Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6206 |
PHA-767491
CAY10572,PHA767491,PHA 767491 |
cholecystokinin; GSK-3; CDK | Cell Cycle/Checkpoint; GPCR/G Protein; PI3K/Akt/mTOR signaling; Stem Cells |
PHA-767491 (CAY10572) 是一种有效的 ATP 竞争性双重 Cdc7/CDK9 抑制剂,IC50 分别为 10 nM 和 34 nM。 | |||
T6940 |
PHA-767491 hydrochloride
CAY10572,PHA-767491,PHA767491 HCl,CAY-10572 hydrochloride |
Apoptosis; GSK-3; CDK | Apoptosis; Cell Cycle/Checkpoint; PI3K/Akt/mTOR signaling; Stem Cells |
PHA-767491 hydrochloride (CAY-10572 hydrochloride) 是一种Cdc7-Dbf4(DDK)/Cdk9的双重抑制剂,IC50值分别为 10 nM 和 34 nM。 |