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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0453L |
DL-Phenylephrine HCl
Eyelo,DL-Phenylephrine hydrochloride |
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DL-Phenylephrine HCl is a selective agonist of the alpha1-adrenergic receptor. | |||
T23557 |
Talibegron hydrochloride
ZD2079 hydrochloride,ZD 2079 |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Talibegron hydrochloride (ZD2079 hydrochloride) 是一种β3肾上腺素能受体激动剂,对苯肾上腺素预收缩大鼠肠系膜动脉的 pD2为3.72。松弛大鼠肠系膜动脉和离体主动脉。在体内抑制瘦小鼠 ob 基因表达和循环瘦素水平。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0453 |
Phenylephrine hydrochloride
NCI-c55641,Phenylephrine HCl,盐酸去氧肾上腺素,(R)-(-)-Phenylephrine hydrochloride |
Endogenous Metabolite; Adrenergic Receptor | GPCR/G Protein; Metabolism; Neuroscience |
Phenylephrine hydrochloride (NCI-c55641) 是选择性的α1-肾上腺素能受体激动剂,对α1A,α1B 和α1D 受体的pKis 分为4.70,4.87和5.86。 | |||
TN1724 |
Harmalol hydrochloride
Harmidol hydrochloride |
P450; Antioxidant | Metabolism; oxidation-reduction |
Harmalol hydrochloride (Harmidol hydrochloride) 是一种可从Peganum harmala L.的种子中提取出来的β-咔啉生物碱。Harmalol hydrochloride 是Harmaline 的主要代谢产物,在转录和翻译后水平上显著抑制二恶英介导的 CYP1A1 诱导。Harmalol hydrochloride 在去氧肾上腺素或KCl 预先收缩的分离大鼠胸主动脉制剂中显示出血管松弛活性。 Harmalol hydrochloride 具有抗氧化活性. |