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Cat. No. Product Name Target Signaling Pathways
T28223 OB-1

OB-1 is an inhibitor of stomatin-like protein-3 (STOML3) oligomerization. OB-1 reversibly reduces the sensitivity of mechanically gated currents in sensory neurons and silence mechanoreceptors in vivo.
T9266 Fatostatin

Lipid; Fatty Acid Synthase Metabolism
Fatostatin A 是一种SREBP 活化的特异性抑制剂,能够抑制 SREBP-1 和 SREBP-2 的活化。它与 SCAP (SREBP 裂解激活蛋白) 结合,抑制 SREBPs 的 ER-Golgi 易位。它具有抗肿瘤活性,能抑制ob/ob 小鼠的高血糖。它抑制细胞中成脂基因的转录。
T6832 Fatostatin hydrobromide

Fatostatin HBr,Fatostatin A,Fatostatin A HBr,Fatostatin

NPC1L1; Fatty Acid Synthase Membrane transporter/Ion channel; Metabolism
Fatostatin hydrobromide (Fatostatin A HBr) 是一种 SREBP 活化的特异性抑制剂,可抑制 SREBP-1 和 SREBP-2 的活化。它与 SCAP (SREBP 裂解激活蛋白) 结合,抑制 SREBPs 的 ER-Golgi 易位。它具有抗肿瘤作用,能抑制 ob/ob 小鼠的高血糖。它抑制了细胞中成脂基因的转录。
T68288 OB-24 free base

OB-24 free base is a potent and selective heme oxygenase 1 (HO-1) inhibitor.
T83696 Gastric Inhibitory Peptide 1 (3-42) (human) TFA

Glucose-dependent Insulinotropic Polypeptide 3-42,GIP-1 (3-42)

胃抑制肽1(GIP-1) (3-42)是肠促胰岛素激素GIP的一个肽段,同时也是GIP受体的拮抗剂。它通过血清二肽基肽酶4(DDP-4)从GIP中形成。GIP-1 (3-42) (100 nM)在减少BRIN-BD11胰腺细胞的胰岛素分泌方面起作用。在以25 nmol/kg剂量给药的ob/ob糖尿病小鼠模型中,它能增加血浆葡萄糖水平并降低血浆胰岛素水平。
T41175 OB 24 hydrochloride

OB 24 hydrochloride is a potent and selective heme oxygenase 1 (HO-1) inhibitor (IC50 values are 1.9 and >100 μM for HO-1 and HO-2 respectively), reduces protein carbonylation and reactive oxygen species formation in advanced prostate cancer cells (PCA). Inhibits cell proliferationin vitroand PCA tumor growth and lymph node/lung metastasesin vivo. Synergizes with Taxol.

化合物

OB-1
Cat.No: T28223
Synonym:
Target:
Fatostatin
Cat.No: T9266
Synonym:
Target: Lipid, Fatty Acid Synthase
Fatostatin hydrobromide
Cat.No: T6832
Synonym: Fatostatin HBr,Fatostatin A,Fatostatin A HBr,Fatostatin
Target: NPC1L1, Fatty Acid Synthase
OB-24 free base
Cat.No: T68288
Synonym:
Target:
Gastric Inhibitory Peptide 1 (3-42) (human) TFA
Cat.No: T83696
Synonym: Glucose-dependent Insulinotropic Polypeptide 3-42,GIP-1 (3-42)
Target:
OB 24 hydrochloride
Cat.No: T41175
Synonym:
Target:
TargetMol Loading
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