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Cat. No. Product Name Target Signaling Pathways
T3962 TPI-1

TPI 1,TPI1

Phosphatase; Glucocorticoid Receptor Endocrinology/Hormones; Metabolism
TPI-1 是一种 SHP-1的抑制剂,其 IC50=40 nM。
T34910 TPI-1917-49

TPI 1917 49

TPI-1917-49 is a promising amyloid reducing agent that works by reducing Aβ levels.
T68570 TPI-287

TPI 287 is a synthetic, third generation taxane with potential antineoplastic activity. TPI 287 binds to tubulin and stabilizes microtubules, resulting in inhibition of microtubule assembly/disassembly dynamics, cell cycle arrest at the G2/M phase, and apoptosis.
T8673 FMOC-L-1,2,3,4-TETRAHYDRONORHARMAN-3-CAR

Fmoc-Tpi-OH,FMOC-L-1,2,3,4-四氢-Β-咔啉-3-羧酸

Others Others
FMOC-L-1,2,3,4-TETRAHYDRONORHARMAN-3-CAR (Fmoc-Tpi-OH) 是THN 的衍生物。
T8140 Tianeptine

噻萘普汀,S-1574,JNJ-39823277,Tianeptine sodium,噻奈普汀,TPI-1062

5-HT Receptor GPCR/G Protein; Neuroscience
Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。
T3658 Trifluridine/tipiracil hydrochloride mixture

Trifluridine-tipiracil hydrochloride mixture,TAS102,TAS-102,TAS 102

Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Trifluridine/tipiracil hydrochloride mixture (TAS-102) 是一种新型口服组合药物,含有摩尔比为 2:1 的曲氟尿苷(TFT) 和盐酸替吡嘧啶 (TTP)。它主要通过抑制胸苷酸合酶 (TS) 和掺入 DNA 来显示抗肿瘤活性。
T8732 CTPI-2

Others; Mitochondrial Metabolism Metabolism; Others
CTPI-2 是一种特异性线粒体柠檬酸盐载体SLC25A1抑制剂,KD=3.5 μM,具有抗肿瘤作用。它能够抑制糖酵解、PPARγ 及其下游靶点葡萄糖转运蛋白 GLUT4。它阻断非酒精性脂肪性肝炎逆转脂肪变性的显著改变,防止演变为脂肪性肝炎,减少肝脏和脂肪组织中炎性巨噬细胞的浸润,并显著减轻由高脂肪饮食引起的肥胖。
T2366 Tipiracil hydrochloride

MA-1 hydrochloride,盐酸替吡嘧啶

Nucleoside Antimetabolite/Analog Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Tipiracil hydrochloride (MA-1 hydrochloride) 是一种胸苷磷酸化酶抑制剂,是抗癌候选药物 TAS-102 中的活性成分之一,用于癌症研究。
T76154 Triosephosphate isomerase

Triosephosphate isomerase (TPI) 是一种能够在糖酵解过程中快速转换磷酸二羟丙酮(dihydroxyacetone phosphate)与D: -甘油醛-3-磷酸(D: -glyceraldehyde-3-phosphate)的酶。其催化位点位于酶的二聚体界面。

化合物

TPI-1
Cat.No: T3962
Synonym: TPI 1,TPI1
Target: Phosphatase, Glucocorticoid Receptor
TPI-1917-49
Cat.No: T34910
Synonym: TPI 1917 49
Target:
TPI-287
Cat.No: T68570
Synonym:
Target:
FMOC-L-1,2,3,4-TETRAHYDRONORHARMAN-3-CAR
Cat.No: T8673
Synonym: Fmoc-Tpi-OH,FMOC-L-1,2,3,4-四氢-Β-咔啉-3-羧酸
Target: Others
Tianeptine
Cat.No: T8140
Synonym: 噻萘普汀,S-1574,JNJ-39823277,Tianeptine sodium,噻奈普汀,TPI-1062
Target: 5-HT Receptor
Trifluridine/tipiracil hydrochloride mixture
Cat.No: T3658
Synonym: Trifluridine-tipiracil hydrochloride mixture,TAS102,TAS-102,TAS 102
Target: Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis
CTPI-2
Cat.No: T8732
Synonym:
Target: Others, Mitochondrial Metabolism
Tipiracil hydrochloride
Cat.No: T2366
Synonym: MA-1 hydrochloride,盐酸替吡嘧啶
Target: Nucleoside Antimetabolite/Analog
Triosephosphate isomerase
Cat.No: T76154
Synonym:
Target:
TargetMol Loading
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