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Cat. No. Product Name Target Signaling Pathways
T82733 Cholecystokinin

CCK-33(human),Cholecystokinin-33(human)

Cholecystokinin是一种通过抑制食物摄入并促进脂肪及蛋白质消化作用的肽类激素,常用于胃肠系统研究。
TP2500 Cholecystokinin (26-33) free acid

CCK (26-33) free acid

cholecystokinin GPCR/G Protein
Cholecystokinin (26-33) free acid 是胆囊收缩素 (CCK) 的一部分, 是脊椎动物中枢神经系统中存在的 CCKB 型受体的高选择性配体,可诱导大鼠轻度味觉厌恶条件反射。
TP2419 V-9-M Cholecystokinin nonapeptide

V 9 M,Prepro CCK Fragment V-9-M,Val-pro-val-glu-ala-val-asp-pro-met,Cholecystokinin Precursor (24-32),V9M,V-9-M

Beta Amyloid Neuroscience
V-9-M Cholecystokinin nonapeptide (Prepro CCK Fragment V-9-M) 是胆囊收缩素(CCK)的前体化合物。胆囊收缩素(CCK)是一种刺激胆囊收缩和胰腺外分泌的脑肠肽,可从狗和猫的小肠中提取的,可以引起胆囊收缩。
TP1198 Sincalide ammonium

SQ19844 ammonium,CCK-8 ammonium,Cholecystokinin octapeptide ammonium

cholecystokinin GPCR/G Protein
Sincalide ammonium (CCK-8 ammonium) 是一种有效的氨基酸多肽激素胆囊收缩素 (CCK) 的类似物,是保留了 CCK 的大部分生物活性的活性片段。Sincalide ammonium 促进胆汁的分泌,使胆囊收缩并使 Oddi 的括约肌松弛,从而促进胆汁排入十二指肠。Sincalide ammonium 可通过注射促进胆囊收缩,常用于辅助诊断胆囊、胰腺疾病和胆囊造影术。
T39170 Cholecystokinin Octapeptide, desulfated TFA

CCK Octapeptide, desulfated TFA,Cholecystokinin Octapeptide, desulfated TFA

Cholecystokinin Octapeptide, desulfated TFA, is a synthetic octapeptide derived from Cholecystokinin (CCK) that has undergone desulfation.
T23886 Cholecystokinin (27-32)-amide

Cholecystokinin (27-32)-NH2

Cholecystokinin (27-32)-amide is a CCK receptor antagonist.
TP1197 Sincalide

SQ19844,辛卡利特,CCK-8,Cholecystokinin octapeptide

Others Others
Sincalide (CCK-8) 是一种速效的胆囊收缩素的氨基酸多肽激素类似物,可在胆囊造影术中静脉使用。它的肝胆生理作用是增加胆汁的分泌,使胆囊收缩并使 Oddi 的括约肌松弛,从而使胆汁排入十二指肠。它是一种通过注射促进胆囊收缩并帮助诊断胆囊和胰腺疾病的药物。
T30904 Cholecystokinin-J

CCK-J

Cholecystokinin-J can be used in cholecystography, radiomanometry and biliary cinematography.
TP2376 Cholecystokinin pentapeptide

CCK-5,Gly-trp-met-asp-phe-NH2

Cholecystokinin pentapeptide is a peptide hormone of the gastrointestinal system responsible for stimulating the digestion of fat and protein.
TP2204 Cholecystokinin Octapeptide, desulfated

CCK Octapeptide, non-sulfated

Others Others
Non-sulfated form of the C-terminal octapeptide of CCK
T82732 Cholecystokinin (1-21)

CCK-1-21

Cholecystokinin (1-21),作为一种胆囊收缩素 (CCK) 片段,能够激活人体脂肪组织的脂肪分解作用。
T20492 Tetragastrin

Cholecystokinin tetrapeptide,Gastrin tetrapeptide

Tetragastrin is the C-terminal tetrapeptide of gastrin. It has the same physiological and pharmacological activity as gastrin.
T83485 [Thr28, Nle31]-Cholecystokinin (25-33), sulfated

[Thr28, Nle31]-Cholecystokinin (25-33) 是一种具备CCK8所有生物活性的胆囊收缩素 (CCK) 类似物,表现出食欲抑制功效。它在胃肠道系统和中枢神经系统中担任激素和神经递质角色。此肽通过 Thr28 和 Nle31 的特殊替代,展现出在酸性条件下的高稳定性,并能抵抗空气氧化(防止蛋氨酸受损)。其主要构象特征为以Thr4为核心的γ转角和Gly5分隔的C末端螺旋片段。
T2312 Loxiglumide

CR-1505,氯谷胺

cholecystokinin GPCR/G Protein
Loxiglumide (CR-1505) 是一种缩胆囊素受体拮抗剂。
TQ0062 Nastorazepide

Z-360

cholecystokinin GPCR/G Protein
Nastorazepide 是一种选择性的、口服有效的1,5-苯并二氮杂环衍生物胃泌素/胆囊收缩素2(CCK-2)受体拮抗剂,具有抗肿瘤的潜能。
T14932 Ceruletide

Cerulein,Caerulein,雨蛙素,FI-6934

cholecystokinin GPCR/G Protein
Ceruletide (Caerulein) 是一种十肽,是一种安全有效的胆囊收缩剂,是一种胆囊收缩素受体激动剂,对胆囊肌肉和胆管有直接的痉挛性作用。
T1052 Proglumide

二丙谷酰胺

cholecystokinin GPCR/G Protein
Proglumide (Binoside) 是一种非肽的、口服具有活性的胆囊收缩素(CCK)-A/B 受体拮抗剂。它能够选择性阻断 CCK 在中枢神经系统中的作用。它能够抑制胃分泌,具有保护胃十二指肠粘膜的能力,并表现出抗癫痫和抗氧化活性。
T4579 Pentagastrin

五肽胃泌素,ICI-50123

Others; cholecystokinin GPCR/G Protein; Others
Pentagastrin (ICI-50123) 是一种选择性的胆囊收缩素 B(CCKB) 受体激动剂,IC50=11 nM。它能够增强胃粘膜对酸的防御机制,并保护胃粘膜免受损伤。
TP2204L CCK Octapeptide, non-sulfated acetate

CCK Octapeptide, non-sulfated acetate(25679-24-7 Free base)

cholecystokinin GPCR/G Protein
CCK Octapeptide, non-sulfated acetate 是一种合成的胆囊收缩素脱硫酸肽。
T15382 GI 181771

cholecystokinin GPCR/G Protein
GI 181771 是胆囊收缩素 1 受体的激动剂。 GI 181771 可用于肥胖研究。
T27503 GV150013

GV 150013,GV-150013

cholecystokinin GPCR/G Protein
GV150013是一种 cholecystokinin-2 (CCK2)受体拮抗剂。
T9343 N-Cbz-DL-tryptophan

cholecystokinin GPCR/G Protein
N-Cbz-DL-tryptophan 是一种胆囊收缩素受体拮抗剂,可消除离体心脏对 CCK-8 的反应。
T34123 Pranazepide

FR120480,FK 480,FR-120480

cholecystokinin GPCR/G Protein
Pranazepide (FK 480) 是一种小分子胆囊收缩素受体拮抗剂,可用于研究消化系统疾病和胰腺炎。
T14932L1 Ceruletide Ammonium Salt

Caerulein Ammonium Salt,Ceruletide Ammonium Salt(17650-98-5 Free base),FI-6934 Ammonium Salt,Cerulein Ammonium Salt

cholecystokinin GPCR/G Protein
Ceruletide Ammonium Salt 是一种十肽,起源于热带青蛙的皮肤,是一种有效的胆囊收缩素受体 (cholecystokinin receptor) 激动剂,也是一种安全有效的胆囊收缩剂,对胆囊肌肉和胆管有直接的痉挛性作用。Ceruletide Ammonium Salt 具有镇静活性,可用于研究慢性精神分裂症。
TP2030L1 Gastrin I (human) acetate

Gastrin I (human) acetate(10047-33-3 free base),Gastrin-17 acetate,Little gastrin I acetate,胃膜素醋酸盐

cholecystokinin GPCR/G Protein
Gastrin I (human) acetate (Gastrin-17 acetate) 是在胃中产生的内源性肽,通过胆囊收缩素 2 (CCK2) 受体增加胃酸分泌。
T11868 Lorglumide sodium salt

CR-1409 sodium salt

cholecystokinin GPCR/G Protein
Lorglumide sodium salt (CR-1409 sodium salt) 是胆囊收缩素受体 (CCK) 的拮抗剂。
T12404 CCK-A receptor inhibitor 1

cholecystokinin GPCR/G Protein
CCK-A receptor inhibitor 1 是一种有效的缩胆囊素 A (CCK-A) 受体抑制剂(IC50:340 nM)。CCK-A receptor inhibitor 1 可用于研究与消化系统相关的疾病。
T25116 Asperlicin D

AsperlicinD,Asperlicin-D

Asperlicin D is a cholecystokinin antagonist agent.
T26483 A-65186

A65186

A 65186 is a Type A Cholecystokinin (CCK) receptor antagonist.
T27664 JNJ-17156516

JNJ17156516,JNJ 17156516

JNJ-17156516 is a potent, and selective cholecystokinin 1 receptor antagonist.
T71277 Amiglumide

Amiglumide is a non-peptide cholecystokinin antagonist.
T32297 Jmv 180

Cck-jmv-180,Jmv-180,Jmv180

Jmv 180, a CCK analog, can distinguish high-affinity cholecystokinin receptors from low-affinity cholecystokinin receptors.
T25551 Jmv 236

Jmv236,t-Boc(nle(28,31))-cck (26-33),Jmv-236

Jmv 236 is a cholecystokinin antagonist.
T26971 Ceclazepide

Ceclazepide is an antagonist of cholecystokinin receptor.
T15105 Dexloxiglumide

Others Others
Dexloxiglumide, an active enantiomer of Loxiglumide, inhibits smooth muscle cell contractions induced by cholecystokinin-octapeptide (CCK-8). It is a selective antagonist of cholecystokinin type A (CCKA) receptors.
T71408 A 68552

A 68552 is a cholecystokinin agonist.
T28613 RP73870

RP 73870,RP-73870

RP73870 is a gastrin/cholecystokinin-B receptor antagonist and H2 receptor antagonist with potent anti-ulcer activity.
T23185 Proglumide sodium

丙谷胺钠,Proglumide sodium salt

Others Others
Non-selective cholecystokinin (CCK) antagonist
T27669 JNJ-26070109

JNJ26070109

JNJ-26070109, an antagonist of cholecystokinin CCK2 receptor, inhibits gastric acid secretion and prevents omeprazole-induced acid rebound in the rat.
T24202 Jmv 167

Jmv-167,Jmv167

Jmv 167 is an antagonist of the Cholecystokinin receptor.
T24204 Jmv 179

Jmv-179,Jmv179

Jmv 179 is an antagonist of the cholecystokinin receptor.
T24293 L 368935

L-368935,L368,935,L-368,935,L 368,935,L368935

L 368935 is an antagonist of the cholecystokinin receptor.
T29502 A 70874

A-70874,A70874

A70874 has high selectivity and potency for cholecystokinin (CCK) a receptor.
T28335 PD 140376

PD-140376,PD140376

PD 140376 is a highly selective antagonist radioligand for the cholecystokinin(B)-gastrin receptor in guinea pig gastric mucosa & cerebral cortex in the peripheral and central nervous systems.
T10055 (Iso)-FK-480

CHEMBL333994

cholecystokinin GPCR/G Protein
(Iso)-FK-480 是一种新型可口服的胆囊收缩素 A(CCK-A)拮抗剂,可用于研究治疗慢性胰腺炎。
T28331 PD 136450

Cam1189,PD136450,Cam-1189,PD-136450,Cam 1189

Cholecystokinin type B receptor antagonist PD-136,450 is a partial secretory agonist in the stomach and a full agonist in the pancreas of the rat. Gastrin (cholecystokinin type B (CCK-B)) receptor antagonists may help to elucidate the physiological role o
T22895 L-365260

L-365,260

Others Others
cholecystokinin receptor 2 (CCK2) antagonist
T15101 Devazepide

L-364,718,地伐西匹,MK-329

Others Others
Devazepide is a competitive and orally active nonpeptide antagonist of cholecystokinin (CCK) receptor (IC50s: 81 pM, 45 pM, and 245 nM for rat pancreatic, bovine gallbladder and guinea pig brain CCK receptors, respectively).
T26198 Snf 9007

Snf-9007,Asp-tyr-D-phe-gly-trp-(N-Me)nle-asp-phe-NH2,Snf9007

Snf 9007 is an antagonist of cholecystokinin.
T34668 Snf 8814

Snf-8814,Snf8814

Snf 8814 is an analog of centrally selective cholecystokinin.

化合物

Cholecystokinin
Cat.No: T82733
Synonym: CCK-33(human),Cholecystokinin-33(human)
Target:
Cholecystokinin (26-33) free acid
Cat.No: TP2500
Synonym: CCK (26-33) free acid
Target: cholecystokinin
V-9-M Cholecystokinin nonapeptide
Cat.No: TP2419
Synonym: V 9 M,Prepro CCK Fragment V-9-M,Val-pro-val-glu-ala-val-asp-pro-met,Cholecystokinin Precursor (24-32),V9M,V-9-M
Target: Beta Amyloid
Sincalide ammonium
Cat.No: TP1198
Synonym: SQ19844 ammonium,CCK-8 ammonium,Cholecystokinin octapeptide ammonium
Target: cholecystokinin
Cholecystokinin Octapeptide, desulfated TFA
Cat.No: T39170
Synonym: CCK Octapeptide, desulfated TFA,Cholecystokinin Octapeptide, desulfated TFA
Target:
Cholecystokinin (27-32)-amide
Cat.No: T23886
Synonym: Cholecystokinin (27-32)-NH2
Target:
Sincalide
Cat.No: TP1197
Synonym: SQ19844,辛卡利特,CCK-8,Cholecystokinin octapeptide
Target: Others
Cholecystokinin-J
Cat.No: T30904
Synonym: CCK-J
Target:
Cholecystokinin pentapeptide
Cat.No: TP2376
Synonym: CCK-5,Gly-trp-met-asp-phe-NH2
Target:
Cholecystokinin Octapeptide, desulfated
Cat.No: TP2204
Synonym: CCK Octapeptide, non-sulfated
Target: Others
Cholecystokinin (1-21)
Cat.No: T82732
Synonym: CCK-1-21
Target:
Tetragastrin
Cat.No: T20492
Synonym: Cholecystokinin tetrapeptide,Gastrin tetrapeptide
Target:
[Thr28, Nle31]-Cholecystokinin (25-33), sulfated
Cat.No: T83485
Synonym:
Target:
Loxiglumide
Cat.No: T2312
Synonym: CR-1505,氯谷胺
Target: cholecystokinin
Nastorazepide
Cat.No: TQ0062
Synonym: Z-360
Target: cholecystokinin
Ceruletide
Cat.No: T14932
Synonym: Cerulein,Caerulein,雨蛙素,FI-6934
Target: cholecystokinin
Proglumide
Cat.No: T1052
Synonym: 二丙谷酰胺
Target: cholecystokinin
Pentagastrin
Cat.No: T4579
Synonym: 五肽胃泌素,ICI-50123
Target: Others, cholecystokinin
CCK Octapeptide, non-sulfated acetate
Cat.No: TP2204L
Synonym: CCK Octapeptide, non-sulfated acetate(25679-24-7 Free base)
Target: cholecystokinin
GI 181771
Cat.No: T15382
Synonym:
Target: cholecystokinin
GV150013
Cat.No: T27503
Synonym: GV 150013,GV-150013
Target: cholecystokinin
N-Cbz-DL-tryptophan
Cat.No: T9343
Synonym:
Target: cholecystokinin
Pranazepide
Cat.No: T34123
Synonym: FR120480,FK 480,FR-120480
Target: cholecystokinin
Ceruletide Ammonium Salt
Cat.No: T14932L1
Synonym: Caerulein Ammonium Salt,Ceruletide Ammonium Salt(17650-98-5 Free base),FI-6934 Ammonium Salt,Cerulein Ammonium Salt
Target: cholecystokinin
Gastrin I (human) acetate
Cat.No: TP2030L1
Synonym: Gastrin I (human) acetate(10047-33-3 free base),Gastrin-17 acetate,Little gastrin I acetate,胃膜素醋酸盐
Target: cholecystokinin
Lorglumide sodium salt
Cat.No: T11868
Synonym: CR-1409 sodium salt
Target: cholecystokinin
CCK-A receptor inhibitor 1
Cat.No: T12404
Synonym:
Target: cholecystokinin
Asperlicin D
Cat.No: T25116
Synonym: AsperlicinD,Asperlicin-D
Target:
A-65186
Cat.No: T26483
Synonym: A65186
Target:
JNJ-17156516
Cat.No: T27664
Synonym: JNJ17156516,JNJ 17156516
Target:
Amiglumide
Cat.No: T71277
Synonym:
Target:
Jmv 180
Cat.No: T32297
Synonym: Cck-jmv-180,Jmv-180,Jmv180
Target:
Jmv 236
Cat.No: T25551
Synonym: Jmv236,t-Boc(nle(28,31))-cck (26-33),Jmv-236
Target:
Ceclazepide
Cat.No: T26971
Synonym:
Target:
Dexloxiglumide
Cat.No: T15105
Synonym:
Target: Others
A 68552
Cat.No: T71408
Synonym:
Target:
RP73870
Cat.No: T28613
Synonym: RP 73870,RP-73870
Target:
Proglumide sodium
Cat.No: T23185
Synonym: 丙谷胺钠,Proglumide sodium salt
Target: Others
JNJ-26070109
Cat.No: T27669
Synonym: JNJ26070109
Target:
Jmv 167
Cat.No: T24202
Synonym: Jmv-167,Jmv167
Target:
Jmv 179
Cat.No: T24204
Synonym: Jmv-179,Jmv179
Target:
L 368935
Cat.No: T24293
Synonym: L-368935,L368,935,L-368,935,L 368,935,L368935
Target:
A 70874
Cat.No: T29502
Synonym: A-70874,A70874
Target:
PD 140376
Cat.No: T28335
Synonym: PD-140376,PD140376
Target:
(Iso)-FK-480
Cat.No: T10055
Synonym: CHEMBL333994
Target: cholecystokinin
PD 136450
Cat.No: T28331
Synonym: Cam1189,PD136450,Cam-1189,PD-136450,Cam 1189
Target:
L-365260
Cat.No: T22895
Synonym: L-365,260
Target: Others
Devazepide
Cat.No: T15101
Synonym: L-364,718,地伐西匹,MK-329
Target: Others
Snf 9007
Cat.No: T26198
Synonym: Snf-9007,Asp-tyr-D-phe-gly-trp-(N-Me)nle-asp-phe-NH2,Snf9007
Target:
Snf 8814
Cat.No: T34668
Synonym: Snf-8814,Snf8814
Target:
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