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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T0245 RS 61443

RS61443,吗替麦考酚酯,Mycophenolate mofetil,TM-MMF

Dehydrogenase Metabolism
RS 61443 (Mycophenolate mofetil) 是一种免疫抑制剂,一种非竞争性、选择性和可逆的肌苷一磷酸脱氢酶 (IMPDH) 抑制剂。
T23035 Mycophenolate mofetil hydrochloride

Others Others
Mycophenolate Mofetil is a non-competitive, selective, and reversible inhibitor of inosine monophosphate dehydrogenase I/II (IC50: 39 nM and 27 nM, respectively).

化合物

RS 61443
Cat.No: T0245
Synonym: RS61443,吗替麦考酚酯,Mycophenolate mofetil,TM-MMF
Target: Dehydrogenase
Mycophenolate mofetil hydrochloride
Cat.No: T23035
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T6293 Mycophenolate Mofetil

TM-MMF,吗替麦考酚酯,RS 61443

Apoptosis; Dehydrogenase; Drug Metabolite Apoptosis; Metabolism
Mycophenolate Mofetil (TM-MMF) 是 Mycophenolic acid 的吗啉乙酯前药。它通过抑制肌苷一磷酸脱氢酶抑制从头嘌呤合成,显示出选择性淋巴细胞抗增殖作用。
T1335 Mycophenolic acid

霉酚酸,Mycophenolate,RS-61443

Apoptosis; Dehydrogenase; Endogenous Metabolite; Antibacterial; Antibiotic; UGT; Antifungal Apoptosis; Metabolism; Microbiology/Virology
Mycophenolic acid (Mycophenolate) 是一种有效的非竞争性肌苷单磷酸脱氢酶 (IMPDH) 抑制剂,EC50为 0.24 µM。它对多种 RNA 病毒具有抗病毒作用。它也是一种免疫抑制剂,具有抗血管生成和抗肿瘤作用。

天然产物

Mycophenolate Mofetil
Cat.No: T6293
Synonym: TM-MMF,吗替麦考酚酯,RS 61443
Target: Apoptosis, Dehydrogenase, Drug Metabolite
Mycophenolic acid
Cat.No: T1335
Synonym: 霉酚酸,Mycophenolate,RS-61443
Target: Apoptosis, Dehydrogenase, Endogenous Metabolite, Antibacterial, Antibiotic, UGT, Antifungal
TargetMol Loading
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