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Cat. No.	Product Name	Target	Signaling Pathways
T21992	Vacuolin-1	PI3K; Autophagy	Autophagy; PI3K/Akt/mTOR signaling
	Vacuolin-1 是一种细胞渗透性抑制剂，可抑制 Ca2+ 依赖性溶酶体与细胞膜的融合。它通过抑制溶酶体内容物的释放起作用。它是一种有效的选择性 PIKfyve 抑制剂，通过损害溶酶体成熟来抑制晚期自噬。
TP1915	Boc-MLF	Others	Others
	Boc-MLF 是甲酰肽受体 1 (FPR1) 的拮抗剂。它减少 fMLF 诱导的超氧化物产生，EC50 为 0.63 μM。几乎完全阻断 fMLF 刺激的初级颗粒胞吐作用。
T31790	FFN200 dihydrochloride FFN200 HCl,FFN200,FFN 200,FFN-200
	FFN200 is a vesicular monoamine transporter 2 (VMAT2) substrate that selectively traces monoamine exocytosis in both neuronal cell culture and brain tissue.
T69194	Endosidin5
	Endosidin5 is a novel exocytosis inhibitor.
T14829	Bromoenol lactone (6E)-Bromoenol lactone	Phospholipase	Metabolism
	Bromoenol lactone is a suicide-based irreversible, selective, potent inhibitor of calcium-independent phospholipase A2 (iPLA2β; IC50: ~7 μM). It inhibits antigen-stimulated mast cell exocytosis without blocking Ca2+ influx.
T81035	TAT-NSF222 Fusion Peptide
	TAT-NSF222 Fusion Peptide为包含TAT和NSF两个结构域的融合多肽，TAT负责通过巨胞饮促进细胞摄取，而NSF结构域则抑制N-乙基马来酰亚胺敏感因子(NSF)活性。该融合多肽是exocytosis的抑制剂。
T61265	Exo2
	Exo2 is a secretion inhibitor that hinders the trafficking of Shiga toxin from endosomes to the trans-Golgi network. It inhibits the exit of secretory cargo from the endoplasmic reticulum (ER) and disrupts the Golgi apparatus. Notably, Exo2 does not impact the morphology of the trans-Golgi network (TGN). Additionally, Exo2 has the ability to induce calcium-dependent exocytosis in permeabilized adrenal chromaffin cells [1] [2].
TP1576	SNAP-25 187-203
	This amino acids187 to 203 fragment is derived from the C-terminal helix of synaptosomal-associated protein of 25 kDa (SNAP-25). This peptide is able to rescue exocytosis from botulinum neurotoxin E (BoNT/E)-treated cells, albeit at higher concentrations
T76549	TAT-NSF700scr
	TAT-NSF700scr拥有完整的TAT结构域和甘氨酸连接肽，后接随机排列的NSF氨基酸序列，该化合物作为非抑制SNARE介导的胞吐作用的对照肽而被使用。
T75793	ω-Agatoxin IVA TFA
	ω-Agatoxin IVA TFA 是一种高效的针对P/Q型Ca2+(Cav2.1)通道的选择性阻滞剂，IC50对P型为2 nM，对Q型为90 nM。此化合物能够抑制高钾条件下的谷氨酸释放和钙流入，IC50在30-225 nM范围。同时，ω-Agatoxin IVA TFA阻断高钾诱发的5-羟色胺及去甲肾上腺素释放，但不影响L型或N型Ca2+通道。