Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T80202 |
Tetrapeptide-1
|
Melanocortin Receptor | GPCR/G Protein; Neuroscience |
Tetrapeptide-1,一种生物活性肽,具抗氧化功能,已报道应用于化妆品成分。 | |||
T20494L |
Acetyl tetrapeptide-15 Acetate
Skinasensyl Acetate,Acetyl tetrapeptide-15 Acetate (928007-64-1 Free base) |
||
Acetyl tetrapeptide-15 Acetate (Skinasensyl Acetate) 是一种用于敏感皮肤的化妆品中的合成肽,是 endomorphin-2 衍生物, 通过内啡肽样通路扩大 μ-阿片受体中的神经元兴奋性阈值范围,可用于研究由皮肤高反应性产生的炎症性和神经性疼痛。 | |||
T20482L |
Acth (1-4) acetate(19405-50-6 free base)
|
Others | Others |
Acth (1-4) acetate(19405-50-6 free base) 是 ACTH N 端四肽。 | |||
T35689 |
MTP 131 acetate
|
Others | Others |
MTP 131 acetate 是一种小的线粒体靶向四肽。 | |||
T34734 |
Substance P (1-4)
SP(1-4) |
||
Substance P (1-4) is a substance P N-terminal tetrapeptide fragment. | |||
TP2354 |
Tetrapeptide-11
Pro-pro-tyr-leu |
||
Tetrapeptide-11 is the reaction product of Acetic Acid and tetrapeptide-11, containing leucine, proline, and tyrosine residues. It boosts cell growth, Syndecan-1, and Collagen XVII synthesis. Tetrapeptide-11 has a face and body anti-wrinkle and anti-aging | |||
T83197 |
Acetyl tetrapeptide-22
|
||
Acetyl tetrapeptide-2,生物活性肽,具修复肌肤功效,报道作为化妆品成分应用。 | |||
T20482 |
Acth (1-4)
(1-4) Corticotropin |
||
Acth (1-4) is the ACTH N-terminal tetrapeptide. | |||
T81006 |
Tetrapeptide-26
|
||
Tetrapeptide-26,一种生物活性肽,具抗衰老(anti-aging)功能,常用作化妆品成分。 | |||
T81564 |
Palmitoyl tetrapeptide-10
|
||
Palmitoyl tetrapeptide-10,一种生物活性肽,具有抗衰老功能,已报道用于化妆品成分。 | |||
T80628 |
Myristoyl tetrapeptide-12
|
TGF-beta/Smad | Stem Cells |
Myristoyl tetrapeptide-12 直接激活SMAD2,并促使SMAD3与DNA结合。该化合物能有效促进毛发,特别是睫毛的生长。 | |||
T36930 |
Palmitoyl Tetrapeptide-7 (acetate)
|
||
Palmitoyl tetrapeptide-7 is a cosmeceutical peptide that stimulates type I collagen, fibronectin, and hyaluronic acid production in skin.1Formulations containing palmitoyl tetrapeptide-7 have been used in the treatment of photoaging, dark circles, and undereye puffiness. 1.Bucay, V.W., and Day, D.Adjunctive skin care of the brow and periorbital regionClin. Plast. Surg.40(1)225-236(2013) | |||
T76247L |
AGPV TFA
|
||
AGPV TFA 是一种四肽,具有用于预防血吸虫寄生虫感染研究的潜力。 | |||
T81007 |
Tetrapeptide-21
|
||
Tetrapeptide-21为一种生物活性肽,具备抗皱功能,常作为化妆品成分使用。 | |||
T76247 |
AGPV
|
||
AGPV 是一种四肽,具有用于预防血吸虫寄生虫感染研究的潜力。 | |||
TP2147 |
LSKL, Inhibitor of Thrombospondin (TSP-1) (TFA)
|
Others | Others |
LSKL, Inhibitor of Thrombospondin (TSP-1) TFA, a latency-associated protein (LAP)-TGFβ derived tetrapeptide, is a competitive antagonist of TGF-β1. | |||
T81563 |
Palmitoyl tetrapeptide-20
PTP20 |
||
Palmitoyl tetrapeptide-20(PTP20)为具保护作用的生物活性肽,旨在维护滤泡黑素细胞,常用作化妆品配料。 | |||
T82780 |
Caprooyl-tetrapeptide-3 acetate
|
||
Caprooyl-tetrapeptide-3 acetate 旨在减少细纹与皱纹。该化合物能够在皮质激素诱导的皮肤老化模型中刺激VII型胶原蛋白及层粘连蛋白5的表达。 | |||
T80207 |
Tetrapeptide
|
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Tetrapeptide 作为α-MSH的类似物,能促进黑色素的合成;其通过降低活性氧化物质生成和提升DNA光产物修复效率,有效减轻DNA损伤。 | |||
T81005 |
Tetrapeptide-4
|
||
Tetrapeptide-4,一种护肤产品中常用的肽,具备减少皱纹与增强胶原蛋白、弹性蛋白及纤连蛋白的功能,展现出显著的抗衰老特性。 | |||
TP1014 |
Z-VRPR-FMK (TFA)
VRPR |
||
Z-VRPR-FMK (TFA) (VRPR) is a tetrapeptide and a selective and irreversible inhibitor of lymphoma translocation protein 1 (MALT1) in mucosa-associated lymphoid tissue. | |||
T76186 |
Tyr-W-MIF-1
|
||
Tyr-W-MIF-1 是一种阿片四肽,具有阿片和抗阿片活性。Tyr-W-MIF-1 可诱导镇痛。 | |||
T76589 |
H-Leu-Trp-Met-Arg-OH
|
||
H-Leu-Trp-Met-Arg-OH是一种四肽,可作为氨基肽酶(aminopeptidase)介导水解研究的底物。 | |||
T81186 |
SDGR
|
||
SDGR是一种四肽,含有Ser-Asp-Gly-Arg序列,能够有效抑制纤连蛋白介导的细胞附着。 | |||
T77993 |
Goralatide acetate
|
||
Goralatide为一种内源性四肽,作为造血生理调节剂。该化合物能够抑制原始造血细胞的增殖。 | |||
T76258 |
Tetrapeptide-30
|
||
Tetrapeptide-30为由四个氨基酸组成的亮肤肽,作用于酪氨酸酶抑制,通过减少酪氨酸酶数量及抑制黑色素细胞激活,以达到淡化色素沉着,均匀肤色之目的。 | |||
T82201 |
H-Gly-Pro-Arg-Pro-NH2
|
||
H-Gly-Pro-Arg-Pro-NH2 是模拟纤维蛋白原(N-末端Gly-Pro-Arg区域)的四肽,具有抑制纤维蛋白聚合的功能。 | |||
T75938 |
Z-VRPR-FMK TFA
|
||
Z-VRPR-FMK (TFA) (VRPR) 为一种四肽类选择性及不可逆的粘膜相关淋巴组织淋巴瘤易位蛋白1 (MALT1) 抑制剂,具有抵抗甲型流感病毒 (IAV) 感染的能力。 | |||
T82307 |
Glp-His-Pro-Gly-NH2
pGlu-His-Pro-Gly-NH2 |
||
pGlu-His-Pro-Gly-NH2(Glp-His-Pro-Gly-NH2)为含四氨基酸肽类化合物,可激发促性腺激素、黄体生成素(LH)与促卵泡激素(FSH)释放。 | |||
T35774 |
HC Toxin
|
||
HC Toxin is a cell-permeable, reversible inhibitor of histone deacetylases (HDACs) (IC50 = 30 nM). Through its effects on HDACs, HC toxin has been shown to up-regulate the expression of 15-lipoxygenase-1 in colorectal cancer cells and induce fetal hemoglobin in human primary erythroid cells. HC Toxin is a cyclic tetrapeptide first isolated from H. carbonum (now C. carbonum), a pathogen of maize. | |||
T76577 |
Antiulcer Agent 2
|
||
Antiulcer Agent 2 是一种四肽,组成包括天冬氨酸、丙氨酸、组氨酸和赖氨酸,存在于人白蛋白N端,并在溃疡及活性氧生成中显示出潜在应用。 | |||
T77888 |
Mal-PEG2-Gly-Gly-Phe-Gly-Exatecan
|
||
Mal-PEG2-Gly-Gly-Phe-Gly-Exatecan是一个ADC药物-linker偶联物,包含Exatecan和linker。该化合物主要用于ADC合成与癌症研究。 | |||
T77910 |
Patritumab deruxtecan
U3-1287,HER3-DXd |
||
Patritumab deruxtecan (HER3-DXd)为一抗体-药物偶联物(ADC),其结构为全人源IgG1单克隆抗体Patritumab通过含四肽的裂解性连接子与拓扑异构酶 I 抑制剂药效团相连。 | |||
T80882 |
Val-Gly-Ser-Glu
NSC 350591 |
||
Val-Gly-Ser-Glu (NSC 350591) 是一种ECF-A四肽。该化合物能剂量依赖性地提升人类嗜酸性粒细胞的数量,而不影响中性粒细胞的数量,并可与补体包被的绵羊红细胞(EAC3b)形成玫瑰花结。 | |||
T35993 |
Epitalon (acetate)
|
||
Epitalon is a synthetic tetrapeptide with anti-aging properties.1,2,3,4 Dietary administration of epitalon (0.00001% w/w) reduces levels of lipid peroxidation products in aged D. melanogaster tissue homogenates.1 Epitalon (1 μg/animal) delays age-related estrous shutdown and decreases the frequency of bone marrow cell chromosomal aberrations in female mice.2 It decreases spontaneous mammary gland and ovarian tumor development and metastasis in aged female mice.3 Epitalon also stimulates melatoni... | |||
T73852 | Ac-YVAD-CHO acetate | ||
Ac-YVAD-CHO(L-709049)醋酸盐是一种高效、可逆、特异的四肽白介素1β转化酶(ICE)抑制剂,小鼠和人类的Ki值分别为3.0 nM和0.76 nM。它同时也能抑制caspase-1,从而抑制成熟IL-lβ的产生。 | |||
T37199 |
Bilaid C
|
||
Bilaid C is a tetrapeptide μ-opioid receptor agonist (Ki= 210 nM in HEK293 cell membranes expressing the human receptor) that has been found inPenicillium.1It inhibits forskolin-induced cAMP accumulation by 77% in HEK293 cells expressing the human μ-opioid receptor when used at a concentration of 10 μM. Bilaid C induces inward rectifying potassium channel (Kir) currents in rat locus coeruleus slices that endogenously express high levels of the μ-opioid receptor (EC50= 4.2 μM). 1.Dekan, Z., Siana... | |||
T75536 | Koshidacin B | ||
Koshidacin B为针对疟原虫的环四肽类化合物,其针对抗疟原虫(P. falciparum) FCR3和K1系的IC50值分别为0.89 μM与0.83 μM。此化合物在体内能有效抑制疟原虫,适用于疟疾感染的科学研究。 | |||
T41146 |
ND1-YL2
ND1-YL2 |
||
ND1-YL2 is a peptide-based PROTAC®Degrader of steroid receptor co-activator 1 (SRC-1; also known as nuclear receptor coactivator 1, NCOA1). ND1-YL2 is composed of a stapled peptide that binds SRC-1 (YL2) joined by a linker to a tetrapeptide that binds UBR box domains. Upon ternary complex formation, SRC-1 is polyubiquitinated and subsequently degraded via the N-degron pathway. This Degrader induces dose-dependent degradation of SRC-1 in the MDA-MB-231 triple negative breast cancer cell line (DC5... | |||
T80735 |
Z-Gly-Pro-Phe-Leu-CHO
Z-GPFL-CHO |
Proteasome | Proteases/Proteasome; Ubiquitination |
Z-Gly-Pro-Phe-Leu-CHO(Z-GPFL-CHO)是一种具有高选择性和高效率的四肽醛类蛋白酶体抑制剂,优先抑制支链氨基酸(Ki为1.5 µM),对小中性氨基酸的Ki值为2.3 µM,胰凝乳蛋白酶样活性的Ki值为40.5 µM,对肽基-谷氨酰肽水解活性的IC50为3.1 µM。 | |||
T35582 |
H-Arg-Gly-Asp-Cys-OH (trifluoroacetate salt)
|
||
H-Arg-Gly-Asp-Cys-OH is a tetrapeptide that contains the arginine-glycine-aspartate (RGD) motif, a sequence that acts as a recognition site for various adhesion proteins.1It inhibits the binding of fibrinogen to endothelial cells and ADP-stimulated platelets with IC50values of 320 and 35 μM, respectively.2Implantation of titanium rods coated with H-Arg-Gly-Asp-Cys-OH increases bone formation in rat femurs.3H-Arg-Gly-Asp-Cys-OH has been conjugated to polyethylenimine to improve gene transfection ... |