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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8978 |
DD1
3,3'-Diamino-4'-methoxyflavone,HUN85111 |
Proteasome | Proteases/Proteasome; Ubiquitination |
DD1 (HUN85111) 是一种蛋白酶体抑制剂,可诱导人髓系肿瘤选择性凋亡。 | |||
T124460 |
5,6,7-Trihydroxy-4'-methoxyflavone
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5,6,7-Trihydroxy-4'-methoxyflavone 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124460,CAS号为 6563-66-2。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8246 |
4'-METHOXYFLAVONE
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Others | Others |
4'-METHOXYFLAVONE 是一种天然产物。 | |||
TN3231 |
Pratol
7-Hydroxy-4'-methoxyflavone,三叶草,车轴草醇 |
Others | Others |
Pratol (7-Hydroxy-4'-methoxyflavone) 显着增加细胞中的黑色素含量和酪氨酸酶活性,而没有细胞毒性。 | |||
T3343 |
5-methoxyflavone
5-methoxy-2-phenylchromen-4-one,5-甲氧基黄酮 |
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
5-methoxyflavone (5-methoxy-2-phenylchromen-4-one) 是一种类黄酮,是DNA 聚合酶 β 的抑制剂和 β-淀粉样蛋白毒性的神经保护剂。它通过调控嗜离子 GABAA 受体,起到镇静中枢神经系统的作用。 | |||
T3981 |
Acacetin
4'-Methoxyapigenin,金合欢素,5,7-Dihydroxy-4'-methoxyflavone,Linarigenin |
Apoptosis; IAP; COX; Autophagy | Apoptosis; Autophagy; Immunology/Inflammation; Neuroscience |
Acacetin (5,7-Dihydroxy-4'-methoxyflavone) 是一种来自狗舌草的口服有效类黄酮。它停在 PI3Kγ 的 ATP 结合口袋中,可导致癌细胞周期停滞,并诱导细胞凋亡和自噬。它有抗癌和抗炎活性,有潜力研究疼痛相关疾病。 | |||
TN1276 |
4'-Hydroxywogonin
5,7,4'-trihydroxy-8-methoxyflavone,4'-羟基汉黄芩素 |
Others | Others |
4'-Hydroxywogonin has positive effect on inhabiting those human tumor lines in vitro, with IC50 value is 8.3-38.4ug/mL . | |||
T3891 |
Oroxylin A-7-O-glucuronide
Oroxylin A Glucoronide,千层纸素A-7-0-Β-D-葡萄糖醛酸苷,Oroxyloside,Oroxylin A 7-O-beta-D-glucuronide |
Others | Others |
Oroxylin A-7-O-glucuronide (Oroxylin A Glucoronide) 是一种类黄酮葡糖苷酸,提取自 Scutellaria baicalensis 干燥的根中,具有脯氨酰寡肽酶(POP)抑制作用。 |