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Search Results for " insulin sensitization "

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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T21955 GQ-16

PPAR DNA Damage/DNA Repair; Metabolism
GQ-16 是 PPARγ 的部分激动剂,Ki 为 160 nM。 GQ-16 可减少脂肪生成作用并促进胰岛素敏化而不会增加体重。
T72947 JBSNF-000028

JBSNF-000028 free base

Others Others
JBSNF-000028 是一种具有口服活性和有效性的烟酰胺 N-甲基转移酶 (NNMT) 抑制剂,对人 NNMT (hNNMT)、猴 NNMT (mkNNMT) 和小鼠 NNMT (mNNMT) 具有抑制作用, IC50 分别为 0.033 μM、0.19 μM 和 0.21 μM。JBSNF-000028 可驱动胰岛素敏化、葡萄糖调节和体重减,可用于研究代谢紊乱。

化合物

GQ-16
Cat.No: T21955
Synonym:
Target: PPAR
JBSNF-000028
Cat.No: T72947
Synonym: JBSNF-000028 free base
Target: Others
Cat. No. Product Name Target Signaling Pathways
TN4584 Morolic acid

IL Receptor; COX; HIV Protease Immunology/Inflammation; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Morolic acid and moronic acid have shown sustained antidiabetic and antihyperglycemic action possibly mediated by an insulin sensitization with consequent changes of glucose, cholesterol and triglycerides, in part mediated by inhibition of 11β-HSD 1. Moro
TN4585 Moronic acid

HIV Protease; Antifection; HSV Microbiology/Virology; Proteases/Proteasome
Moronic acid shows oral therapeutic efficacy in HSV-infected mice and possessed novel anti-HSV activity. It also shows significant anti-HIV activity (EC(50) 186) and was modified to develop more potent anti-AIDS agents. Moronic acid is a new structural lead for anti-EBV drug development, can substantially reduce the numbers of EBV particles produced by the cells after lytic induction. Morolic and moronic acids have shown sustained antidiabetic and antihyperglycemic action possibly mediated by an...

天然产物

Morolic acid
Cat.No: TN4584
Synonym:
Target: IL Receptor, COX, HIV Protease
Moronic acid
Cat.No: TN4585
Synonym:
Target: HIV Protease, Antifection, HSV
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