Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4277 |
Osilodrostat
LCI699 |
Glucocorticoid Receptor; Others; Hydroxylase | Endocrinology/Hormones; Metabolism; Others |
Osilodrostat (LCI699) 是一种有效的人11β-羟化酶和醛固酮合成酶抑制剂,IC50分别值为2.5 和0.7nM。 | |||
T0293 |
Metyrapone
美替拉酮,甲吡酮,NSC-25265,Su-4885 |
Others; P450; Dehydrogenase; Autophagy | Autophagy; Metabolism; Others |
Metyrapone (NSC-25265) 是 STEROID 11-BETA-MONOOXYGENASE 酶抑制剂。 它被用作库欣综合征诊断中下丘脑-垂体反馈机制的测试。 | |||
T0293L |
Metyrapone Tartrate
SU 4885,Metopirone tartrate,SU-4885,SU4885 |
||
Metyrapone Tartrate is an inhibitor of the STEROID 11-beta-monooxygenase enzyme which is used as a test for feedback hypothalamic-pituitary mechanism in the diagnosis of Cushing SYNDROME. |