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Cat. No.	Product Name	Target	Signaling Pathways
T20789	S-23 (S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide,S23	Androgen Receptor	Endocrinology/Hormones
	S-23 ((S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide) 是口服选择性雄激素受体调节剂(Ki:1.7 nM)。它能够诱导 CV-1 细胞雄激素受体介导的转录激活，提高去势大鼠前列腺、精囊和肛提肌重量。
T8457	NPS2390	GluR	Neuroscience
	NPS2390 是钙敏感受体抑制剂，也是 mGluR1 和 mGluR5 的非竞争性拮抗剂。
T60002	DC-S239	Histone Methyltransferase	Chromatin/Epigenetic
	DC-S239 (DC-S239) 是一种选择性的组蛋白甲基转移酶 SETD7 抑制剂 (IC50 = 4.59 μM)，具有抗癌活性。
T30176	ASS234 AS S234,AS-S234
	ASS234 is a multi-target propylamine used in the treatment of Alzheimer's disease.
T70345	JAS239
	JAS239 is a novel carbocyanine dye that binds and competitively inhibits choline kinase (ChoK) intracellularly. JAS239 attenuated choline phosphorylation and viability in a panel of human breast cancer cell lines. Antibody blockade prevented cellular retention of JAS239 indicating direct interaction with ChoKα independent of the choline transporters and catabolic choline pathways. In mice bearing orthotopic MCF7 breast xenografts, optical imaging with JAS239 distinguished tumors overexpressing C...
T82158	Human IgG1 (S239D/I332E) kappa, Isotype Control
	HumanIgG1(S239D/I332E) kappa, Isotype Control为一种人源-鼠源嵌合型单克隆抗体，作为HumanIgG1(S239D/I332E)κ抗体之同型对照物。
T62532	MRS2395
	MRS2395 是一种二戊酰衍生物，是一种 P2Y12 受体的有效拮抗剂。MRS2395 抑制 ADP 诱导的血小板活化 (Ki: 3.6 μM)。MRS2395 在 PGE1 存在下，对大鼠血小板中 ADP 诱导的 cAMP 具有抑制作用 (IC50: 7 μM)。MRS2395 增强血小板致密颗粒释放以响应 TRAP-6。
T34473	S2366 HCl S2366 hydrochloride,S 2366,S-2366,S2366
	S 2366 is a chromogenic substrate for Factor XI in plasma.
T25084	AM-TS23 AM TS23
	AM-TS23 is used as a DNA polymerase lambda and beta inhibitor.
T26171	S23757 S-23757,S 23757
	S23757 is an imidazoline 1 receptor (I1R) selective ligand.
T68613	DC-S238
	DC-S238 is a potent and selective histone methyltransferase SET7 inhibitor.