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抑制剂 & 化合物

6

天然产物

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Cat. No. Product Name Target Signaling Pathways
T8978 DD1

3,3'-Diamino-4'-methoxyflavone,HUN85111

Proteasome Proteases/Proteasome; Ubiquitination
DD1 (HUN85111) 是一种蛋白酶体抑制剂,可诱导人髓系肿瘤选择性凋亡。
T124460 5,6,7-Trihydroxy-4'-methoxyflavone

5,6,7-Trihydroxy-4'-methoxyflavone 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124460,CAS号为 6563-66-2。

化合物

DD1
Cat.No: T8978
Synonym: 3,3'-Diamino-4'-methoxyflavone,HUN85111
Target: Proteasome
5,6,7-Trihydroxy-4'-methoxyflavone
Cat.No: T124460
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T8246 4'-METHOXYFLAVONE

Others Others
4'-METHOXYFLAVONE 是一种天然产物。
TN3231 Pratol

7-Hydroxy-4'-methoxyflavone,三叶草,车轴草醇

Others Others
Pratol (7-Hydroxy-4'-methoxyflavone) 显着增加细胞中的黑色素含量和酪氨酸酶活性,而没有细胞毒性。
T3343 5-methoxyflavone

5-methoxy-2-phenylchromen-4-one,5-甲氧基黄酮

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
5-methoxyflavone (5-methoxy-2-phenylchromen-4-one) 是一种类黄酮,是DNA 聚合酶 β 的抑制剂和 β-淀粉样蛋白毒性的神经保护剂。它通过调控嗜离子 GABAA 受体,起到镇静中枢神经系统的作用。
T3981 Acacetin

4'-Methoxyapigenin,金合欢素,5,7-Dihydroxy-4'-methoxyflavone,Linarigenin

Apoptosis; IAP; COX; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; Neuroscience
Acacetin (5,7-Dihydroxy-4'-methoxyflavone) 是一种来自狗舌草的口服有效类黄酮。它停在 PI3Kγ 的 ATP 结合口袋中,可导致癌细胞周期停滞,并诱导细胞凋亡和自噬。它有抗癌和抗炎活性,有潜力研究疼痛相关疾病。
TN1276 4'-Hydroxywogonin

5,7,4'-trihydroxy-8-methoxyflavone,4'-羟基汉黄芩素

Others Others
4'-Hydroxywogonin has positive effect on inhabiting those human tumor lines in vitro, with IC50 value is 8.3-38.4ug/mL .
T3891 Oroxylin A-7-O-glucuronide

Oroxylin A Glucoronide,千层纸素A-7-0-Β-D-葡萄糖醛酸苷,Oroxyloside,Oroxylin A 7-O-beta-D-glucuronide

Others Others
Oroxylin A-7-O-glucuronide (Oroxylin A Glucoronide) 是一种类黄酮葡糖苷酸,提取自 Scutellaria baicalensis 干燥的根中,具有脯氨酰寡肽酶(POP)抑制作用。

天然产物

4'-METHOXYFLAVONE
Cat.No: T8246
Synonym:
Target: Others
Pratol
Cat.No: TN3231
Synonym: 7-Hydroxy-4'-methoxyflavone,三叶草,车轴草醇
Target: Others
5-methoxyflavone
Cat.No: T3343
Synonym: 5-methoxy-2-phenylchromen-4-one,5-甲氧基黄酮
Target: DNA/RNA Synthesis
Acacetin
Cat.No: T3981
Synonym: 4'-Methoxyapigenin,金合欢素,5,7-Dihydroxy-4'-methoxyflavone,Linarigenin
Target: Apoptosis, IAP, COX, Autophagy
4'-Hydroxywogonin
Cat.No: TN1276
Synonym: 5,7,4'-trihydroxy-8-methoxyflavone,4'-羟基汉黄芩素
Target: Others
Oroxylin A-7-O-glucuronide
Cat.No: T3891
Synonym: Oroxylin A Glucoronide,千层纸素A-7-0-Β-D-葡萄糖醛酸苷,Oroxyloside,Oroxylin A 7-O-beta-D-glucuronide
Target: Others
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