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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T1491 Atovaquone

Atavaquone,阿托伐醌

Others; P450; Dehydrogenase; Antibiotic; Parasite Metabolism; Microbiology/Virology; Others
Atovaquone (Atavaquone) 是具有口服活性的选择性寄生虫线粒体细胞色素bc1复合物的抑制剂。它抑制人类和P. falciparum 细胞色素bc1活性,IC50值分别为 460 nM 和 2.0 nM。它有抗疟作用,有潜力用于疟疾、弓形体病、肺孢子虫肺炎和巴贝斯虫病的相关研究。
T10785 Chalcone 4 hydrate

Others; Parasite Microbiology/Virology; Others
Chalcone 4 hydrate 是一种抗寄生虫剂,可抑制 Babesia 和 Theileria 的生长。
T23132 Pentamidine dihydrochloride

喷他脒二盐酸盐,MP-601205 dihydrochloride

Phosphatase; Antibacterial; Antibiotic; Parasite; Antifungal Metabolism; Microbiology/Virology
Pentamidine dihydrochloride (MP-601205 dihydrochloride) 是一种抗微生物剂,会干扰 DNA 的生物合成。它是选择性蛋白酪氨酸磷酸酶和再生肝磷酸酶抑制剂。它可用于冈比亚锥虫病,抗锑利什曼病和卡氏肺孢子虫肺炎的研究,有抗肿瘤活性,抗菌活性。
T28488 Quinuronium Sulfate

Pirevan,Zothelone,Acaprin

Quinuronium sulfate is a drug used to treat Babesia divergens infections in calves. It did not prevent treated animals from being disease carriers. It may also cause hepatic centrilobular fatty degeneration, but no depletion of hepatic glutathione (GSH).
T19198 Atovaquone-d4

阿托伐醌D4

Others Others
Atovaquone D4 is the deuterium-labeled Atovaquone. Atovaquone is a medication used to treat or prevent pneumocystis babesia, malaria, toxoplasmosis, and pneumonia.

化合物

Atovaquone
Cat.No: T1491
Synonym: Atavaquone,阿托伐醌
Target: Others, P450, Dehydrogenase, Antibiotic, Parasite
Chalcone 4 hydrate
Cat.No: T10785
Synonym:
Target: Others, Parasite
Pentamidine dihydrochloride
Cat.No: T23132
Synonym: 喷他脒二盐酸盐,MP-601205 dihydrochloride
Target: Phosphatase, Antibacterial, Antibiotic, Parasite, Antifungal
Quinuronium Sulfate
Cat.No: T28488
Synonym: Pirevan,Zothelone,Acaprin
Target:
Atovaquone-d4
Cat.No: T19198
Synonym: 阿托伐醌D4
Target: Others
Cat. No. Product Name Target Signaling Pathways
TN1453 Bruceantinol

Anti-infection Microbiology/Virology
Bruceantinol 是一种quassinol 化合物,分离自Brucea javanica 的 CH3OH 提取物。它能够将系统性寄主植物中灭活。有效的抑制浓度为 10 μM。

天然产物

Bruceantinol
Cat.No: TN1453
Synonym:
Target: Anti-infection
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