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4

抑制剂 & 化合物

2

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Cat. No. Product Name Target Signaling Pathways
T21980 PD 198306

MEK MAPK
PD 198306 是一种具有抗痛觉过敏作用的 MAPK/ERK 激酶 (MEK) 选择性抑制剂。 PD 198306 可降低链脲佐菌素诱导的活性 ERK1 水平升高。
T67752 Compound V007-6018

Others Others
Compound V007-6018是一种类药化合物,用于药物筛选。
T78520 CYT296

Others Others
CYT296是一种靶向染色质去凝集的化合物,能增强定义因子(OSKM)介导诱导多能干细胞(iPSC)的生成,并通过诱导小鼠胚胎成纤维细胞(MEFs)染色质的开放状态来促进体细胞的重编程,适用于细胞替代治疗和药物筛选的研究领域。
T36695 TAS-103

TAS-103 is a dual inhibitor of DNA topoisomerase I/II, used for cancer research. TAS-103 is a dual inhibitor of DNA topoisomerase I/II. TAS-103 (0.1-10 μM) is active on CCRF-CEM cells, with an IC50 value of 5 nM. TAS-103 (0.1 μM) significantly increases levels of topo IIα FITC immunofluorescence in individual CCRF-CEM cells[1]. TAS-103 (0.01-1 μM) is highly cytotoxic to Lewis lung carcinoma (LLC) cells, and Liposomal TAS-103 is almost as active as free TAS-103[2]. TAS-103 inhibits the viability ...

化合物

PD 198306
Cat.No: T21980
Synonym:
Target: MEK
Compound V007-6018
Cat.No: T67752
Synonym:
Target: Others
CYT296
Cat.No: T78520
Synonym:
Target: Others
TAS-103
Cat.No: T36695
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T17143 Toyocamycin

丰加霉素,Vengicide

Apoptosis; Others; IRE1; Antibiotic; Antifungal Apoptosis; Cell Cycle/Checkpoint; Microbiology/Virology; Others
Toyocamycin (Vengicide) 是放线菌类产生的腺苷类似物,为 X 盒结合蛋白 1 (XBP1) 抑制剂,抑制 IRE1α 诱导的 ATP 依赖性 XBP1 mRNA 的断裂,IC50值为 80 nM。它还诱导凋亡。
T4S0051 Coptisine sulfate

Indoleamine 2,3-Dioxygenase (IDO) Metabolism
Coptisine Sulfate 是一种从黄连中分离到的生物碱,是非竞争性的IDO 抑制剂,Ki=为 5.8 μM,IC50=6.3 μM。

天然产物

Toyocamycin
Cat.No: T17143
Synonym: 丰加霉素,Vengicide
Target: Apoptosis, Others, IRE1, Antibiotic, Antifungal
Coptisine sulfate
Cat.No: T4S0051
Synonym:
Target: Indoleamine 2,3-Dioxygenase (IDO)
TargetMol Loading
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