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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T19950 Paliperidone Palmitate

RO 92670,RO92670,RO-92670

Paliperidone is a dopamine antagonist and 5-HT2A antagonist of the atypical antipsychotic class of medications. Paliperidone has an antagonist effect at α1 and α2 adrenergic receptors and at H1 histamine receptors. In addition, it binds with dopamine and

化合物

Paliperidone Palmitate
Cat.No: T19950
Synonym: RO 92670,RO92670,RO-92670
Target:
Cat. No. Product Name Target Signaling Pathways
T0076 Paliperidone

9-羟基利培酮,帕潘立酮,9-hydroxyrisperidone

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Paliperidone (9-hydroxyrisperidone) 是 Risperidone 的主要活性代谢产物,是多巴胺 D2 拮抗剂和5-HT2A 拮抗剂。它用作非典型抗精神病药,用于精神分裂症的急性及维持治疗。它对α1和α2肾上腺素能受体和 H1组胺能受体也有拮抗作用。

天然产物

Paliperidone
Cat.No: T0076
Synonym: 9-羟基利培酮,帕潘立酮,9-hydroxyrisperidone
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
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