203,KRP203

Mocravimod is an agonist of sphingosine 1-phosphate receptor type 1. Mocravimod ameliorates atherosclerosis in LDL-R-/- mice. KRP-203 attenuates rat autoimmune myocarditis. KRP-203 combined with cyclosporine prolonged graft survival and abrogated transpla
T34999 UNIL-088

UNIL 088

UNIL088 is a water-soluble prodrug of cyclosporine A (CsA) designed for topical ocular delivery. The pro-moiety is grafted via an ester function to CsA and the solubilizing group is a phosphate ion. UNIL-088 can be rapidly hydrolysed under physiological c
T0679 Ketoconazole

R-41400,Xolegel,(±)-Ketoconazol,酮康唑,Extina

NADPH-oxidase; P450; Hydroxylase; Antifungal; Ras GPCR/G Protein; Immunology/Inflammation; MAPK; Metabolism; Microbiology/Virology
Ketoconazole (R-41400) 是一种咪唑类抗真菌剂,也是一种 CYP3A4 抑制剂。

化合物

Cyclosporine
Cat.No: T6459
Synonym:
Target: Phosphatase
ZX-J-19J
Cat.No: T9936
Synonym: N-(2,3-Diphenyl-6-quinoxalinyl)octanamide
Target: Others
Oxeclosporin
Cat.No: T70889
Synonym:
Target:
Gusperimus
Cat.No: T32020
Synonym: Deoxyspergualin,15-Deoxyspergualin
Target:
Mocravimod
Cat.No: T28080
Synonym: KRP 203 free base,KRP-203,KRP203
Target:
UNIL-088
Cat.No: T34999
Synonym: UNIL 088
Target:
Ketoconazole
Cat.No: T0679
Synonym: R-41400,Xolegel,(±)-Ketoconazol,酮康唑,Extina
Target: NADPH-oxidase, P450, Hydroxylase, Antifungal, Ras
Cat. No. Product Name Target Signaling Pathways
T0945 Cyclosporin A

环孢素,Cyclosporine A,Ciclosporin,Cyclosporine,环孢菌素

Phosphatase; Antibiotic; Complement System Immunology/Inflammation; Metabolism; Microbiology/Virology
Cyclosporin A 属于天然产物,是一种真菌的活性代谢产物,一种环状多肽。Cyclosporin A 是一种能与亲环素结合的免疫抑制剂,可以抑制 calcineurin (IC50=7 nM)。

天然产物

Cyclosporin A
Cat.No: T0945
Synonym: 环孢素,Cyclosporine A,Ciclosporin,Cyclosporine,环孢菌素
Target: Phosphatase, Antibiotic, Complement System
TargetMol Loading
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