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Cat. No. Product Name Target Signaling Pathways
T6250 H-89 dihydrochloride

Protein kinase inhibitor H-89 dihydrochloride,H 89 2HCl,5-Isoquinolinesulfonamide

PKA; S6 Kinase; Autophagy Autophagy; MAPK; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
H-89 dihydrochloride (5-Isoquinolinesulfonamide) 是一种选择性 cAMP 依赖性蛋白激酶A(PKA) 抑制剂,IC50值为 48 nM。也可轻微抑制 PKG、PKC 和酪蛋白激酶活性。
T11524 H-89

Protein kinase inhibitor H-89

Others Others
H-89 is a selective inhibitor of cyclic AMP-dependent protein kinase (protein kinase A; IC50: 48 nM). H-89 has weak inhibition on PKG, Casein Kinase, PKC, and other kinases.

化合物

H-89 dihydrochloride
Cat.No: T6250
Synonym: Protein kinase inhibitor H-89 dihydrochloride,H 89 2HCl,5-Isoquinolinesulfonamide
Target: PKA, S6 Kinase, Autophagy
H-89
Cat.No: T11524
Synonym: Protein kinase inhibitor H-89
Target: Others
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