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11

抑制剂 & 化合物

3

天然产物

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Cat. No. Product Name Target Signaling Pathways
T4502 BISMUTH SUBGALLATE

次没食子酸铋,Dermatol Puder,Bismuth Gallate

Others Others
Bismuth subgallate (Dermatol Puder) 是一种止血剂,可作用于凝血因子 XII ,促使凝血级联的激活,改善纤维蛋白凝块的早期形成。
T19786 Hematin

Ferrihemate,Ferriheme hydroxide,Ferriheme,Ferrihemic acid,羟高铁血红素

Others Others
Hematin (Ferrihemic acid) 是含铁卟啉,可以结合止血蛋白诱导其失活,降低凝血因子的活性以及阻碍纤维蛋白凝块的溶解。它可用于研究急性卟啉症和癌症。
TP1049L Ornipressin Acetate(3397-23-7,free)

鸟氨酸加压素,Orpressin,POR-8

Others Others
Ornipressin Acetate (POR-8) 是一种有效的血管收缩剂、止血剂和肾脏剂。
T9992 SphK1&2-IN-1

S1P Receptor GPCR/G Protein
SphK1&2-IN-1 是一种鞘氨醇激酶抑制剂,具有抗炎、抗肿瘤和止血作用。
T0312 Toluidine Blue

氯托洛宁,Blutene chloride

Others Others
Toluidine Blue (Blutene chloride) 是碱性噻嗪异染染料,能够高度亲和酸性组织成分,广泛应用于活体组织的重要染色及特殊染色。
T0002 Ethamsylate

Cyclonamine,Etamsylate,酚磺乙胺,Dicynene,Aglumin

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Ethamsylate (Dicynene) 通常用作止血药,增加毛细血管内皮阻力和血小板粘附,抑制前列腺素的生物合成和作用。
T0948 Adrenalone hydrochloride

Adrenalone HCl,肾上腺酮盐酸盐,盐酸肾上腺酮

Adrenergic Receptor GPCR/G Protein; Neuroscience
Adrenalone hydrochloride (Adrenalone HCl) 是一种多巴胺β氧化酶 (dopamine β oxidase) 抑制剂,结构与去甲肾上腺素转运蛋白 (NET) 配体相似,IC50=36.9 μM。它是一种肾上腺素能 (adrenergic) 激动剂,用作局部血管收缩剂和止血剂。
T3616 Carbazochrome

AC-17,Adrenostazin,Cromadrenal,Adona,Adchnon,卡巴克络,Adedolon

Others; Phospholipase Metabolism; Others
Carbazochrome (Adchnon) 是毛细管稳定剂,是抗出血剂,用于研究出血。
T28128 Naftazone

Etioven,C05CX02

Naftazone is a vasoprotectant drug used for hemostasis. Naftazone is shown to accelerate human saphenous vein endothelial cell proliferation in vitro at concentrations which did not alter the hemostatic balance.
T24442 Mecrylate

Mecrylate polymerizes in contact with moisture. It is used as a tissue adhesive. It also has higher homologs have hemostatic and antibacterial properties.
T37964 Dicresulene diammonium

Dicresulene diammonium is an impurity found in Policresulen, which is an organic acid possessing hemostatic, antimicrobial, and antiviral properties[1][2].

化合物

BISMUTH SUBGALLATE
Cat.No: T4502
Synonym: 次没食子酸铋,Dermatol Puder,Bismuth Gallate
Target: Others
Hematin
Cat.No: T19786
Synonym: Ferrihemate,Ferriheme hydroxide,Ferriheme,Ferrihemic acid,羟高铁血红素
Target: Others
Ornipressin Acetate(3397-23-7,free)
Cat.No: TP1049L
Synonym: 鸟氨酸加压素,Orpressin,POR-8
Target: Others
SphK1&2-IN-1
Cat.No: T9992
Synonym:
Target: S1P Receptor
Toluidine Blue
Cat.No: T0312
Synonym: 氯托洛宁,Blutene chloride
Target: Others
Ethamsylate
Cat.No: T0002
Synonym: Cyclonamine,Etamsylate,酚磺乙胺,Dicynene,Aglumin
Target: Prostaglandin Receptor
Adrenalone hydrochloride
Cat.No: T0948
Synonym: Adrenalone HCl,肾上腺酮盐酸盐,盐酸肾上腺酮
Target: Adrenergic Receptor
Carbazochrome
Cat.No: T3616
Synonym: AC-17,Adrenostazin,Cromadrenal,Adona,Adchnon,卡巴克络,Adedolon
Target: Others, Phospholipase
Naftazone
Cat.No: T28128
Synonym: Etioven,C05CX02
Target:
Mecrylate
Cat.No: T24442
Synonym:
Target:
Dicresulene diammonium
Cat.No: T37964
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T7106 Menaquinone-4

四烯甲萘醌,Vitamin K2,Menaquinone K4

Others; Endogenous Metabolite Metabolism; Others
Menaquinone-4 (Vitamin K2) 是维生素 K 的一种,用作止血剂,有潜力用于骨质疏松的研究。
TL0001 dencichine

L-Dencichin,ODAP,Dencichin,三七素

Others; HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; Metabolism; Others
Dencichine (ODAP) 是抑制从三七中分到的非蛋白氨基酸,可抑制 HIF-prolyl hydroxylase-2 的活性。
T40758 Hydrastinine

Hydrastinine, a key alkaloid component found in Hydrastis canadensis (goldenseal), serves as an effective hemostatic agent.

天然产物

Menaquinone-4
Cat.No: T7106
Synonym: 四烯甲萘醌,Vitamin K2,Menaquinone K4
Target: Others, Endogenous Metabolite
dencichine
Cat.No: TL0001
Synonym: L-Dencichin,ODAP,Dencichin,三七素
Target: Others, HIF/HIF Prolyl-Hydroxylase
Hydrastinine
Cat.No: T40758
Synonym:
Target:
TargetMol Loading
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