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Cat. No. | Product Name | Target | Signaling Pathways |
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T74513 |
RPR103611
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RPR103611,一个桦木酸衍生物,作为HIV-1入侵抑制剂表现出高效性,其对CCR5(热带)病毒YU2、CXCR4(热带)病毒NL4-3及双热带病毒89.6的IC50分别达到80、0.27和0.17。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2830 |
Betulinic acid
白桦脂酸,桦木酸,ALS-357,Lupatic acid,Betulic acid |
Apoptosis; Mitophagy; NF-κB; HIV Protease; Topoisomerase; Endogenous Metabolite; Aminopeptidase; Autophagy | Apoptosis; Autophagy; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome |
Betulinic acid (ALS-357) 是从白桦树皮中分离出来的一种五环三萜类天然产物,是真核细胞拓扑异构酶 I 的抑制剂,IC50值为 5 μM,具有抗逆转录病毒、抗疟疾、抗癌和抗炎特性。 | |||
TN1442 | Betulinic acid methyl ester | Antifection | Microbiology/Virology |
Betulinic acid methyl ester showed antiplasmodial activity against chloroquine-resistant Plasmodium falciparum parasites in vitro.It also inhibited B16 2F2 cell proliferation by induction of apoptosis. |