5
1
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T16390 |
Omtriptolide
|
ERK | MAPK |
Omtriptolide, triptolide purified from the Chinese herb, is a water-soluble derivative prodrug. | |||
T33798 |
Omtriptolide sodium
YM-274,YM274,YM 274 |
||
Omtriptolide sodium is a biochemical. | |||
T12042 | Minnelide | Others | Others |
Minnelide is a prodrug of triptolide,and shows potent antitumor activity in a number of tumor types. | |||
T64111 | Antitumor agent-76 | ||
Antitumor agent-76 是一种水溶性的、口服具有活力的、快速释放的 Triptolide 前药,表现出抗癌效果。 | |||
T64128 | Antitumor agent-56 | ||
Antitumor agent-56 是一种口服具有活力的 triptolide 衍生物,能够明显抑制黑色素瘤的生长,表现出抗肿瘤、抗炎和 NO 释放作用。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2179 |
Triptolide
PG490,NSC 163062,雷公藤甲素 |
Apoptosis; Mdm2; HSP; NF-κB | Apoptosis; Cytoskeletal Signaling; Metabolism; NF-κB |
Triptolide (PG490) 属于三环二萜类天然产物,是一种 NF-κB 活化的抑制剂。Triptolide 具有免疫抑制、抗风湿、抗炎、抗增殖和抗肿瘤活性。 |