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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7941 |
Imipramine hydrochloride
盐酸丙咪嗪,Imipramine (hydrochloride),Tofranil,G 22355,Imipramine HCl,Melipramine |
Serotonin Transporter | Neuroscience |
Imipramine hydrochloride (Imipramine HCl) 可抑制血清素转运蛋白,IC50=32 nM。它可阻止胰酶的易位,阻碍 MV 和外泌体的分泌。 | |||
T20025 |
Imipramine
Melipramine,HSDB3100,HSDB 3100,Dimipressin,HSDB-3100 |
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Imipramine is an agent of tricyclic antidepressants. | |||
T21364 |
Trimipramine
Stangyl,Rhotrimine,Surmontil |
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Trimipramine is an antidepressant with an anxiety-reducing sedative component to its action. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1045 |
Trimipramine maleate
Surmontil maleate,马来酸三甲丙咪嗪,三甲丙咪嗪马来酸盐 |
Dopamine Receptor; 5-HT Receptor; Antibacterial; Adrenergic Receptor; Norepinephrine; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience |
Trimipramine maleate (Surmontil maleate) 是一种 5-HT 受体拮抗剂,对 5-HT1C、5-HT2和 5-HT1A 受体的 pKi 值分别为 6.39、8.10和 4.66。 |