Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3962 |
TPI-1
TPI 1,TPI1 |
Phosphatase; Glucocorticoid Receptor | Endocrinology/Hormones; Metabolism |
TPI-1 是一种 SHP-1的抑制剂,其 IC50=40 nM。 | |||
T34910 |
TPI-1917-49
TPI 1917 49 |
||
TPI-1917-49 is a promising amyloid reducing agent that works by reducing Aβ levels. | |||
T68570 | TPI-287 | ||
TPI 287 is a synthetic, third generation taxane with potential antineoplastic activity. TPI 287 binds to tubulin and stabilizes microtubules, resulting in inhibition of microtubule assembly/disassembly dynamics, cell cycle arrest at the G2/M phase, and apoptosis. | |||
T8673 |
FMOC-L-1,2,3,4-TETRAHYDRONORHARMAN-3-CAR
Fmoc-Tpi-OH,FMOC-L-1,2,3,4-四氢-Β-咔啉-3-羧酸 |
Others | Others |
FMOC-L-1,2,3,4-TETRAHYDRONORHARMAN-3-CAR (Fmoc-Tpi-OH) 是THN 的衍生物。 | |||
T8140 |
Tianeptine
噻萘普汀,S-1574,JNJ-39823277,Tianeptine sodium,噻奈普汀,TPI-1062 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。 | |||
T3658 |
Trifluridine/tipiracil hydrochloride mixture
Trifluridine-tipiracil hydrochloride mixture,TAS102,TAS-102,TAS 102 |
Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Trifluridine/tipiracil hydrochloride mixture (TAS-102) 是一种新型口服组合药物,含有摩尔比为 2:1 的曲氟尿苷(TFT) 和盐酸替吡嘧啶 (TTP)。它主要通过抑制胸苷酸合酶 (TS) 和掺入 DNA 来显示抗肿瘤活性。 | |||
T8732 |
CTPI-2
|
Others; Mitochondrial Metabolism | Metabolism; Others |
CTPI-2 是一种特异性线粒体柠檬酸盐载体SLC25A1抑制剂,KD=3.5 μM,具有抗肿瘤作用。它能够抑制糖酵解、PPARγ 及其下游靶点葡萄糖转运蛋白 GLUT4。它阻断非酒精性脂肪性肝炎逆转脂肪变性的显著改变,防止演变为脂肪性肝炎,减少肝脏和脂肪组织中炎性巨噬细胞的浸润,并显著减轻由高脂肪饮食引起的肥胖。 | |||
T2366 |
Tipiracil hydrochloride
MA-1 hydrochloride,盐酸替吡嘧啶 |
Nucleoside Antimetabolite/Analog | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Tipiracil hydrochloride (MA-1 hydrochloride) 是一种胸苷磷酸化酶抑制剂,是抗癌候选药物 TAS-102 中的活性成分之一,用于癌症研究。 | |||
T76154 | Triosephosphate isomerase | ||
Triosephosphate isomerase (TPI) 是一种能够在糖酵解过程中快速转换磷酸二羟丙酮(dihydroxyacetone phosphate)与D: -甘油醛-3-磷酸(D: -glyceraldehyde-3-phosphate)的酶。其催化位点位于酶的二聚体界面。 |