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2

抑制剂 & 化合物

11

天然产物

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Cat. No. Product Name Target Signaling Pathways
T82171 HS-291

ROS Kinase Tyrosine Kinase/Adaptors
HS-291是一种针对伯氏螺旋体(Bb) HtpG的抑制剂,组成包括具有高亲和力的BX-2819、PEG连接剂以及光活性毒素verteporfin。在光激活条件下,HS-291通过产生活性氧来氧化HtpG以及其邻近的伴侣蛋白和离散蛋白质子集,能够迅速并不可逆地灭活Bb。
T33363 Metochalcone

NSC 97905,Gebyl,NSC97905,Vesidril,NSC-97905

Metochalcone is a bioactive chemical.

化合物

HS-291
Cat.No: T82171
Synonym:
Target: ROS Kinase
Metochalcone
Cat.No: T33363
Synonym: NSC 97905,Gebyl,NSC97905,Vesidril,NSC-97905
Target:
Cat. No. Product Name Target Signaling Pathways
T3936 PATULIN

Expansin,Claviform,散毒素,Clavacin,棒曲霉素

Apoptosis; Others; Antibacterial; Antibiotic; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Others
Patulin (Claviform) 是由 Aspergillus、Penicillium 和 Byssochlamys 几种真菌属产生的霉菌毒素,有致染色体断裂、突变,致畸和细胞毒性作用。它通过溶酶体-线粒体轴诱导自噬依赖性细胞凋亡,能造成 DNA 损伤。
T35704 2-Methoxybenzaldehyde

o-Anisaldehyde

Antibacterial; Antifungal Microbiology/Virology
2-Methoxybenzaldehyde (o-Anisaldehyde) (o-Anisaldehyde), obtained from cinnamon essential oil (CEO), exhibits antibacterial and antifungal properties [1].
T7985 4,4'-Dimethoxychalcone

4,4'-甲氧基查耳酮,4,4'-二甲氧基查耳酮,4,4-Dimethoxychalcone

Others; Autophagy Autophagy; Others
4,4'-Dimethoxychalcone (4,4-Dimethoxychalcone) 是苏木中的一种查尔酮,是一种自噬诱导剂,具有抗衰老活性。
TN1860 Licoflavone B

甘草黄酮 B,甘草黄酮B

ATPase; Anti-infection; Parasite Membrane transporter/Ion channel; Microbiology/Virology
Licoflavone B 是从甘草中得到的一种类黄酮,抑制曼氏血吸虫 ATPase 和 ADPase 的活性,IC50值分别为 23.78 µM 和 31.50 µM。
TQ0188 Miquelianin

槲皮素-3-O-葡萄糖醛酸苷,Quercetin 3-glucuronide,Quercetin 3-O-glucuronide

stilbene oxidase; Endogenous Metabolite Metabolism
Miquelianin (Quercetin 3-glucuronide) 是槲皮素的代谢产物,属于类黄酮化合物。
TN1160 1,2,3,6-Tetragalloylglucose

1,2,3,6-Tetra-O-galloyl-β-D-glucose,1,2,3,6-四-O-没食子酰-Β-D-葡萄糖,TeGG

LDL; UGT Metabolism
1,2,3,6-Tetragalloylglucose (TeGG) 是 UDP-葡萄糖醛酸转移酶 1 家族成员,是多肽A1 的抑制剂(Ki:1.68 μM)。
TN6239 Caryatin

Caryatin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6239,CAS号为 1486-66-4。
TN4613 (-)-N-methylcoclaurine

N-Methylcoclaurine

Others Others
N-Methylcoclaurine shows binding affinities for the ĸ opioid receptor with the equilibrium dissociation constant (Ki) value of 0.9 ± 0.1 uM. N-methylcoclaurine also shows promising butyrylcholinesterase inhibition activities, with the IC50 value of 1
TN6383 (+)-Hannokinol

(+)-Hannokinol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6383,CAS号为 408324-76-5。
TN1919 (+)-Medioresinol

梣皮树脂醇,皮树脂醇,Medioresinol

Beta Amyloid; ROS; Antifection Immunology/Inflammation; Microbiology/Virology; Neuroscience
Medioresinol possesses antioxidative, a lesishmanicidal activity and cardiovascular disease risk reduction, it has antiamyloidogenic activity via reduction in the amount of α²-secretase, it is a potentially valuable antiamyloidogenic agent for the prevent
TN2928 Pygenic acid A

3-Epicorosolic acid,脓毒酸A

3-Epicorosolic acid has a potent inhibitory effect on Epstein-Barr virus early antigen (EBV-EA) induction, it has potential anti-inflammatory activities as well as cancer chemopreventive activity.3-Epicorosolic acid shows both potent α-glucosidase and pro

天然产物

PATULIN
Cat.No: T3936
Synonym: Expansin,Claviform,散毒素,Clavacin,棒曲霉素
Target: Apoptosis, Others, Antibacterial, Antibiotic, Autophagy
2-Methoxybenzaldehyde
Cat.No: T35704
Synonym: o-Anisaldehyde
Target: Antibacterial, Antifungal
4,4'-Dimethoxychalcone
Cat.No: T7985
Synonym: 4,4'-甲氧基查耳酮,4,4'-二甲氧基查耳酮,4,4-Dimethoxychalcone
Target: Others, Autophagy
Licoflavone B
Cat.No: TN1860
Synonym: 甘草黄酮 B,甘草黄酮B
Target: ATPase, Anti-infection, Parasite
Miquelianin
Cat.No: TQ0188
Synonym: 槲皮素-3-O-葡萄糖醛酸苷,Quercetin 3-glucuronide,Quercetin 3-O-glucuronide
Target: stilbene oxidase, Endogenous Metabolite
1,2,3,6-Tetragalloylglucose
Cat.No: TN1160
Synonym: 1,2,3,6-Tetra-O-galloyl-β-D-glucose,1,2,3,6-四-O-没食子酰-Β-D-葡萄糖,TeGG
Target: LDL, UGT
Caryatin
Cat.No: TN6239
Synonym:
Target:
(-)-N-methylcoclaurine
Cat.No: TN4613
Synonym: N-Methylcoclaurine
Target: Others
(+)-Hannokinol
Cat.No: TN6383
Synonym:
Target:
(+)-Medioresinol
Cat.No: TN1919
Synonym: 梣皮树脂醇,皮树脂醇,Medioresinol
Target: Beta Amyloid, ROS, Antifection
Pygenic acid A
Cat.No: TN2928
Synonym: 3-Epicorosolic acid,脓毒酸A
Target:
TargetMol Loading
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