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Search Results for " andrographolide "

4

抑制剂 & 化合物

14

天然产物

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Cat. No. Product Name Target Signaling Pathways
T125901 14-Epiandrographolide

14-Epiandrographolide 是从穿心莲地上部分提取到的化合物,可诱导细胞分化,可用于研究多发性硬化症。
T40971 Dehydroandrographolide succinate potassium sodium salt

Dehydroandrographolide succinate (potassium sodium salt), derived from the herbal medicine Andrographis paniculata (Burm f) Nees, is a versatile compound highly utilized for the treatment of viral pneumonia and viral upper respiratory tract infections due to its potent immunostimulatory, anti-infective, and anti-inflammatory properties.
T74895 Anti-inflammatory agent 31

Anti-inflammatory agent 31 是一种穿心莲内酯衍生物,是一种抗炎剂 (anti-inflammatoryagent)。Anti-inflammatory agent 31 通过上游阻断PI3K/Akt 和ERK1/2 MAPK 激活来抑制NF-kB 激活。Anti-inflammatory agent 31 能够恢复细胞内 GSH 水平并对肝脏具有保护作用。
T73292 ZIKV-IN-3

ZIKV-IN-3, 一个穿心莲内酯衍生物,作为有效的ZIKV NS5甲基转移酶(MTase)抑制剂,展示了18.34 μM的IC50值。该化合物能抑制ZIKV的复制与感染,适用于寨卡病毒(ZIKV)的研究。

化合物

14-Epiandrographolide
Cat.No: T125901
Synonym:
Target:
Dehydroandrographolide succinate potassium sodium salt
Cat.No: T40971
Synonym:
Target:
Anti-inflammatory agent 31
Cat.No: T74895
Synonym:
Target:
ZIKV-IN-3
Cat.No: T73292
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T2898 Andrographolide

Andrographis,穿心莲内酯

SARS-CoV; Influenza Virus; NF-κB; Autophagy Autophagy; Microbiology/Virology; NF-κB
Andrographolide (Andrographis) 是 NF-κB 的不可逆拮抗剂,具有抗病毒、抗炎和抗血小板聚集活性和潜在的抗肿瘤作用。
TQ0185 14-Deoxy-11,12-didehydroandrographolide

AP10,14-脱氧-11,12-二去氢穿心莲内酯,14-dehydro Andrographolide

NF-κB NF-κB
14-Deoxy-11,12-didehydroandrographolide (AP10) 是一种 Andrographolide 的类似物,能够抑制 NF-κB 活性。
T3884 Neoandrographolide

Neoandrographiside,新穿心莲内酯

NOS; COX Immunology/Inflammation; Neuroscience
Neoandrographolide (Neoandrographiside) 是一种二萜类化合物,从穿心莲中分离得到。
T2S0257 Dehydroandrographolide succinate

Others; Influenza Virus Microbiology/Virology; Others
Dehydroandrographolide succinate 是从中药穿心莲中提取的一种天然产物,具有免疫刺激、抗感染和抗炎作用,有潜力研究病毒性肺炎和病毒性上呼吸道感染。
TQ0218 Deoxyandrographolide

去氧穿心莲内酯,14-deoxyandrographolide

IL Receptor; TNF Apoptosis; Immunology/Inflammation
Deoxyandrographolide (14-deoxyandrographolide) 抑制 LPS 诱导的 iNOS mRNA 水平升高以及促炎症介质 TNF-α 和 IL-6 的产生。它增强 NGF 诱导的神经突起生长。
T8288 14-Deoxyandrographolide

去氧穿心莲内酯,14-去氧穿心莲内酯

Apoptosis; Others Apoptosis; Others
14-Deoxyandrographolide 是穿心莲中的一种天然产物,是一种钙通道阻断剂,具有保肝功效。它通过诱导 TNFRSF1A 的释放,使肝细胞对 TNF-α 介导的凋亡脱敏。
TN2463 14-Deoxy-11-oxoandrographolide

Others Others
14-Deoxy-11-oxoandrographolide is a natural product from Andrographis paniculata
TN3518 Bisandrographolide A

Others Others
Bisandrographolide A activates TRPV4 channels, could play a role in some of the effects of Andrographis extract described in traditional medicine.
TN2623 14-Deoxy-17-hydroxyandrographolide

Antifection Microbiology/Virology
14-Deoxy-17-hydroxyandrographolide是一种天然产物,属于爵床科穿心莲属,其产品编号为 TN2623,CAS号为 869384-82-7。14-Deoxy-17-hydroxyandrographolide可用作对照参考。
T72580 Isoandrographolide

Isoandrographolide 具有诱导细胞分化和保肝活性。Isoandrographolide 可抑制 NLRP3炎症小体激活并减轻小鼠矽肺。
T2738 Dehydroandrographolide

NOS; Influenza Virus Immunology/Inflammation; Microbiology/Virology
Dehydroandrographolide 是从草药穿心莲中提取的一种天然产物。它通过使 iNOS 失活来降低 LPS 诱导的急性肺损伤中的氧化应激,有抗感染活性。
T13582 Bisandrographolide C

Others Others
Bisandrographolide C is identified from Andrographis paniculata. Bisandrographolide C activates TRPV1 and TRPV3 channels (Kds: 289 and 341 μM) and protects cardiomyocytes from hypoxia-reoxygenation injury.
TN5585 14-Deoxy-11-hydroxyandrographolide

14-Deoxy-11-hydroxyandrographolide shows potent cell differentiation-inducing activity towards mouse myeloid leukemia (M1) cells.
TN5586 14-Deoxy-12-hydroxyandrographolide

14-Deoxy-12-hydroxyandrographolide是一种天然产物,属于爵床科穿心莲属,其产品编号为 TN5586,CAS号为 219721-33-2。14-Deoxy-12-hydroxyandrographolide可用作对照参考。

天然产物

Andrographolide
Cat.No: T2898
Synonym: Andrographis,穿心莲内酯
Target: SARS-CoV, Influenza Virus, NF-κB, Autophagy
14-Deoxy-11,12-didehydroandrographolide
Cat.No: TQ0185
Synonym: AP10,14-脱氧-11,12-二去氢穿心莲内酯,14-dehydro Andrographolide
Target: NF-κB
Neoandrographolide
Cat.No: T3884
Synonym: Neoandrographiside,新穿心莲内酯
Target: NOS, COX
Dehydroandrographolide succinate
Cat.No: T2S0257
Synonym:
Target: Others, Influenza Virus
Deoxyandrographolide
Cat.No: TQ0218
Synonym: 去氧穿心莲内酯,14-deoxyandrographolide
Target: IL Receptor, TNF
14-Deoxyandrographolide
Cat.No: T8288
Synonym: 去氧穿心莲内酯,14-去氧穿心莲内酯
Target: Apoptosis, Others
14-Deoxy-11-oxoandrographolide
Cat.No: TN2463
Synonym:
Target: Others
Bisandrographolide A
Cat.No: TN3518
Synonym:
Target: Others
14-Deoxy-17-hydroxyandrographolide
Cat.No: TN2623
Synonym:
Target: Antifection
Isoandrographolide
Cat.No: T72580
Synonym:
Target:
Dehydroandrographolide
Cat.No: T2738
Synonym:
Target: NOS, Influenza Virus
Bisandrographolide C
Cat.No: T13582
Synonym:
Target: Others
14-Deoxy-11-hydroxyandrographolide
Cat.No: TN5585
Synonym:
Target:
14-Deoxy-12-hydroxyandrographolide
Cat.No: TN5586
Synonym:
Target:
TargetMol Loading
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