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2

抑制剂 & 化合物

15

天然产物

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Cat. No. Product Name Target Signaling Pathways
T70277 Cynandione A

Others Others
Cynandione A 是从 Cynanchum wilfordii 中提取的苯乙酮,具有抗炎活性,可通过巨噬细胞 α7 nAChR 激活和随后的 IL-10 表达来显着减少促炎细胞因子的过表达。
T123808 Triptonoterpene

Triptonoterpene 是在 Tripterygium wilfordii 和 Tripterygium doianum 中发现的一种天然产物。Triptonoterpene 是一种双乙烷二萜。

化合物

Cynandione A
Cat.No: T70277
Synonym:
Target: Others
Triptonoterpene
Cat.No: T123808
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T5S1058 Triptonide

雷公藤内酯酮,PG 492,NSC 165677

Apoptosis; Wnt/beta-catenin; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; Stem Cells
Triptonide (PG 492) 是从雷公藤中鉴定出的一种天然产物,是一种 Wnt 信号抑制剂,其 IC50约为 0.3 nM。它具有免疫抑制、抗炎、避育、神经保护和抗淋巴瘤作用。
T3393 Triptophenolide

Hypolide,(+)-Triptophenolide,鼠尾草酸,雷酚内酯

Androgen Receptor Endocrinology/Hormones
Triptophenolide (Hypolide) 是一种无色晶体,从雷公藤的乙酸乙酯萃取部位分离得到。
T6S1049 Wilforine

ATPase Membrane transporter/Ion channel
Wilforine 是一倍半萜吡啶化合物,T. wilfordii 植物中的重要生物活性化合物,可有效治疗特发性肺纤维化。它具有抗炎和杀虫活性。
T3382 Wilforlide A

Abruslactone A,雷公藤内酯甲,3-Epiabruslactone A,Regelide

Tyrosinase Proteases/Proteasome
Wilforlide A (3-Epiabruslactone A) 是一种具有生物活性的三萜,从雷公藤中分离得到,具有抗炎和免疫抑制活性。
T3418 Demethylzeylasteral

去甲泽拉木醛,Demethylzeylasteral (T-96)

Apoptosis; UGT Apoptosis; Metabolism
Demethylzeylasteral (Demethylzeylasteral (T-96)) 分离自雷公藤,具有抗炎、免疫抑制和抗肿瘤活性。它通过阻断 TGF-β 信号通路,抑制三阴性乳腺癌的侵袭,它能显著减轻动脉粥样硬化。
TN5255 Wilforol A

Others Others
Wilforol A is a natural product from Tripterygium wilfordii Hook. f.
TN5185 Triptonodiol

Others Others
Triptonodiol is a natural product from Tripterygium wilfordii Hook.f.
T80940 Triptonoterpenol

Triptonoterpenol(化合物6)是雷公藤(Tripterygium wilfordii)的一种次级代谢产物。
TN5188 Triptoquinonide

Others Others
Triptoquinonide is a natural product from Tripterygium wilfordii.
T80941 Triptonoterpene Me ether

Triptonoterpene Me ether(compound 5)为一种从中药雷公藤(Tripterygium wilfordii Hook. f.)分离出的松香烷型二萜类化合物。
T80942 Triptonoditerpenic acid

Triptonoditerpenic acid 为一芳香族松香烷二萜类化合物,源自Tripterygium wilfordii。该化合物对HepG2、Hep3B 及 Bcap37细胞株展现细胞毒性作用,其IC50值依次为42.53 μM、29.74 μM 与37.63 μM。
TN5960 Polpunonic acid

Maytenonic acid,美登木酸,Maytenoic acid

Polpunonic acid is a natural product from Tripterygium wilfordii Hook.f.
T40252 Peritassine A

Peritassine A, an alkaloid derived from Tripterygium wilfordii Hook. f., exhibits anti-HIV properties.
T13936 Triptotriterpenic acid A

Maytenfolic acid,Abrusgenic acid

Others Others
Triptotriterpenic acid A is a natural product isolate from Tripterygium wilfordii.
T80938 Triptotriterpenic acid C

Triptotriterpenic acid C, 提取自雷公藤根部, 属于乌索酸类化合物。

天然产物

Triptonide
Cat.No: T5S1058
Synonym: 雷公藤内酯酮,PG 492,NSC 165677
Target: Apoptosis, Wnt/beta-catenin, Autophagy
Triptophenolide
Cat.No: T3393
Synonym: Hypolide,(+)-Triptophenolide,鼠尾草酸,雷酚内酯
Target: Androgen Receptor
Wilforine
Cat.No: T6S1049
Synonym:
Target: ATPase
Wilforlide A
Cat.No: T3382
Synonym: Abruslactone A,雷公藤内酯甲,3-Epiabruslactone A,Regelide
Target: Tyrosinase
Demethylzeylasteral
Cat.No: T3418
Synonym: 去甲泽拉木醛,Demethylzeylasteral (T-96)
Target: Apoptosis, UGT
Wilforol A
Cat.No: TN5255
Synonym:
Target: Others
Triptonodiol
Cat.No: TN5185
Synonym:
Target: Others
Triptonoterpenol
Cat.No: T80940
Synonym:
Target:
Triptoquinonide
Cat.No: TN5188
Synonym:
Target: Others
Triptonoterpene Me ether
Cat.No: T80941
Synonym:
Target:
Triptonoditerpenic acid
Cat.No: T80942
Synonym:
Target:
Polpunonic acid
Cat.No: TN5960
Synonym: Maytenonic acid,美登木酸,Maytenoic acid
Target:
Peritassine A
Cat.No: T40252
Synonym:
Target:
Triptotriterpenic acid A
Cat.No: T13936
Synonym: Maytenfolic acid,Abrusgenic acid
Target: Others
Triptotriterpenic acid C
Cat.No: T80938
Synonym:
Target:
TargetMol Loading
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