Cat. No. | Product Name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
T36848 | Combretastatin A-1
康普瑞汀A-1
|
109971-63-3 | 97.49% |
|
Combretastatin A-1 是一种有效的微管抑制剂,具有抗肿瘤和抗血管活性,通过微管蛋白解聚介导的 AKT 失活抑制 Wnt/β-catenin 通路发挥作用,可用于研究肝癌。 | ||||
T16997 | Tasidotin hydrochloride
化合物 T16997
|
623174-20-9 | 98% |
|
Tasidotin hydrochloride is a peptide analog of the antimitotic depsipeptide dolastatin 15. Tasidotin hydrochloride is an inhibitor of microtubule assembly and mi... | ||||
T17229 | Verubulin
化合物 T17229
|
827031-83-4 | 98% |
|
Verubulin is a microtubule-disrupting agent with potent and broad-spectrum in vitro and in vivo cytotoxic activities. | ||||
T6721 | Vinblastine
长春质碱
|
865-21-4 | 98% |
|
Vinblastine 抑制微管形成并抑制 nAChR 活性,IC50 为 8.9 μM,用于治疗某些类型的癌症。 | ||||
TQ0112 | Tubulysin A
化合物Tubulysin A
|
205304-86-5 | 98% |
|
Tubulysin A is a natural product from myxobacterial. It has many function in vitro assays, including anti-microtubule, anti-mitotic, an apoptosis inducer, antica... | ||||
T13227 | Tubulin inhibitor 1
化合物 T13227
|
2237054-53-2 | 98% |
|
Tubulin inhibitor 1 is an inhibitor of tubulin, inhibits tubulin polymerization, with potent anti-tumor activity, induces cellular apoptosis causes and cellular ... | ||||
T10428 | AZ82
化合物 T10428
|
1449578-65-7 | 98% |
|
AZ82 is a selective kinesin-like protein KIFC1 (HSET/KIFC1) inhibitor (Ki: 43 nM; IC50: 300 nM for KIFC1). | ||||
T10704 | CCB02
化合物CCB02
|
2100864-57-9 | 98% |
|
CCB02 是选择性的 CPAP-tubulin 相互作用抑制剂。CCB02能够与 tubulin 结合,竞争 β-tubulin 的 CPAP 结合位点,IC50 值为 689 nM,显示出高效的抗肿瘤活性。CCB02 对其他的蛋白没有抑制作用,包括中心体、细胞周期相关蛋白,对 Aurora A,Plk1,Plk2,C... | ||||
T11712 | Jasplakinolide
肌动蛋白多聚化肽
|
102396-24-7 | 98% |
|
Jasplakinolide(Jaspamide) 是一种来自海洋海绵 (marine sponge) 的天然环状肽,是一种有效的肌动蛋白聚合反应 (actin polymerization) 诱导剂。Jasplakinolide 具有抗真菌和抗肿瘤活性,可以稳定先前存在的肌动蛋白丝。Jasplakinolide 与鬼笔... | ||||
T12805 | S-methyl DM1
化合物 T12805
|
912569-84-7 | 98% |
|
S-methyl DM1 is a thiomethyl derivative of Maytansine. S-methyl DM1 binds to tubulin(Kd of 0.93 μM) and inhibts microtubule polymerization. | ||||
T12052 | Mivobulin
化合物 T12052
|
122332-18-7 | 98% |
|
Mivobulin is an inhibitor of tubulin . | ||||
T13901 | SS28
化合物 T13901
|
141172-08-9 | 98% |
|
SS28 inhibits tubulin polymerization to cause cell cycle arrest at G2/M phase. | ||||
T16543 | Pironetin
化合物 T16543
|
151519-02-7 | 98% |
|
Pironetin binds to α-tubulin and is an effective inhibitor of microtubule polymerization. It also has cell cycle arrest and antitumor activity. Pironetin is an α... | ||||
T6722 | Vinflunine Tartrate
长春氟宁酒石酸盐
|
1201898-17-0 | 98% |
|
Vinflunine Tartrate 是一种独特的新型长春花生物碱,具有抑制有丝分裂和微管蛋白相互作用活性的特性。 | ||||
T16387 | Ombrabulin
化合物 T16387
|
181816-48-8 | 98% |
|
Ombrabulin is a derivative of CA-4 phosphate. It is known to show antivascular effects through selective disruption of the tubulin cytoskeleton of endothelial ce... | ||||
T12823 | S516
化合物 T12823
|
1016543-77-3 | 98% |
|
S516 is an active CKD-516 metabolite and is a potent inhibitor of tubulin polymerization(IC50 of 4.29 μM), has marked antitumor activity. | ||||
TQ0202 | Epothilone D
埃博霉素
|
189453-10-9 | 98% |
|
Epothilone D (KOS 862) is an effective microtubule stabilizer. | ||||
T16386 | Ombrabulin hydrochloride
化合物 T16386
|
253426-24-3 | 98% |
|
Ombrabulin hydrochloride 是一种合成的、具有选择性的 CA-4 磷酸酯或 Ombrabulin 的衍生物,能破坏内皮细胞的微管蛋白细胞骨架,具有抗血管作用。Ombrabulin 是是一种微管蛋白聚合抑制剂,是 combretastatin a -4化合物类的一员,是一种水溶性的微管蛋白解聚肿瘤血管... | ||||
T13225 | Tubulin inhibitor 7
化合物 T13225
|
1309925-41-4 | 98% |
|
Tubulin inhibitor 7 is an inhibitor of tubulin and a potent inhibitor of multiple cancer cell lines (tubulin polymerization (IC50: 0.52 μM), K562 cell growth (IC... | ||||
TQ0141 | Taltobulin
化合物Taltobulin
|
228266-40-8 | 98% |
|
Taltobulin (HTI-286) is a potent tubulin inhibitor. |