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Search Results for " histone acetyltransferases "

4

抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T8778 TTK21

Epigenetic Reader Domain Chromatin/Epigenetic
TTK21 是 CBP/p300 组蛋白乙酰转移酶活性的激活剂,与葡萄糖基碳纳米球结合时,可通过血脑屏障,对成人大脑神经发生和长期记忆功能有益。
T4362 WM-8014

MOZ-IN-3

Histone Acetyltransferase Chromatin/Epigenetic
WM-8014 (MOZ-IN-3) 是一种 MOZ,属于组蛋白乙酰转移酶的抑制剂,IC50值为 55 nM。
T10901 Curcumin-d6

Turmeric yellow D6,Natural Yellow 3 D6,Curcumin D6,Diferuloylmethane D6

Others Others
Curcumin D6 (difluoroformylmethane D6) is deuterium-labeled curcumin (Turmeric yellow). Curcumin (Turmeric yellow) is a natural phenolic compound with various pharmacological effects, including anti-inflammatory, antioxidant, anti-proliferative and anti-a
T36626 Lys-CoA

Selective p300 histone acetyltransferase (HAT) inhibitor (IC50 = 50-500 nM). Exhibits approximately 100-fold selectivity for p300 over PCAF (IC50 = 200 μM). Inhibits p300-dependent transcription. Active in vivo. Lau et al (2000) HATs off: selective synthetic inhibitors of the histone acetyltransferases p300 and PCAF. Mol.Cell. 5 589 PMID:10882143 |Liu et al (2008) The structural basis of protein acetylation by the p300/CBP transcriptional coactivator. Nature. 451 846 PMID:18273021 |Burns et al (...

化合物

TTK21
Cat.No: T8778
Synonym:
Target: Epigenetic Reader Domain
WM-8014
Cat.No: T4362
Synonym: MOZ-IN-3
Target: Histone Acetyltransferase
Curcumin-d6
Cat.No: T10901
Synonym: Turmeric yellow D6,Natural Yellow 3 D6,Curcumin D6,Diferuloylmethane D6
Target: Others
Lys-CoA
Cat.No: T36626
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T11366 Garcinol

Apoptosis; Endogenous Metabolite; Histone Acetyltransferase; AChR; AChE Apoptosis; Chromatin/Epigenetic; Metabolism; Neuroscience
Garcinol 是一种从印度藤黄提取的聚异戊二烯基二苯甲酮,对乙酰胆碱酯酶和丁酰胆碱酯酶具有抗胆碱酯酶的特性,IC50分别为 0.66 µM 和 7.39 µM。它还抑制组蛋白乙酰转移酶和 p300/CPB 相关因子,具有抗炎和抗癌活性。

天然产物

Garcinol
Cat.No: T11366
Synonym:
Target: Apoptosis, Endogenous Metabolite, Histone Acetyltransferase, AChR, AChE
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