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抑制剂 & 化合物

1

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Cat. No. Product Name Target Signaling Pathways
T12598 Pz-1

VEGFR; c-RET Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
Pz-1 是 VEGFR2 和 RET 酪氨酸激酶的抑制剂,可阻断 RET 刺激生长所需的血液供应。
T81336 PZ-1190

Dopamine Receptor GPCR/G Protein; Neuroscience
PZ-1190是一种多靶点配体,针对啮齿动物的serotonin和dopamine受体,展现出潜在的抗精神病活性。
T81335 PZ-1922

5-HT Receptor GPCR/G Protein; Neuroscience
PZ-1922(Compound 16),是能穿透大脑屏障的5-HT6R/5-HT3R拮抗剂,其Ki值分别为17 nM和0.45 nM。该化合物还能可逆地抑制MAO-B(pIC50:8.93)。在大鼠的新物体识别(NOR)测试中,PZ-1922逆转了Scopolamine (SCOP)诱导的记忆缺陷;同样,在T迷宫测试中,它防止了Aβ诱发的记忆衰退。

化合物

Pz-1
Cat.No: T12598
Synonym:
Target: VEGFR, c-RET
PZ-1190
Cat.No: T81336
Synonym:
Target: Dopamine Receptor
PZ-1922
Cat.No: T81335
Synonym:
Target: 5-HT Receptor
Cat. No. Product Name Target Signaling Pathways
T37442 Aspergillin PZ

Aspergillin PZ is a fungal metabolite originally isolated from A. awamori. It induces morphological deformation of P. oryzae conidia when used at a concentration of 89 nM. Aspergillin PZ is active against S. epidermidis (MIC = 20 μM) but not S. aureus, E. coli, or B. cereus (MICs = >20 μM). It is cytotoxic to HL-60 promyelocytic leukemia cells (IC50 = 56.61 μM) but not THP-1 acute monocytic leukemia or PC3 prostate cancer cells (IC50s = >80 μM).

天然产物

Aspergillin PZ
Cat.No: T37442
Synonym:
Target:
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