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Search Results for " verapamil "

18

抑制剂 & 化合物

3

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T20656	Verapamil NSC 135784,维拉帕米,NSC-135784,CP-16533-1,(±)-Verapamil	P450; Calcium Channel; P-gp	Membrane transporter/Ion channel; Metabolism; Neuroscience
	Verapamil (CP-16533-1) 是一种钙通道阻滞剂，是一种口服有效的 P-gp 抑制剂。Verapamil 抑制 CYP3A4，可用于治疗高血压、心律失常和心绞痛的研究。
T1010	Verapamil hydrochloride Manidon,盐酸维拉帕米,(±)-Verapamil hydrochlorid,Verapamil HCl,Calcan hydrochloride	P450; Calcium Channel; P-gp	Membrane transporter/Ion channel; Metabolism; Neuroscience
	Verapamil hydrochloride (Verapamil HCl) 是一种钙通道阻滞剂，是一种可口服的 P 糖蛋白 (P-gp) 抑制剂，可抑制CYP3A4，用于高血压、心律不齐和心绞痛的研究。
T13879	(S)-Verapamil hydrochloride (S)-(-)-Verapamil hydrochloride	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	(S)-Verapamil hydrochloride is an inhibitor of leukotriene C4 (LTC4) and calcein transport by MRP1,and leads to the death of potentially resistant tumor cells.
T12646	(R)-Verapamil hydrochloride (R)-(+)-Verapamil hydrochloride	Others	Others
	(R)-Verapamil hydrochloride ((R)-(+)-Verapamil hydrochloride) is a inhibitor of P-Glycoprotein.
T40591	Verapamil EP Impurity C hydrochloride NSC-609249 hydrochloride
	NSC-609249 hydrochloride, an impurity of Verapamil, is a calcium channel blocker with potent orally active properties. It also functions as a first-generation P-glycoprotein (P-gp) inhibitor.
T11353	Gallopamil Methoxyverapamil,戈洛帕米	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	Gallopamil (Methoxyverapamil) 是一种苯烷基胺钙拮抗剂，以浓度依赖性方式抑制酸分泌 (IC50 = 10.9 μM)。Gallopamil 显示出抗心律失常和血管扩张剂的功效。
T11353L	Gallopamil hydrochloride Methoxyverapamil hydrochloride	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	Gallopamil hydrochloride (Methoxyverapamil hydrochloride) 是苯烷基胺钙的拮抗剂。Gallopamil hydrochloride 可用于抗心律失常和血管扩张剂研究。
T16339	Norverapamil hydrochloride (±)-Norverapamil hydrochloride,D591 hydrochloride,盐酸去甲维拉帕米	Calcium Channel; P-gp; Drug Metabolite	Membrane transporter/Ion channel; Metabolism; Neuroscience
	Norverapamil hydrochloride (D591 hydrochloride) 是 Verapamil 的 N-去甲基代谢物，是 L 型钙通道阻滞剂和 P-糖蛋白 (P-gp) 功能抑制剂。
T30146	Arverapamil (R)-Norverapamil,Agi-003,UNII-3J8P56R04P,Rezular
	Arverapamil is a chiral metabolite of Verapamil.
T69317	Dexverapamil
	Dexverapamil is the R-enantiomer of the calcium channel blocker verapamil. Dexverapamil competitively inhibits the multidrug resistance efflux pump P-glycoprotein (MDR-1), thereby potentially increasing the effectiveness of a wide range of antineoplastic drugs which are inactivated by MDR-1 mechanisms.
T12244	Norverapamil D591,(±)-Norverapamil	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .
T12243	Norverapamil-d7 D591 D7,(±)-Norverapamil D7	Others	Others
	Norverapamil D7 is a deuterium labeled Norverapamil . Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .
T0563	Homoveratronitrile	Others	Others
	Homoveratronitrile 是Verapamil 的杂质。它也是制备肌肉松弛剂罂粟碱的中间体。
T69956	KR30031
	KR30031 is a novel P-glycoprotein inhibitor with potential anticancer activity. KR30031 is a verapamil analog with fewer cardiovascular effects. The ability of KR-30031 to reduce this efflux transport is equal to that of verapamil, a well-known P-glycoprotein inhibitor. The bioavailability of paclitaxel could be enhanced by coadministration of a P-glycoprotein inhibitor, KR-30031.
T26120	Ronipamil Ronipamilo
	Ronipamil is an analogue of verapamil that used as a calcium entry blocker.
T32912	Lu49888 HCl Azidopamil,LU49888,LU 49888,Ludopamil,LU-49888
	LU 49888 is a photoaffinity analog of verapamil that has been used to identify specific binding sites for phenylalkylamines of calcium channels present in rabbit skeletal muscle microsomes.
T27302	Falipamil AQ-A 39,AQ-A-39,AQ-A39
	Falipamil is a verapamil derivative and a calcium channel antagonist. Falipamil exerts antitachycardic effects by a direct action on the sinus node. Falipamil decreases HR at exercise in normal subjects and may exert antianginal effects in patients with m
T35568	BODIPY-aminoacetaldehyde diethyl acetal
	BODIPY-aminoacetaldehyde diethyl acetal (BAAA-DA) is a stable precursor to BODIPY-aminoacetaldehyde, a cell-permeable fluorescent substrate for aldehyde dehydrogenase (ALDH).1,2BODIPY-aminoacetaldehyde diethyl acetal is converted under acidic conditions to BODIPY-aminoacetaldehyde (BAAA).2BAAA is cell-permeant and is converted intracellularly by ALDH to BODIPY aminoacetate (BAA), which is retained by cells and can be used to identify cells with high ALDH activity.1BAA is a substrate for the effl...

化合物

Cat.No: T20656

Synonym: NSC 135784,维拉帕米,NSC-135784,CP-16533-1,(±)-Verapamil

Target: P450, Calcium Channel, P-gp

Verapamil hydrochloride

Cat.No: T1010

Synonym: Manidon,盐酸维拉帕米,(±)-Verapamil hydrochlorid,Verapamil HCl,Calcan hydrochloride

Target: P450, Calcium Channel, P-gp

(S)-Verapamil hydrochloride

Cat.No: T13879

Synonym: (S)-(-)-Verapamil hydrochloride

Target: Calcium Channel

(R)-Verapamil hydrochloride

Cat.No: T12646

Synonym: (R)-(+)-Verapamil hydrochloride

Target: Others

Verapamil EP Impurity C hydrochloride

Cat.No: T40591

Synonym: NSC-609249 hydrochloride

Cat.No: T11353

Synonym: Methoxyverapamil,戈洛帕米

Target: Calcium Channel

Gallopamil hydrochloride

Cat.No: T11353L

Synonym: Methoxyverapamil hydrochloride

Target: Calcium Channel

Norverapamil hydrochloride

Cat.No: T16339

Synonym: (±)-Norverapamil hydrochloride,D591 hydrochloride,盐酸去甲维拉帕米

Target: Calcium Channel, P-gp, Drug Metabolite

Cat.No: T30146

Synonym: (R)-Norverapamil,Agi-003,UNII-3J8P56R04P,Rezular

Cat.No: T69317

Cat.No: T12244

Synonym: D591,(±)-Norverapamil

Target: Calcium Channel

Norverapamil-d7

Cat.No: T12243

Synonym: D591 D7,(±)-Norverapamil D7

Target: Others

Homoveratronitrile

Cat.No: T0563

Target: Others

Cat.No: T69956

Cat.No: T26120

Synonym: Ronipamilo

Cat.No: T32912

Synonym: Azidopamil,LU49888,LU 49888,Ludopamil,LU-49888

Cat.No: T27302

Synonym: AQ-A 39,AQ-A-39,AQ-A39

BODIPY-aminoacetaldehyde diethyl acetal

Cat.No: T35568

Cat. No.	Product Name	Target	Signaling Pathways
TCS0102	Pulegone 胡薄荷酮,(+)-Pulegone,蒲勒酮，胡薄荷酮，长叶薄荷酮	Calcium Channel; Endogenous Metabolite; TRP/TRPV Channel	Membrane transporter/Ion channel; Metabolism
	Pulegone ((+)-Pulegone) 是 Calamintha nepeta (L.) Savi 的精油的主要化学成分，也是禽类驱虫剂之一。它在禽类物种中驱避作用的分子靶点是伤害感受性 TRP 锚蛋 1。它刺激鸡感觉神经元中的 TRPM8 和 TRPA1 通道，并在高浓度下抑制前者但不抑制后者。
TN2726	Jatrophane 5	P-gp	Membrane transporter/Ion channel; Neuroscience
	Jatrophane 5 demonstrates the most powerful inhibition of P-gp, higher than R(+)-verapamil and tariquidar in colorectal multi-drug resistant (MDR) cells (DLD1-TxR).
TN2727	Jatrophane 2	P-gp; Antifection	Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
	2,5,7,8,9,14-Hexaacetoxy-3-benzoyloxy-15-hydroxyjatropha-6(17),11E-diene (Jatrophane 2 ) exhibits significant antifeedant activity against a generalist plant-feeding insect, the cotton bollworm (Helicoverpa armigera). Jatrophane 2 also demonstrates the mo

天然产物

Cat.No: TCS0102

Synonym: 胡薄荷酮,(+)-Pulegone,蒲勒酮，胡薄荷酮，长叶薄荷酮

Target: Calcium Channel, Endogenous Metabolite, TRP/TRPV Channel

Cat.No: TN2726

Target: P-gp

Cat.No: TN2727

Target: P-gp, Antifection

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