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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T6993 Tauroursodeoxycholate sodium

牛磺熊脱氧胆酸钠,Sodium tauroursodeoxycholate,Tauroursodeoxycholic acid sodium salt,TUDC,牛磺熊去氧胆酸钠,Sodium Tauroursodeoxycholate (TUDC)

Apoptosis; ERK; Caspase Apoptosis; MAPK; Proteases/Proteasome
Tauroursodeoxycholate sodium (TUDC) 是一种内质网应激抑制剂。Tauroursodeoxycholate sodium (TUDC) 抑制ERK,显著降低凋亡分子表达,如caspase-3和caspase-12。
T16998 Tauroursodeoxycholate dihydrate

牛磺熊去氧胆酸二水合物,Taurolite dihydrate,TUDCA dihydrate,UR 906 dihydrate

ERK; Caspase Apoptosis; MAPK; Proteases/Proteasome
Tauroursodeoxycholate dihydrate is an endoplasmic reticulum stress inhibitor. Tauroursodeoxycholate also inhibits ERK. Tauroursodeoxycholate significantly decreases the expression of apoptosis molecules, such as caspase-3 and caspase-12.

化合物

Tauroursodeoxycholate sodium
Cat.No: T6993
Synonym: 牛磺熊脱氧胆酸钠,Sodium tauroursodeoxycholate,Tauroursodeoxycholic acid sodium salt,TUDC,牛磺熊去氧胆酸钠,Sodium Tauroursodeoxycholate (TUDC)
Target: Apoptosis, ERK, Caspase
Tauroursodeoxycholate dihydrate
Cat.No: T16998
Synonym: 牛磺熊去氧胆酸二水合物,Taurolite dihydrate,TUDCA dihydrate,UR 906 dihydrate
Target: ERK, Caspase
Cat. No. Product Name Target Signaling Pathways
T2532 Tauroursodeoxycholate

Taurolite,牛磺熊去氧胆酸,Tauroursodeoxycholic Acid,UR 906,Ursodeoxycholyltaurine,TUDCA

Apoptosis; ERK; P450; Caspase; Endogenous Metabolite Apoptosis; MAPK; Metabolism; Proteases/Proteasome
Tauroursodeoxycholate (UR 906),又称 ursodoxicoltaurine,是一种高度亲水性的三级胆汁酸,在人体内以低浓度产生。Tauroursodeoxycholate 是 ursodeoxycholic acid 更亲水的形式,而 ursodeoxycholic acid 是人类体内自然产生的更丰富的胆汁酸。Tauroursodeoxycholate 正在研究用于几种疾病,如原发性胆汁性肝硬化(PBC)、胰岛素抵抗、淀粉样变性、囊性纤维化、胆汁淤滞和肌萎缩性侧索硬化症。

天然产物

Tauroursodeoxycholate
Cat.No: T2532
Synonym: Taurolite,牛磺熊去氧胆酸,Tauroursodeoxycholic Acid,UR 906,Ursodeoxycholyltaurine,TUDCA
Target: Apoptosis, ERK, P450, Caspase, Endogenous Metabolite
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