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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T3578L Pyridoxal calcium phosphate

Pyridoxal phosphate (PLP, pyridoxal 5'-phosphate, P5P), known as an active form of vitamin B6, is a coenzyme involved in many enzymatic reactions.
T75316 Pyridoxamine 5′-phosphate

Pyridoxamine 5′-phosphate 是维生素 B6 与磷酸结合的活性形式。Pyridoxamine 5′-phosphatePyridoxal 5'-phosphate hydrate 的胺化形式,是多种酶的中心代谢物、强力抗氧化剂、维生素 B6 和酶底物的辅助因子。Pyridoxamine 5′-phosphate 能与 Pyridoxal 5'-phosphate hydrate 相互转化。
T38294 4-Deoxypyridoxine hydrochloride

S1P Receptor GPCR/G Protein
4-Deoxypyridoxine hydrochloride 通过抑制 S1P 裂解酶 (SPL) 活性来抑制细胞内 S1P 的降解,与 S1P 一样,减少化学诱导的胰岛素瘤细胞系的细胞凋亡。
T73614 Tyrosine decarboxylase

Tyrosine decarboxylase (TDC; TyrDC),即酪氨酸脱羧酶,广泛存在于植物、昆虫和不同微生物中,常用于生化研究。Tyrosine decarboxylase 是一种5'-磷酸吡哆醛 (PLP) 依赖性脱羧酶,可以催化酪氨酸中羧基的去除,产生酪胺和二氧化碳。
T79929 L-Methionine γ-lyase

Methionine lyase

L-Methionine γ-lyase(Methionine lyase)是一种依赖磷酸吡哆醛的多功能酶,专门催化L-蛋氨酸(L-methionine)及其类似物的α, γ-裂解反应。该酶因其抗癌和抗感染活性被用于相关疾病的研究,同时也适用于同型半胱氨酸血症研究领域。

化合物

Pyridoxal calcium phosphate
Cat.No: T3578L
Synonym:
Target:
Pyridoxamine 5′-phosphate
Cat.No: T75316
Synonym:
Target:
4-Deoxypyridoxine hydrochloride
Cat.No: T38294
Synonym:
Target: S1P Receptor
Tyrosine decarboxylase
Cat.No: T73614
Synonym:
Target:
L-Methionine γ-lyase
Cat.No: T79929
Synonym: Methionine lyase
Target:
Cat. No. Product Name Target Signaling Pathways
T8083 Pyridoxal 5'-​phosphate monohydrate

Pyridoxal phosphate monohydrate,Pyridoxal 5-phosphate monohydrate,5-磷酸吡哆醛

Others Others
Pyridoxal 5'-​phosphate monohydrate 是维生素 B6的活性形式,也是多种酶的重要辅因子。它是维生素 B6 在细胞内磷酸化过程中重要的辅酶变异体,能够与其他变异体(如 PNP 、 PMP)发生互换。
T5085 Pyridoxal 5'-phosphate hydrate

Codecarboxylase,Pyridoxal 5'-phosphate hydrate(1:x),5-磷酸吡多醛水合物,PLP,Pyridoxal 5'-phosphate hydrate

Others; Endogenous Metabolite Metabolism; Others
Pyridoxal 5'-phosphate hydrate (PLP) 是内源性代谢产物的一种。
T3578 Pyridoxal phosphate

PLP,PAL-P,磷酸吡哆醛,pyridoxal 5'-phosphate,Pyridoxyl phosphate,Pyridoxal 5′-phosphate,Vitamin B6 phosphate

Reverse Transcriptase; Endogenous Metabolite Metabolism; Microbiology/Virology
Pyridoxal phosphate (Vitamin B6 phosphate) 是维生素 B6 的活性形式,可抑制逆转录酶活性,用于研究迟发性运动障碍症。
T0710 L-Cycloserine

Levcycloserine,Levcicloserina,(-)-Cycloserine,(S)-Cycloserine,Levcycloserinum,环丝氨酸,(S)-4-Amino-3-isoxazolidone

HIV Protease; GABA Receptor Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; Proteases/Proteasome
L-Cycloserine ((-)-Cycloserine) 不可逆地抑制大肠杆菌以及各种动物大脑中的 GABA 吡哆醛 5'-磷酸依赖性转氨酶,导致体内抑制性神经递质 γ-氨基丁酸水平升高。
T0973 Pyridoxine

吡哆醇,Pyridoxol,Vitamin B6,Gravidox,吡多素(维生素B6)

PLK; Nrf2; Endogenous Metabolite Cell Cycle/Checkpoint; Immunology/Inflammation; Metabolism
Pyridoxine (Vitamin B6) 是一种吡啶衍生物,通过 Nrf-2/HO-1 途径发挥抗氧化作用,作用于阿尔茨海默病细胞模型。

天然产物

Pyridoxal 5'-​phosphate monohydrate
Cat.No: T8083
Synonym: Pyridoxal phosphate monohydrate,Pyridoxal 5-phosphate monohydrate,5-磷酸吡哆醛
Target: Others
Pyridoxal 5'-phosphate hydrate
Cat.No: T5085
Synonym: Codecarboxylase,Pyridoxal 5'-phosphate hydrate(1:x),5-磷酸吡多醛水合物,PLP,Pyridoxal 5'-phosphate hydrate
Target: Others, Endogenous Metabolite
Pyridoxal phosphate
Cat.No: T3578
Synonym: PLP,PAL-P,磷酸吡哆醛,pyridoxal 5'-phosphate,Pyridoxyl phosphate,Pyridoxal 5′-phosphate,Vitamin B6 phosphate
Target: Reverse Transcriptase, Endogenous Metabolite
L-Cycloserine
Cat.No: T0710
Synonym: Levcycloserine,Levcicloserina,(-)-Cycloserine,(S)-Cycloserine,Levcycloserinum,环丝氨酸,(S)-4-Amino-3-isoxazolidone
Target: HIV Protease, GABA Receptor
Pyridoxine
Cat.No: T0973
Synonym: 吡哆醇,Pyridoxol,Vitamin B6,Gravidox,吡多素(维生素B6)
Target: PLK, Nrf2, Endogenous Metabolite
TargetMol Loading
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