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6

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T0188 Fluticasone (propionate)

丙酸氟替卡松,CCI-187881,氟替卡松丙酸酯,Fluticasone propionate

Glucocorticoid Receptor; Virus Protease; Estrogen/progestogen Receptor; Phospholipase; Endogenous Metabolite Endocrinology/Hormones; Metabolism; Microbiology/Virology
Fluticasone propionate (CCI-187881) 是一种选择性糖皮质激素受体激动剂,是一种局部抗炎激素,亲和力KD 为 0.5 nM。具有抗病毒活性。
T20663 Oxyfluorfen

Goldate,乙氧氟草醚,Galigan,RH-2915,RH 2915,Boxer,Koltar

Others Others
Oxyfluorfen (Boxer) 是一种硝基二苯醚类除草剂,用于控制各种大田作物中的一年生和多年生阔叶杂草和莎草。
T30898 Chloropon

Omnidel,TCP

Chloropon is a herbicide that controls annnual & perennial grasses including couch and foxtails.
T32851 Lolitrem B

Lolitrem B is one of many toxins produced by a fungus called Epichloë festucae (var. lolii), which grows in perennial ryegrass. The fungus is symbiotic with the ryegrass; it doesn't harm the plant, and the toxins it produces kill insects that feed on ryeg
T62654 Fluocortin butyl ester

Fluocortin butyl ester 是一种发达的皮质类固醇化合物,局部使用时无法检测到全身性的皮质类固醇活性。Fluocortin butyl ester 似乎是一种有效的、耐受性良好的局部类固醇,能够用于常年性鼻炎的研究。
T31194 Dalapon

Basfapon B,Dowpon M,Dawpon-Rae

Dalapon is a selective herbicide used to control perennial grasses. The major use of dalapon is on food crops including sugarcane and sugar beets. Its use is no longer authorized in France. The National Institute for Occupational Safety and Health in the

化合物

Fluticasone (propionate)
Cat.No: T0188
Synonym: 丙酸氟替卡松,CCI-187881,氟替卡松丙酸酯,Fluticasone propionate
Target: Glucocorticoid Receptor, Virus Protease, Estrogen/progestogen Receptor, Phospholipase, Endogenous Metabolite
Oxyfluorfen
Cat.No: T20663
Synonym: Goldate,乙氧氟草醚,Galigan,RH-2915,RH 2915,Boxer,Koltar
Target: Others
Chloropon
Cat.No: T30898
Synonym: Omnidel,TCP
Target:
Lolitrem B
Cat.No: T32851
Synonym:
Target:
Fluocortin butyl ester
Cat.No: T62654
Synonym:
Target:
Dalapon
Cat.No: T31194
Synonym: Basfapon B,Dowpon M,Dawpon-Rae
Target:
Cat. No. Product Name Target Signaling Pathways
T8203 Gentianose

Others Others
Gentianose 是一种碳水化合储备物,来源于多年生黄龙胆贮藏根中。
T3149 Salvianolic Acid C

丹酚酸C,丹酚酸 C

Others; P450 Metabolism; Others
Salvianolic acid C 是一种细胞色素 P4502C8(CYP2C8)的非竞争性抑制剂及细胞色素 P4502J2(CYP2J2)中等强度的混合抑制剂,对 CYP2C8 和 CYP2J2 的 Ki 分别为 4.82 μM 和 5.75 μM。

天然产物

Gentianose
Cat.No: T8203
Synonym:
Target: Others
Salvianolic Acid C
Cat.No: T3149
Synonym: 丹酚酸C,丹酚酸 C
Target: Others, P450
TargetMol Loading
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