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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T70277 |
Cynandione A
|
Others | Others |
Cynandione A 是从 Cynanchum wilfordii 中提取的苯乙酮,具有抗炎活性,可通过巨噬细胞 α7 nAChR 激活和随后的 IL-10 表达来显着减少促炎细胞因子的过表达。 | |||
T123808 |
Triptonoterpene
|
||
Triptonoterpene 是在 Tripterygium wilfordii 和 Tripterygium doianum 中发现的一种天然产物。Triptonoterpene 是一种双乙烷二萜。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5S1058 |
Triptonide
雷公藤内酯酮,PG 492,NSC 165677 |
Apoptosis; Wnt/beta-catenin; Autophagy | Apoptosis; Autophagy; Cytoskeletal Signaling; Stem Cells |
Triptonide (PG 492) 是从雷公藤中鉴定出的一种天然产物,是一种 Wnt 信号抑制剂,其 IC50约为 0.3 nM。它具有免疫抑制、抗炎、避育、神经保护和抗淋巴瘤作用。 | |||
T3393 |
Triptophenolide
Hypolide,(+)-Triptophenolide,鼠尾草酸,雷酚内酯 |
Androgen Receptor | Endocrinology/Hormones |
Triptophenolide (Hypolide) 是一种无色晶体,从雷公藤的乙酸乙酯萃取部位分离得到。 | |||
T6S1049 |
Wilforine
|
ATPase | Membrane transporter/Ion channel |
Wilforine 是一倍半萜吡啶化合物,T. wilfordii 植物中的重要生物活性化合物,可有效治疗特发性肺纤维化。它具有抗炎和杀虫活性。 | |||
T3382 |
Wilforlide A
Abruslactone A,雷公藤内酯甲,3-Epiabruslactone A,Regelide |
Tyrosinase | Proteases/Proteasome |
Wilforlide A (3-Epiabruslactone A) 是一种具有生物活性的三萜,从雷公藤中分离得到,具有抗炎和免疫抑制活性。 | |||
T3418 |
Demethylzeylasteral
去甲泽拉木醛,Demethylzeylasteral (T-96) |
Apoptosis; UGT | Apoptosis; Metabolism |
Demethylzeylasteral (Demethylzeylasteral (T-96)) 分离自雷公藤,具有抗炎、免疫抑制和抗肿瘤活性。它通过阻断 TGF-β 信号通路,抑制三阴性乳腺癌的侵袭,它能显著减轻动脉粥样硬化。 | |||
TN5255 |
Wilforol A
|
Others | Others |
Wilforol A is a natural product from Tripterygium wilfordii Hook. f. | |||
TN5185 | Triptonodiol | Others | Others |
Triptonodiol is a natural product from Tripterygium wilfordii Hook.f. | |||
T80940 |
Triptonoterpenol
|
||
Triptonoterpenol(化合物6)是雷公藤(Tripterygium wilfordii)的一种次级代谢产物。 | |||
TN5188 |
Triptoquinonide
|
Others | Others |
Triptoquinonide is a natural product from Tripterygium wilfordii. | |||
T80941 | Triptonoterpene Me ether | ||
Triptonoterpene Me ether(compound 5)为一种从中药雷公藤(Tripterygium wilfordii Hook. f.)分离出的松香烷型二萜类化合物。 | |||
T80942 |
Triptonoditerpenic acid
|
||
Triptonoditerpenic acid 为一芳香族松香烷二萜类化合物,源自Tripterygium wilfordii。该化合物对HepG2、Hep3B 及 Bcap37细胞株展现细胞毒性作用,其IC50值依次为42.53 μM、29.74 μM 与37.63 μM。 | |||
TN5960 |
Polpunonic acid
Maytenonic acid,美登木酸,Maytenoic acid |
||
Polpunonic acid is a natural product from Tripterygium wilfordii Hook.f. | |||
T40252 |
Peritassine A
|
||
Peritassine A, an alkaloid derived from Tripterygium wilfordii Hook. f., exhibits anti-HIV properties. | |||
T13936 |
Triptotriterpenic acid A
Maytenfolic acid,Abrusgenic acid |
Others | Others |
Triptotriterpenic acid A is a natural product isolate from Tripterygium wilfordii. | |||
T80938 |
Triptotriterpenic acid C
|
||
Triptotriterpenic acid C, 提取自雷公藤根部, 属于乌索酸类化合物。 |