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Cat. No. Product Name Target Signaling Pathways
T1777 Nintedanib

BIBF 1120,Intedanib,尼达尼布

VEGFR; FGFR; FLT; PDGFR; Src Angiogenesis; Tyrosine Kinase/Adaptors
Nintedanib (Intedanib) 是一种三重血管激酶抑制剂,抑制 VEGFR1、VEGFR2、VEGFR3 (IC50=34/13/13 nM),FGFR1、FGFR2、FGFR3 (IC50=69/37/108 nM),PDGFRα、PDGFRβ (IC50=59/65 nM)。Nintedanib 具有抗肿瘤活性,通过抑制血管生成来抑制肿瘤生长。
T5001 Nintedanib esylate

Intedanib,乙磺酸尼达尼布,BIBF 1120 (esylate),尼达尼布乙磺酸盐,Nintedanib Ethanesulfonate Salt,BIBF 1120

VEGFR; FGFR; PDGFR Angiogenesis; Tyrosine Kinase/Adaptors
Nintedanib esylate (BIBF 1120 esylate) 是一种有效的三重血管激酶抑制剂,能够抑制 VEGFR1 (IC50:34 nM)、VEGFR2 (IC50:13 nM)、VEGFR3 (IC50:13 nM),FGFR1 (IC50:69 nM)、FGFR2 (IC50:37 nM)、FGFR3 (IC50:108 nM),PDGFRα (IC50:59 nM)、PDGFRβ (IC50:65 nM)。
T11997 MELK-IN-1

Nintedanib Impurity L,MELK inhibitor 17,尼达尼布杂质L

MELK PI3K/Akt/mTOR signaling
MELK-IN-1 (MELK inhibitor 17)是一种母体胚胎亮氨酸拉链激酶的有效抑制剂,IC50=3 nM,Ki=0.39 nM。
T68229 Nintedanib esylate hemihydrate

Nintedanib esylate hemihydrate is a potent inhibitor of multiple receptor tyrosine kinases (RTKs) and non-receptor tyrosine kinases (nRTKs).

化合物

Nintedanib
Cat.No: T1777
Synonym: BIBF 1120,Intedanib,尼达尼布
Target: VEGFR, FGFR, FLT, PDGFR, Src
Nintedanib esylate
Cat.No: T5001
Synonym: Intedanib,乙磺酸尼达尼布,BIBF 1120 (esylate),尼达尼布乙磺酸盐,Nintedanib Ethanesulfonate Salt,BIBF 1120
Target: VEGFR, FGFR, PDGFR
MELK-IN-1
Cat.No: T11997
Synonym: Nintedanib Impurity L,MELK inhibitor 17,尼达尼布杂质L
Target: MELK
Nintedanib esylate hemihydrate
Cat.No: T68229
Synonym:
Target:
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