Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3277 |
Tulobuterol hydrochloride
Lobuterol,Hokunalin,Berachin,盐酸妥布特罗 |
Influenza Virus; Adrenergic Receptor; Antibiotic | GPCR/G Protein; Microbiology/Virology; Neuroscience |
Tulobuterol hydrochloride (Hokunalin) 是一种长效的 β2肾上腺素受体激动剂,可减少慢性阻塞性肺疾病和支气管哮喘的发作频率。它也是一种拟交感神经药,用作透皮贴剂,可增加正常的横膈膜肌肉力量。它抑制鼻病毒复制并调节气道炎症。 | |||
T3463 |
NVP-ACC789
ACC-789,ZK202650 |
VEGFR; PDGFR | Angiogenesis; Tyrosine Kinase/Adaptors |
NVP-ACC789 (ZK202650) 是一种人VEGFR-1,VEGFR-2(鼠VEGFR-2),VEGFR-3 和 PDGFR-β 的抑制剂,它们的 IC50 值分别为 0.38,0.02 (0.23),0.18 和 1.4 μM。 | |||
T16355 |
NSC781406
|
PI3K; mTOR | PI3K/Akt/mTOR signaling |
NSC781406是一种高效PI3K 和mTOR 抑制剂,其PI3Kα的IC50值为2 nM。 | |||
T16439 |
PC786
|
Others | Others |
PC786 shows effective antiviral activity against RSV-A (IC50 <0.09 to 0.71 nM) and RSV-B (IC50, 1.3 to 50.6 nM). PC786 is an inhaled respiratory syncytial virus L protein polymerase inhibitor. |