Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3068 |
AT9283
J-504568 |
Apoptosis; FLT; JAK; Bcr-Abl; Aurora Kinase; Autophagy | Angiogenesis; Apoptosis; Autophagy; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors |
AT9283 (J-504568) 是一种多靶点激酶抑制剂,抑制多种实体瘤在体内外的生长和存活,有效抑制Aurora A/B,JAK2/3,Abl (T315I),和Flt3,IC50值范围为 1-30 nM。 | |||
T21151 |
AT-9283 L-lactate
AT-9283,AT 9283,AT9283 |
||
AT-9283 L-lactate is an inhibitor of aurora kinase. | |||
T26675 |
AT-9283 HCl
AT-9283,AT-9283 hydrochloride,AT9283,AT 9283 |
||
AT-9283, a multi-targeted kinase inhibitor, is used potentially for the treatment of multiple myeloma. | |||
T28199 |
NS9283
NS 9283,NS-9283 |
AChR | Neuroscience |
NS9283 是有效的(α4)3(β2)2烟碱型ACh 受体的正向变构调节剂。NS9283在一系列神经系统疾病中有研究价值,如注意力缺陷多动障碍、精神分裂症、帕金森病和阿尔茨海默病。 |