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Search Results for " oxytocin "

73

抑制剂 & 化合物

4

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T21534L	Oxytocin C-terminal tripeptide Acetate Oxytocin C-terminal tripeptide Acetate(2002-44-0 Free base)	Others	Others
	Oxytocin C-terminal tripeptide Acetate 是 Oxytocin 的 C-末端三肽。Oxytocin 是哺乳动物的神经垂体激素，催产素受体的配体。
T40756	[Asp5]-Oxytocin [Asp5]-Oxytocin
	[Asp5]-Oxytocin is the first 5-position neurohypophyseal hormone analogue possessing significant biological activity.
T40536	[Glu4]-Oxytocin [Glu4]-Oxytocin
	[Glu4]-Oxytocin is a suitable derivative of oxytocin for conducting a thorough investigation, utilizing various methods, into the conformation of "oxytocin-like" molecules in aqueous solution.
T40534	[Leu3]-Oxytocin [Leu3]-Oxytocin
	[Leu3]-Oxytocin, an oxytocin analogue, is a derivative of oxytocin wherein the leucine amino acid (Leu) has been substituted at the 3rd position in the sequence.
T40658	[D-Asn5]-Oxytocin [D-Asn5]-Oxytocin
	[D-Asn5]-Oxytocin exhibits minimal specific oxytocic and vasodepressor effects. Comparative cumulative dose-response investigations reveal that [D-Asn5]-Oxytocin demonstrates a similar intrinsic activity to oxytocin in terms of oxytocic activity.
T33850	Oxytocin, deamino-6-carba- Deamino-6-carbaoxytocin,beta-Deaminocystathionine-oxytocin
	Deamino-6-carba-oxytoxin (dC60), a potent oxytocin analog considered to be resistant to some of the physiologically significant enzymic systems.
T39420	Oxytocin antiparallel dimer
	Oxytocin antiparallel dimer is the disulfide-bridged homo peptide dimer.
T39388	Oxytocin parallel dimer
	Oxytocin parallel dimer is the disulfide-bridged homo peptide dimer.
T40528	Oxytocin free acid 9-Deamidooxytocin
	Oxytocin free acid, also known as 9-Deamidooxytocin, is an analog of oxytocin where the glycinamide residue at position 9 has been substituted with a glycine residue. Oxytocin, a pleiotropic peptide hormone, has wide-ranging implications for general health, adaptation, development, reproduction, and social behavior.
T33849	Oxytocin, deamino-1-carba- Deamino-1-carbaoxytocin
	Oxytocin, deamino-1-carba- is a biochemical.
T80136	Val9-Oxytocin	Vasopressin Receptor	GPCR/G Protein
	Val9-Oxytocin为完全抗拮抗加压素(1a)受体的化合物，其结构上是Oxytocin的衍生物，特点在于Gly9位点被Val9取代。
T76624	(Ile8)-Oxytocin
	(Ile8)-Oxytocin 是一种神经垂体激素间催产素，在有袋动物中产生。
T12331L	OT-R antagonist 1 Oxytocin receptor antagonist 1	Others	Others
	OT-R antagonist 1 inhibits oxytocin-evoked intracellular Ca2+ mobilization (IC50 = 8 nM). OT-R antagonist 1 is a new effective and selective nonpeptide low molecular weight OT-R antagonist.
T12331	OT-R antagonist 2 Oxytocin receptor antagonist 2	Others	Others
	OT-R antagonist 2 is a nonpeptide low molecular weight antagonist of OT-R .
T80133	Pro8-Oxytocin	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Pro8-Oxytocin是一种改良的OXT配体。在灵长类动物OXTR中，Pro8-Oxytocin比标准哺乳动物OXT配体Leu8-Oxytocin诱发更强效的反应和显著的行为影响。相较于Vasopressin (AVP)，Pro8-Oxytocin对人类AVPR1a的活性较低，但对狨猴AVPR1a的激活作用则高于AVP。
T76211	[Asp5]-Oxytocin acetate
	[Asp5]-Oxytocin acetate 是一款功能强大的5位 (5-position) 神经垂体激素类似物，能引发体外大鼠子宫收缩，其效果可被 Mg2+ 增强。此化合物展现出在大鼠子宫收缩、禽血管抑制及大鼠抗利尿作用方面的活性。
T4996	Atosiban 阿托西班,RWJ22164,RW22164	Oxytocin Receptor; Vasopressin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Atosiban (RW22164) 是一种脱氨基催产素类似物，是一种九肽，也是竞争性的催产素受体拮抗剂。它是一种宫缩抑制剂，可用于自发早产的研究。
T76629	(Phe2,Orn8)-Oxytocin
	'(Phe2,Orn8)-Oxytocin' 作为选择性 V1 加压素激动剂，具有引发兔附睾持续收缩的功能，其EC50值达280 nM。
T76265	(Thr4,Gly7)-Oxytocin
	(Thr4,Gly7)-Oxytocin，一种Oxytocin类似物，特异性激活OT受体。通过激活TRPV1通道及抑制K+通道，诱导眼下神经元兴奋。
T80140	(Val3,Pro8)-Oxytocin	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	"(Val3,Pro8)-Oxytocin"为Gq依赖性途径的激动剂，同时作为β-arrestin结合及催产素受体（OXTR）内化作用的次级激动剂。
T80134	Pro8-Oxytocin TFA	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Pro8-Oxytocin TFA 作为一种优化的OXT配体，在灵长类动物OXTR上展现出较Leu8-Oxytocin更强的功能反应和行为效应。相对于AVP，在人类AVPR1a上的活性较低，但在狨猴AVPR1a上则显示出更高的活性。
T78021	Oxytocin parallel dimer TFA
	Oxytocin parallel dimer TFA为具有催产素和加压素样活性的二硫键桥连同肽二聚体，其毒性低于催产素。
T81583	Oxytocin antiparallel dimer TFA
	Oxytocin antiparallel dimer TFA为一种通过二硫键桥联形成的同肽二聚体。该化合物展现出催产素和加压素样的生物活性，同时具有低于催产素的毒性。
T76630	(Phe2,Orn8)-Oxytocin acetate
	(Phe2,Orn8)-Oxytocin acetate 是一种选择性 V1 加压素 (V1 vasopressin) 激动剂，能诱导兔附睾持续收缩，其EC50值为 280 nM。
T5148	Atosiban acetate RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164,醋酸阿托西班	Oxytocin Receptor; Vasopressin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Atosiban acetate (RW22164) 是一种脱氨基催产素类似物，是一种九肽，也是竞争性的催产素受体拮抗剂。它是一种宫缩抑制剂，可用于自发早产的研究。
T11857	LIT-001	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	LIT-001 是非肽类催产素受体激动剂，EC50为55 nM，Ki 为226 nM。它可改善孤独症小鼠模型的社交互动。
T80126	(d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	'(d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin (OVT)' 是催产素受体的一种拮抗剂，主要应用于神经系统疾病的研究领域。
T7601L	Carbetocin acetate 醋酸卡贝缩宫素,Carbetocin acetate(37025-55-1 free base),卡贝缩宫素醋酸盐	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Carbetocin acetate 是催产素类似物，是催产素受体激动剂，Ki 是 7.1 nM。它对催产素受体的嵌合 N 末端具有高亲和力，Ki 为 1.17 μM。它能透过血脑屏障，可以通过激活 CNS 中的催产素受体而具有类抗抑郁活性，具有用于产后出血的研究潜力。
T7601	Carbetocin 卡贝缩宫素,醋酸卡贝缩宫素	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Carbetocin 是催产素类似物，是催产素受体激动剂，Ki 是 7.1 nM。它对催产素受体的嵌合 N 末端具有高亲和力，Ki 为 1.17 μM。它能透过血脑屏障，可以通过激活 CNS 中的催产素受体而具有类抗抑郁活性，具有用于产后出血的研究潜力。
T76049	Demoxytocin
	Demoxytocin为一种异源性环肽，属于催产素类似物。其通过影响细胞膜通透性，提升平滑肌细胞内钙离子含量，进而加强平滑肌细胞收缩力，具备刺激子宫平滑肌收缩的能力，发挥催产素功能。此外，Demoxytocin在研究早产破裂引发的分娩刺激中有应用。
T37694	N-Acetyloxytocin
	N-Acetyloxytocin, a chemical compound, has been identified and analyzed in the neurointermediate lobe of the rat pituitary (NIL). Furthermore, its presence has also been detected in various brain regions of the rat[1].
T3347	PF3274167 PF 3274167,Cligosiban,PF-3274167	OX Receptor	GPCR/G Protein; Neuroscience
	PF3274167 (Cligosiban) 是一种有效的、选择性的、高亲和力的非肽催产素受体拮抗剂。
T28855	SSR126768A SSR-126768A,SSR 126768A	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	SSR126768A 是一种新型且具有选择性、口服活性和有效性的催产素(OT)受体拮抗剂，对子宫收缩有抑制作用，可用于预防早产。
TP1400L	[Arg8]-Vasotocin acetate（113-80-4 free base)	Others	Others
	[Arg8]-Vasotocin acetate（113-80-4 free base) 是一种存在于非哺乳动物脊椎动物神经垂体中的激素，与加压素和催产素有关。
T15682	L-371,257	Oxytocin Receptor; Vasopressin Receptor	Endocrinology/Hormones; GPCR/G Protein
	L-371,257 是催产素受体的竞争性拮抗剂，pA2 为 8.4，Ki 为 19 nM。 L-371,257 对加压素受体 1a 的 Ki 值为 3.7 nM。
TP2082L	d[Cha4]-AVP acetate(500170-27-4 free base)	Vasopressin Receptor	GPCR/G Protein
	d[Cha4]-AVP acetate(500170-27-4 free base) 是一种有效的选择性人血管加压素 V1B 受体激动剂（V1B、V1A、催产素和 V2 受体的 Ki 值分别为 1.2、151、240 和 750 nM）。刺激 ACTH 和皮质酮分泌，并在体内表现出微不足道的血管加压活性。
T16736	Retosiban GSK 221149,GSK 221149A	Others	Others
	Retosiban is an effective and selective oxytocin antagonist (Ki: 0.65 nM).
T23441	TC OT 39	Others	Others
	oxytocin receptor partial agonist
T24286	L 364918 L364,918,L-364918,L-364,918,L 364,918,L364918
	L 364918 is an oxytocin antagonist.
T23528	WAY-267464	Others	Others
	oxytocin receptor (OTR) agonist
T27763	L-366509 L 366,509,L 366509,L366,509,L-366,509
	L-366,509 is an antagonist of oxytocin.
T11502	Epelsiban GSK 557296	Others	Others
	Epelsiban is a selective and orally bioavailable oxytocin receptor antagonist (pKi: 9.9 for human oxytocin receptor).
T24291	L 366811 L 366,811,L-366,811,L366811,L366,811,L-366811
	L 366811 is a potent oxytocin antagonist.
T24278	L 156373 L-156373,L156373
	L 156373 is an oxytocin antagonist.
T28018	Merotocin FE202767,FE 202767,FE-202767
	Merotocin is a potent and highly selective peptidic agonist of the oxytocin receptor.
T69504	Barusiban
	Barusiban is an oxytocin receptor antagonist.
T70511	F-327
	F-327 is an oxytocin antagonist.
T24289	L 366682 L366,682,L-66,682,L 366,682,L-366682,L366682
	L 366682 is an oxytocin antagonist.
T24288	L 365209 L365,209,L365209,L 365,209,L-365,209,L-365209
	L 365209 is an oxytocin antagonist.
T25902	Ota-vasotocin OVTA
	Ota-vasotocin is a ligand utilized in quantitative receptor autoradiography for oxytocin receptors.

化合物

Oxytocin C-terminal tripeptide Acetate

Cat.No: T21534L

Synonym: Oxytocin C-terminal tripeptide Acetate(2002-44-0 Free base)

Target: Others

[Asp5]-Oxytocin

Cat.No: T40756

Synonym: [Asp5]-Oxytocin

[Glu4]-Oxytocin

Cat.No: T40536

Synonym: [Glu4]-Oxytocin

[Leu3]-Oxytocin

Cat.No: T40534

Synonym: [Leu3]-Oxytocin

[D-Asn5]-Oxytocin

Cat.No: T40658

Synonym: [D-Asn5]-Oxytocin

Oxytocin, deamino-6-carba-

Cat.No: T33850

Synonym: Deamino-6-carbaoxytocin,beta-Deaminocystathionine-oxytocin

Oxytocin antiparallel dimer

Cat.No: T39420

Oxytocin parallel dimer

Cat.No: T39388

Oxytocin free acid

Cat.No: T40528

Synonym: 9-Deamidooxytocin

Oxytocin, deamino-1-carba-

Cat.No: T33849

Synonym: Deamino-1-carbaoxytocin

Val9-Oxytocin

Cat.No: T80136

Target: Vasopressin Receptor

(Ile8)-Oxytocin

Cat.No: T76624

OT-R antagonist 1

Cat.No: T12331L

Synonym: Oxytocin receptor antagonist 1

Target: Others

OT-R antagonist 2

Cat.No: T12331

Synonym: Oxytocin receptor antagonist 2

Target: Others

Pro8-Oxytocin

Cat.No: T80133

Target: Oxytocin Receptor

[Asp5]-Oxytocin acetate

Cat.No: T76211

Cat.No: T4996

Synonym: 阿托西班,RWJ22164,RW22164

Target: Oxytocin Receptor, Vasopressin Receptor

(Phe2,Orn8)-Oxytocin

Cat.No: T76629

(Thr4,Gly7)-Oxytocin

Cat.No: T76265

(Val3,Pro8)-Oxytocin

Cat.No: T80140

Target: Oxytocin Receptor

Pro8-Oxytocin TFA

Cat.No: T80134

Target: Oxytocin Receptor

Oxytocin parallel dimer TFA

Cat.No: T78021

Oxytocin antiparallel dimer TFA

Cat.No: T81583

(Phe2,Orn8)-Oxytocin acetate

Cat.No: T76630

Atosiban acetate

Cat.No: T5148

Synonym: RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164,醋酸阿托西班

Target: Oxytocin Receptor, Vasopressin Receptor

Cat.No: T11857

Target: Oxytocin Receptor

(d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin

Cat.No: T80126

Target: Oxytocin Receptor

Carbetocin acetate

Cat.No: T7601L

Synonym: 醋酸卡贝缩宫素,Carbetocin acetate(37025-55-1 free base),卡贝缩宫素醋酸盐

Target: Oxytocin Receptor

Cat.No: T7601

Synonym: 卡贝缩宫素,醋酸卡贝缩宫素

Target: Oxytocin Receptor

Cat.No: T76049

N-Acetyloxytocin

Cat.No: T37694

Cat.No: T3347

Synonym: PF 3274167,Cligosiban,PF-3274167

Target: OX Receptor

Cat.No: T28855

Synonym: SSR-126768A,SSR 126768A

Target: Oxytocin Receptor

[Arg8]-Vasotocin acetate（113-80-4 free base)

Cat.No: TP1400L

Target: Others

Cat.No: T15682

Target: Oxytocin Receptor, Vasopressin Receptor

d[Cha4]-AVP acetate(500170-27-4 free base)

Cat.No: TP2082L

Target: Vasopressin Receptor

Cat.No: T16736

Synonym: GSK 221149,GSK 221149A

Target: Others

Cat.No: T23441

Target: Others

Cat.No: T24286

Synonym: L364,918,L-364918,L-364,918,L 364,918,L364918

Cat.No: T23528

Target: Others

Cat.No: T27763

Synonym: L 366,509,L 366509,L366,509,L-366,509

Cat.No: T11502

Synonym: GSK 557296

Target: Others

Cat.No: T24291

Synonym: L 366,811,L-366,811,L366811,L366,811,L-366811

Cat.No: T24278

Synonym: L-156373,L156373

Cat.No: T28018

Synonym: FE202767,FE 202767,FE-202767

Cat.No: T69504

Cat.No: T70511

Cat.No: T24289

Synonym: L366,682,L-66,682,L 366,682,L-366682,L366682

Cat.No: T24288

Synonym: L365,209,L365209,L 365,209,L-365,209,L-365209

Cat.No: T25902

Synonym: OVTA

Cat. No.	Product Name	Target	Signaling Pathways
T5026	Oxytocin 催产素,α-Hypophamine,Oxytocic hormone,Oxytocin (Syntocinon)	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Oxytocin (Oxytocin (Syntocinon)) 是哺乳动物的神经垂体激素，是多效的下丘脑肽，是催产素受体的配体，有助于分娩、哺乳和亲社会行为。它可作为一种压力应对分子，具有抗炎、抗氧化剂和保护作用。
T5145	Oxytocin acetate Oxytocic hormone acetate,α-Hypophamine acetate,Oxytocin acetate (50-56-6 free base),醋酸催产素	Oxytocin Receptor	Endocrinology/Hormones; GPCR/G Protein
	Oxytocin acetate (α-Hypophamine acetate) 是哺乳动物的神经垂体激素，是多效的下丘脑肽，是催产素受体的配体，有助于分娩、哺乳和亲社会行为。它可作为一种压力应对分子，具有抗炎、抗氧化剂和保护作用。
T5065	GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD Monosodium-GMP,cGMP sodium salt,鸟苷-3',5'-环磷酸一钠盐,Cyclic GMP	PKA	Tyrosine Kinase/Adaptors
	GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD (cGMP sodium salt) 也称为 cGMP，是一种细胞调节剂，被描述为第二信使。它的水平随着各种激素的增加而增加，包括乙酰胆碱、胰岛素和催产素。 cGMP 激活蛋白激酶 G(PKG) 并调节离子通道电导，信号传导影响多种过程，包括平滑肌松弛和增殖、光转导和能量稳态。
T36931	Penicillide
	Penicillide is a fungal metabolite originally isolated from Penicillium that has diverse biological activities. It is an inhibitor of calpain 2/m-calpain (IC50 = 7.1 μM) and acyl-coenzyme A:cholesterol acyltransferase (ACAT; IC50 = 22.9 μM). It is also an antagonist of oxytocin receptors (IC50 = 67 μM). Penicillide inhibits RNA synthesis in P388 murine leukemia cells.

天然产物

Cat.No: T5026

Synonym: 催产素,α-Hypophamine,Oxytocic hormone,Oxytocin (Syntocinon)

Target: Oxytocin Receptor

Oxytocin acetate

Cat.No: T5145

Synonym: Oxytocic hormone acetate,α-Hypophamine acetate,Oxytocin acetate (50-56-6 free base),醋酸催产素

Target: Oxytocin Receptor

GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD

Cat.No: T5065

Synonym: Monosodium-GMP,cGMP sodium salt,鸟苷-3',5'-环磷酸一钠盐,Cyclic GMP

Target: PKA

Cat.No: T36931

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