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3

抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T2451 GlyH-101

GlyH 101

CFTR; Autophagy Autophagy; Membrane transporter/Ion channel
GlyH-101 是一种可渗透入细胞的 CFTR 阻断剂,Ki 为1.4 uM。
T81539 PAT1inh-B01

PAT1inh-B01为选择性SLC26A6抑制剂,抑制PAT1(Cl-/HCO3-交换器)介导的阴离子交换(IC50: 350 nM),并阻断小肠液体吸收,适用于小肠分泌不足相关疾病研究。
T71303 Flufenamic Acid-d4

Flufenamic acid-d4 is intended for use as an internal standard for the quantification of flufenamic acid by GC- or LC-MS. Flufenamic acid is a non-steroidal anti-inflammatory drug (NSAID) and COX inhibitor (IC50s = 3 and 9.3 µM for human COX-1 and COX-2, respectively). Flufenamic acid inhibits TNF-α-induced increases in COX-2 levels and NF-κB activation in HT-29 colon cancer cells in a concentration-dependent manner. It inhibits calcium influx induced by fMLP or A23187 in human polymorphonuclear...

化合物

GlyH-101
Cat.No: T2451
Synonym: GlyH 101
Target: CFTR, Autophagy
PAT1inh-B01
Cat.No: T81539
Synonym:
Target:
Flufenamic Acid-d4
Cat.No: T71303
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN5147 Tilifodiolide

IL Receptor; TNF; GABA Receptor Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience
Tilifodiolide exerts in vitro and in vivo anti-inflammatory activity and in vivo antinociceptive effects. Tilifodiolide exerted antidiarrheal activity by decreasing the intestinal fluid accumulation and vasorelaxant effects mediated by nitric oxide and cyclic guanosine monophosphate, it also showed anxiolytic and antidepressant effects by the partial involvement of gamma-Aminobutyric acid (GABA) receptors and the possible participation of α2-adrenoreceptors, respectively.

天然产物

Tilifodiolide
Cat.No: TN5147
Synonym:
Target: IL Receptor, TNF, GABA Receptor
TargetMol Loading
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