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Cat. No. Product Name Target Signaling Pathways
T9223 RO-0335

Reverse Transcriptase Microbiology/Virology
RO-0335 是新高效二苯醚非核苷逆转录酶抑制剂。它 (IC50= 1.1 nM) 可以抑制Wt HIV-1病毒,对 92% 的 NNRTI 耐药临床分离株具有保留活性 (IC50<100 nM)。
TQ0122L VCH-916 free acid(1200133-34-1 free base)

HCV Protease Microbiology/Virology; Proteases/Proteasome
VCH-916 free acid(1200133-34-1 free base) 是一种新型非核苷 HCV NS5B 聚合酶抑制剂。
T27260 Emivirine

MKC442,MKC-442,MKC 442,DRG-0302,DRG 0302,DRG0302

HIV Protease Microbiology/Virology; Proteases/Proteasome
Emivirine (MKC-442) 是一种有效和选择性的人类免疫缺陷病毒1型(HIV-1)的非核苷逆转录酶抑制剂。
T12715 Reverse transcriptase-IN-1

HIV Protease Microbiology/Virology; Proteases/Proteasome
Reverse transcriptase-IN-1 是一种二芳基苯并嘧啶类似物,是一种有效的 HIV-1 非核苷类逆转录酶抑制剂,IC50 为 13.7 nM。
T8800 NSAH

2-hydroxy-N'-[(E)-(2-hydroxynaphthalen-1-yl)methylidene]benzohydrazide

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
NSAH (2-hydroxy-N'-[(E)-(2-hydroxynaphthalen-1-yl)methylidene]benzohydrazide) 是一种可逆竞争性非核苷类的核苷酸还原酶抑制剂,无细胞 IC50 为 32 μM,基于细胞的 IC50 约为 250 nM。
T25363 Efavirenz, (R)-

L 743725,L-743725,L743725

Efavirenz, (R)- is an antiviral agent and a nonnucleoside HIV-1 reverse transcriptase inhibitor.
TQ0122 VCH-916

HCV Protease Microbiology/Virology; Proteases/Proteasome
VCH-916 是一种新型非核苷类 HCV NS5B 聚合酶抑制剂。
T14086 ABT-072

Others Others
ABT-072 is a nonnucleoside NS5B polymerase inhibitor and a candidate drug evaluated for treatment of hepatitis C virus.
T26442 A 75925

A-75925,A75925

A 75925, a nonnucleoside reverse transcriptase inhibitors (NNRTI), works to inhibit HIV-1 replication.
T24794 SJ-3366

SJ 3366

SJ3366 is a unique and highly potent nonnucleoside reverse transcriptase human immunodeficiency virus type 1 and HIV-2 inhibitor.
T70212 U 95133

U 95133 is a potent, broad-spectrum nonnucleoside reverse transcriptase inhibitor of drug-resistant isolates of human immunodeficiency virus type 1.
T31085 CP-94707

UNII-YGC6408B5O

CP-94707 is a new inhibitor of nonnucleoside reverse transcriptase (NNRTI).
T27442 GSK 224876

GSK-224876,GSK224876

GSK 224876 is a novel next-generation nonnucleoside reverse transcriptase inhibitor (NNRTI). It has activity against efavirenz-resistant strains in the treatment of treatment-naive HIV-1-infected subjects.
T30185 AT 61

AT61,AT-61

AT-61 is a nonnucleoside analogue inhibitor of hepatitis B virus (HBV) replication.
T16081 MIV-150

PC 815

Others Others
MIV-150 is a nonnucleoside inhibitor of reverse transcriptase (NNRT). MIV-150 also blocking HIV-1 and HIV-2 infections (EC50<1 nM against HIV-1/HIV-2MN).
T78167 PYR01

PYR01为一种高效的HIV-1非核苷逆转录酶抑制剂,同时作为针对消除表达HIV-1细胞的细胞杀伤分子的靶向激活剂。
T72283 (+)-Dihydrocalanolide A

NSC 678323,DHCal A ; NSC 678323,DHCal A

(+)-Dihydrocalanolide A (DHCal A ; NSC 678323) 是一种口服有效、非核苷的逆转录酶 (Reverse Transcriptase) 抑制剂。(+)-Dihydrocalanolide A 可用于 HIV

化合物

RO-0335
Cat.No: T9223
Synonym:
Target: Reverse Transcriptase
VCH-916 free acid(1200133-34-1 free base)
Cat.No: TQ0122L
Synonym:
Target: HCV Protease
Emivirine
Cat.No: T27260
Synonym: MKC442,MKC-442,MKC 442,DRG-0302,DRG 0302,DRG0302
Target: HIV Protease
Reverse transcriptase-IN-1
Cat.No: T12715
Synonym:
Target: HIV Protease
NSAH
Cat.No: T8800
Synonym: 2-hydroxy-N'-[(E)-(2-hydroxynaphthalen-1-yl)methylidene]benzohydrazide
Target: DNA/RNA Synthesis
Efavirenz, (R)-
Cat.No: T25363
Synonym: L 743725,L-743725,L743725
Target:
VCH-916
Cat.No: TQ0122
Synonym:
Target: HCV Protease
ABT-072
Cat.No: T14086
Synonym:
Target: Others
A 75925
Cat.No: T26442
Synonym: A-75925,A75925
Target:
SJ-3366
Cat.No: T24794
Synonym: SJ 3366
Target:
U 95133
Cat.No: T70212
Synonym:
Target:
CP-94707
Cat.No: T31085
Synonym: UNII-YGC6408B5O
Target:
GSK 224876
Cat.No: T27442
Synonym: GSK-224876,GSK224876
Target:
AT 61
Cat.No: T30185
Synonym: AT61,AT-61
Target:
MIV-150
Cat.No: T16081
Synonym: PC 815
Target: Others
PYR01
Cat.No: T78167
Synonym:
Target:
(+)-Dihydrocalanolide A
Cat.No: T72283
Synonym: NSC 678323,DHCal A ; NSC 678323,DHCal A
Target:
TargetMol Loading
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