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Search Results for " heptapeptide "

31

抑制剂 & 化合物

3

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T83201	Acetyl heptapeptide-4
	Acetyl heptapeptide-4，一种抗过敏(antiallergic)生物活性肽，已报道作为化妆品成分使用。
T83198	Acetyl sh-heptapeptide-1
	Acetyl sh-heptapeptide-1，一种多肽，有效对抗面部老化。
T7748	Dermorphin TFA 皮啡肽三氟乙酸盐	Others; Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience; Others
	Dermorphin TFA 是在两栖类皮肤中发现的天然七肽，是 μ-阿片受体激动剂，可用于抑制神经痛。
T7404	Dermorphin 皮啡肽	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	Dermorphin 是在两栖类皮肤中发现的天然七肽，是 μ-阿片受体激动剂，可用于抑制神经痛。
TP1351L	Kemptide TFA	Others	Others
	Kemptide TFA (65189-71-1 free base) 是一种合成七肽，可作为 cAMP 依赖性蛋白激酶 (PK) 的底物。
T8455	Spinorphin	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	Spinorphin 是一种脑非肽降解酶抑制剂，能够抑制氨基肽酶、二肽基氨基肽酶III、血管紧张素转换酶和脑非肽酶。它可用于研究疼痛的缓解。
T5146	Eptifibatide acetate (148031-34-9 free base) Eptifibatide acetate,依菲巴特醋酸盐	Others	Others
	Eptifibatide acetate (148031-34-9 free base) (Eptifibatide acetate) 是一种糖蛋白 IIb/IIIa 抑制剂类的抗血小板药物，是一种由 6 个氨基酸和一个巯基丙酰基残基构成的环状七肽。
T7339	Angiotensin (1-7) Ang-(1-7),Angiotensin 1-7,ASP-ARG-VAL-TYR-ILE-HIS-PRO	RAAS; Endogenous Metabolite	Endocrinology/Hormones; Metabolism
	Angiotensin (1-7) (ASP-ARG-VAL-TYR-ILE-HIS-PRO) 是肾素-血管紧张素系统中的内源性七肽。Angiotensin 1-7在心肌细胞中具有抗炎和抗纤维化活性，因此具有心脏保护作用。它能抑制血管紧张素转换酶和释放一氧化氮，是激肽诱导的血管舒张的局部协同调节剂。它阻断 Ang II 诱导的平滑肌细胞增殖和肥大，并显示对内皮的抗血管生成和生长抑制作用。它显示出抗炎活性。
TP1351	Kemptide 肯普肽	PKA	Tyrosine Kinase/Adaptors
	Kemptide 是一种 cAMP 依赖性蛋白激酶的特异性底物，是一种合成的七肽。
T30872	CHEC-7 CHEC7
	CHEC-7 is a neuroprotective cyclic heptapeptide.
T25480	H 256 H-256,H256,Pro-thr-glu-phe-CH2NH-phe-arg-glu
	H 256 is a pepsin heptapeptide inhibitor.
T24474	MK 0852 MK-0852,L-367,073,MK0852,L 367,073,L367,073
	MK 0852 is the platelet GP IIb/IIIa cyclic heptapeptide antagonist.
T31133	Cyclo-cadagac Cyclo cadagac
	Cyclo-cadagac is a cyclic heptapeptide.
T70418	TLN-232
	TLN-232, also known as CAP-232, is a synthetic cyclic heptapeptide with potential antineoplastic activity. Pyruvate kinase (PK) inhibitor TLN-232 targets pyruvate kinase M2 (M2PK), which may disrupt tumor cell anaerobic glycolysis. M2PK is a dimeric isoform of PK and the predominant PK isoform found in tumor cells.
T32408	KNI 122 Ser-Phe-Asn-Pns-Pro-Ile-Val-NH2,KNI-122,KNI122
	KNI 122is a heptapeptide analog.
TP2343	Lagatide
	Lagatide is a synthetic heptapeptide that has antisecretory activity.
T24203	Jmv 170 Jmv-170,Jmv170
	Jmv 170 is the C-terminal heptapeptide of cholecystokinin. It has partial agonist CCK activity on pancreatic amylase release.
T25507	HP 228 HP-228,Ac-Nle-gln-his-D-phe-arg-D-trp-gly-NH2,HP228
	HP 228 is a heptapeptide by inhibits the induction of nitric oxide synthase.
T38191	Unguisin B
	Unguisin B is a cyclic heptapeptide originally isolated from the marine fungus E. unguis whose structure is comprised of amino acids and GABA.
TP1331	Super-TDU (1-31) TFA
	Super-tdu (1-31) TFA is an endogenous ligand of heptapeptide receptor and has a strong anti-analgesic effect.
T71935	WIN 66306
	WIN 66306 is a cyclic heptapeptide antagonist of neurokinin-1 (NK1) and NK2 receptors originally isolated from A. flavipes. It binds to NK1 and NK2 receptors and inhibits contractions induced by substance P in isolated guinea pig ileum in a concentration-dependent manner.
T76454	Substance P (5-11)
	Substance P (5-11) 是 Substance P (Substance P ) 的 C 端七肽，是一种神经肽，可以与NK-1速激肽受体结合。
TP1261	Alexamorelin Met 1 (D-Mrp)-Ala-Trp-(D-Phe)
	Alexamorelin Met 1 is one of the metabolites of alexamorelin. The heptapeptide Ala-His-D-2-methyl-Trp-Ala-Trp-D-Phe-Lys-NH2 (Alexamorelin) is a synthetic molecule which inhibits growth hormone secretagogue binding in vitro.
TP1870	Dermorphin Analog
	Dermorphin Analog is an analog of Dermorphin. Dermorphin is a natural heptapeptide μ-opioid receptor agonist found in amphibian skin. The dermorphin-derived peptide [Dmt1] dermorphin analog labels m-opioid receptors with high affinity and selectivity in r
T76354	LH-RH (4-10)
	LH-RH (4-10)，一种性腺激素释放激素(LHRH)的主要降解产物，属于七肽类，主要在巨噬细胞和II型肺细胞中产生。
T5020	Eptifibatide Eptifibatide Acetate,Mpr-Har-Gly-Asp-Trp-Pro-Cys-NH2,依替巴肽	Others	Others
	Eptifibatide (Eptifibatide Acetate) 是一种糖蛋白 IIb/IIIa 抑制剂类的抗血小板药物，是一种由 6 个氨基酸和一个巯基丙酰基残基构成的环状七肽。
T36471	Ternatin
	Ternatin is a cyclic heptapeptide first isolated from the mushroom C. versicolor that has been shown to have cytotoxic and anti-adipogenic effects in vitro. It inhibits adipogenesis with an IC50 value of 27 nM and becomes cytotoxic to 3T3-L1 mouse adipocytes at 10-fold higher concentrations. Ternatin is reported to inhibit HCT116 cell proliferation with an IC50 value of 71 nM. Note that this metabolite should not be confused with the plant flavonoid of the same name.
T83734	PapRIV TFA
	PapRIV是最初从B. cereus分离出的一种群体感应七肽。它被转译为一个48-氨基酸多肽，由NprB蛋白酶在细胞外分泌和加工形成活性七肽。PapRIV（1-25 µM）在BV-2微胶质细胞中诱导IL-6和TNF-α的产生，并促使NF-κB转移。
T37496	Alamandine
	Alamandine can be formed from angiotensin A by action of ACE-2 or directly from angiotensin-(1-7) by decarboxylation of its aspartate residue. The angiotensin A analog produces effects resembling those of Ang II (1-7). However, it acts independently of the two known vasodilators receptors of the RAS (Mas and angiotensin II type 2). To produce its effects, alamandine binds to the Mas-related receptor, MrgD. A novel orally active formulation of alamandine produced a long-term antihypertensive effe...
T37495	Angiotensin (1-7) (acetate)
	Angiotensin 1-7 (Ang-(1-7)) acetate 是RAS中的一种内源性七肽，具备心脏保护作用，主要表现为对心肌细胞的抗炎与抗纤维化活性。该化合物能抑制纯化的犬ACE活性（IC50=0.65 μM），通过降低ACE活性并促进一氧化氮释放，作为血管舒张调节的局部协同因子。此外，Angiotensin 1-7 acetate 可阻止血管紧张素Ⅱ诱发的平滑肌细胞增殖和肥大，同时对内皮细胞表现出抗血管生成和生长抑制作用。
T83122	Amyloid-Forming peptide GNNQQNY
	Amyloid-Forming peptide GNNQQNY是由酵母蛋白Sup35的N-末端朊病毒决定结构域中得来的七肽段，具有生物活性，并能形成淀粉样纤维。它的详细原子低聚结构之研究，使其成为揭示早期聚集阶段的理想模型。GNNQQNY二聚体以三种稳定构形存在：寄存器内并排、寄存器外并排和反向并排。对准的平行二聚体其β-pleated sheet结构中肽链间氢键较少，强调了疏水作用的重要性，相较于反向并排结构有更高的构象熵。

化合物

Acetyl heptapeptide-4

Cat.No: T83201

Acetyl sh-heptapeptide-1

Cat.No: T83198

Cat.No: T7748

Synonym: 皮啡肽三氟乙酸盐

Target: Others, Opioid Receptor

Cat.No: T7404

Synonym: 皮啡肽

Target: Opioid Receptor

Cat.No: TP1351L

Target: Others

Cat.No: T8455

Target: Opioid Receptor

Eptifibatide acetate (148031-34-9 free base)

Cat.No: T5146

Synonym: Eptifibatide acetate,依菲巴特醋酸盐

Target: Others

Angiotensin (1-7)

Cat.No: T7339

Synonym: Ang-(1-7),Angiotensin 1-7,ASP-ARG-VAL-TYR-ILE-HIS-PRO

Target: RAAS, Endogenous Metabolite

Cat.No: TP1351

Synonym: 肯普肽

Target: PKA

Cat.No: T30872

Synonym: CHEC7

Cat.No: T25480

Synonym: H-256,H256,Pro-thr-glu-phe-CH2NH-phe-arg-glu

Cat.No: T24474

Synonym: MK-0852,L-367,073,MK0852,L 367,073,L367,073

Cat.No: T31133

Synonym: Cyclo cadagac

Cat.No: T70418

Cat.No: T32408

Synonym: Ser-Phe-Asn-Pns-Pro-Ile-Val-NH2,KNI-122,KNI122

Cat.No: TP2343

Cat.No: T24203

Synonym: Jmv-170,Jmv170

Cat.No: T25507

Synonym: HP-228,Ac-Nle-gln-his-D-phe-arg-D-trp-gly-NH2,HP228

Cat.No: T38191

Super-TDU (1-31) TFA

Cat.No: TP1331

Cat.No: T71935

Substance P (5-11)

Cat.No: T76454

Alexamorelin Met 1

Cat.No: TP1261

Synonym: (D-Mrp)-Ala-Trp-(D-Phe)

Dermorphin Analog

Cat.No: TP1870

Cat.No: T76354

Cat.No: T5020

Synonym: Eptifibatide Acetate,Mpr-Har-Gly-Asp-Trp-Pro-Cys-NH2,依替巴肽

Target: Others

Cat.No: T36471

Cat.No: T83734

Cat.No: T37496

Angiotensin (1-7) (acetate)

Cat.No: T37495

Amyloid-Forming peptide GNNQQNY

Cat.No: T83122

Cat. No.	Product Name	Target	Signaling Pathways
T81816	Met-Enkephalin-Arg-Phe
	Met-Enkephalin-Arg-Phe 是一种天然七肽，具有镇痛活性。
T83245	7-Desmethylmicrocystin-LR
	7-Desmethylmicrocystin-LR为有毒七肽类化合物，可自无菌铜绿微囊藻菌株（K-139）中提取。
T75635	Microcystin-LY
	Microcystin-LY 是一种铜绿微囊藻蓝藻的环状七肽毒素，可作为 Nrf2通路的激活剂引起氧化应激反应,在3μM 时诱导效果非常明显。

天然产物

Met-Enkephalin-Arg-Phe

Cat.No: T81816

7-Desmethylmicrocystin-LR

Cat.No: T83245

Cat.No: T75635

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