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Cat. No. Product Name Target Signaling Pathways
T17252 SIM-688

SIM688

Estrogen/progestogen Receptor; NF-κB Endocrinology/Hormones; NF-κB
SIM-688 是一种选择性和口服活性的雌激素受体抑制剂,抑制 NF-κB 转录活性(在 HAECT-1 细胞中 IC50 = 122 nM)。
T26520 ABP688

ABP-688,ABP 688

GluR Neuroscience
ABP688 是一种非竞争性和选择性的 mGluR5 拮抗剂 (Ki = 1.7 nM)。 ABP688 可用作临床成像的 PET 示踪剂。
T1158L Phenoxybenzamine

NSC-37448,A688,NSC 37448,NSC37448,A-688

Phenoxybenzamine is an α-1 adrenergic receptor antagonist. Phenoxybenzamine may exert a neuroprotective effect by reducing neuroinflammation after traumatic brain injury.
T69649 NITD-688

NITD-688 是一种具有口服活性的登革病毒 (dengue virus)NS4B 蛋白的泛血清型抑制剂。 NITD-688 可用于登革热病毒 (DENV) 的研究。
T25737 Linetastine

TMK 688,TMK-688,TMK688

Lipoxygenase; LTR; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Linetastine (TMK-688) 是一种 5-脂氧合酶抑制剂(5-LOX),能抑制白三烯的产生,并能拮抗组胺的作用。Linetastine可用于研究哮喘、动脉粥样硬化和消化性溃疡。
T65213 2-(2-Aminoacetamido)-4-methylpentanoic acid

2-(2-Aminoacetamido)-4-methylpentanoic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65213,CAS号为 688-14-2。
T37419 Zetomipzomib

KZR-616, a first-in-class inhibitor of the immunoproteasome, selectively targets the LMP7 (IC50: 39/57 nM=hLMP7/mLMP7) and LMP2 (IC50: 131/179 nM=hLMP7/mLMP7) subunits of the immunoproteasome. KZR-616 has the potential for the research of multiple autoimmune diseases[1][2]. KZR-616 also inhibits MECL-1 subunit (IC50=623 nM) and constitutive proteasome β5 subunit (IC50=688 nM). KZR-616 maintains LMP7 and LMP2 selective inhibition in MOLT-4 cells. KZR-616 (250 nM) shows a comparable cytokine inhib...

化合物

SIM-688
Cat.No: T17252
Synonym: SIM688
Target: Estrogen/progestogen Receptor, NF-κB
ABP688
Cat.No: T26520
Synonym: ABP-688,ABP 688
Target: GluR
Phenoxybenzamine
Cat.No: T1158L
Synonym: NSC-37448,A688,NSC 37448,NSC37448,A-688
Target:
NITD-688
Cat.No: T69649
Synonym:
Target:
Linetastine
Cat.No: T25737
Synonym: TMK 688,TMK-688,TMK688
Target: Lipoxygenase, LTR, Histamine Receptor
2-(2-Aminoacetamido)-4-methylpentanoic acid
Cat.No: T65213
Synonym:
Target:
Zetomipzomib
Cat.No: T37419
Synonym:
Target:
TargetMol Loading
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