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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6380 |
AMG 900
AMG900,AMG-900,莪术醇.姜黄醇 |
p38 MAPK; Tyrosine Kinases; Aurora Kinase | Cell Cycle/Checkpoint; Chromatin/Epigenetic; MAPK; Tyrosine Kinase/Adaptors |
AMG 900 是一种有效且高度选择性的泛极光激酶抑制剂,对Aurora A、B 和C 的IC50分别为 5 nM、4 nM 和 1 nM。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2853 |
Curcumol
莪术醇,(-)-Curcumol,姜黄醇 |
Apoptosis; JAK | Angiogenesis; Apoptosis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells |
Curcumol ((-)-Curcumol) 是一种倍半萜,具有抗癌,抗微生物,抗真菌,抗病毒和抗炎活性。它通过靶向关键信号通路,在许多癌细胞中有效地诱导凋亡。 | |||
T2840 |
Phloracetophenone
2,4,6-三羟基苯乙酮,2,4,6-trihydroxyacetophenone,1-(2,4,6-Trihydroxyphenyl)ethanone |
Others; P450; Antibacterial; Antibiotic | Metabolism; Microbiology/Virology; Others |
Phloracetophenone (1-(2,4,6-Trihydroxyphenyl)ethanone) 是多叶姜黄中苯乙酮糖苷的糖苷配基部分,具有抗肥胖,降血脂和降低胆固醇作用,能够增强胆固醇 7α-羟化酶的活性。 |