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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T63637 ROCK-IN-4

ROCK-IN-4ROCK 的有效抑制剂,可维持 NO 释放能力。ROCK-IN-4 能够可逆地解聚 F-肌动蛋白,并阻碍人小梁网 (HTM) 细胞的线粒体呼吸。ROCK-IN-4 能够用于研究青光眼或高眼压。
T79809 ROCK-IN-8

ROCK Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells
ROCK-IN-8 (Example 4) 是ROCK抑制剂,IC50值不足100 nM,并显示出抗炎活性,适用于呼吸系统和胃肠道疾病的研究。
T37847 Zonisamide-13C2,15N

Zonisamide-13C2,15N

Zonisamide-13C2,15N is intended for use as an internal standard for the quantification of zonisamide by GC- or LC-MS. Zonisamide is an antiepileptic agent.1 It selectively inhibits the repeated firing of sodium channels (IC50 = 2 μg/ml) in mouse embryo spinal cord neurons and inhibits spontaneous channel firing when used at concentrations greater than 10 μg/ml.2 In rat cerebral cortex neurons, zonisamide (1-1,000 μM) inhibits T-type calcium channels with a maximum reduction of 60% of the calcium...

化合物

ROCK-IN-4
Cat.No: T63637
Synonym:
Target:
ROCK-IN-8
Cat.No: T79809
Synonym:
Target: ROCK
Zonisamide-13C2,15N
Cat.No: T37847
Synonym: Zonisamide-13C2,15N
Target:
Cat. No. Product Name Target Signaling Pathways
T4S1962 beta-Asarone

β-细辛脑,(Z)-1,2,4-三甲氧基-5-丙烯基苯;顺式细辛脑,Cis-Isoasarone,Cis-Asarone,Cis-Isoelemicin

NF-κB; JNK MAPK; NF-κB
beta-Asarone (Cis-Isoelemicin) 是一种石菖蒲中的主要成分,具有免疫抑制、促进安定、中枢神经系统抑制、降温等功能。它可透过血脑屏障,能够预防帕金森病。
T5S0053 Coptisine

黄连碱,Coptisin

Indoleamine 2,3-Dioxygenase (IDO) Metabolism
Coptisine (Coptisin) 是一种从黄连中分离到的生物碱,是非竞争性的IDO 抑制剂,Ki=为 5.8 μM,IC50=6.3 μM。

天然产物

beta-Asarone
Cat.No: T4S1962
Synonym: β-细辛脑,(Z)-1,2,4-三甲氧基-5-丙烯基苯;顺式细辛脑,Cis-Isoasarone,Cis-Asarone,Cis-Isoelemicin
Target: NF-κB, JNK
Coptisine
Cat.No: T5S0053
Synonym: 黄连碱,Coptisin
Target: Indoleamine 2,3-Dioxygenase (IDO)
TargetMol Loading
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