首页 工具
登录
购物车

搜索结果

Search Results for " pk 26124 "

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T0349 Riluzole

PK 26124,RP-54274,利鲁唑

GABA Receptor; Sodium Channel; NMDAR Membrane transporter/Ion channel; Neuroscience
Riluzole (RP-54274) 是一种谷氨酸拮抗剂,用作抗惊厥药并延长肌萎缩侧索硬化症患者的生存期。它还抑制 GABA 摄取,IC50值为 43 μM。
T37608 Riluzole-13C,15N2

Riluzole-13C,15N2

Riluzole-13C,15N2 is intended for use as an internal standard for the quantification of riluzole by GC- or LC-MS. Riluzole is a benzothiazole derivative with anti-excitotoxic effects that acts by blocking the presynaptic release of glutamate, indirectly antagonizing glutamate receptors, and inactivating neuronal voltage-gated Na+ channels (ED50 = 2.3 μM). Riluzole suppresses glutamate-induced seizures in rats at an ED50 value of 3.2 mg/kg and displays neuroprotective effects in hypoxic animals a...
T41265 Riluzole hydrochloride

Riluzole hydrochloride 是一种抗惊厥药物,属于依赖于使用的钠通道阻滞剂家族,也可以抑制 GABA 摄取,IC50值为 43 μM。

化合物

Riluzole
Cat.No: T0349
Synonym: PK 26124,RP-54274,利鲁唑
Target: GABA Receptor, Sodium Channel, NMDAR
Riluzole-13C,15N2
Cat.No: T37608
Synonym: Riluzole-13C,15N2
Target:
Riluzole hydrochloride
Cat.No: T41265
Synonym:
Target:
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼