Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0711 |
Niclosamide
BAY2353,Niclocide,氯硝柳胺 |
Antibiotic; STAT; Parasite | JAK/STAT signaling; Microbiology/Virology; Stem Cells |
Niclosamide (Niclocide) 是一种口服生物可利用的氯化水杨酰苯胺。它通过抑制 DNA 复制,具有驱虫和潜在的抗肿瘤活性。 | |||
T0711L |
Niclosamide olamine
Niclosamide-olamine,Niclosamide Ethanolamine salt |
Antibiotic; STAT; Parasite; Autophagy | Autophagy; JAK/STAT signaling; Microbiology/Virology; Stem Cells |
Niclosamide olamine (Niclosamide Ethanolamine salt) 是一种驱虫剂,可破坏寄生虫和动物模型中的线粒体代谢。它可逆地抑制雷帕霉素复合物的哺乳动物靶标,从而抑制STAT3(IC50为 0.25 μM) 并刺激自噬反应。 | |||
T23068 |
Niclosamide monohydrate
|
Others | Others |
Niclosamide Monohydrate is used for the treatment of most tapeworm infections by inhibiting DNA replication. | |||
T72519 |
Niclosamide sodium
BAY2353 sodium |
||
Niclosamide (BAY2353) sodium 为用于研究寄生虫感染的口服抗蠕虫化合物,同时是STAT3抑制剂,在HeLa细胞中IC50为0.25μM。此化合物显示抗癌生物活性,并可抑制Vero E6细胞DNA复制。 | |||
T60919 |
SARS-CoV-2-IN-13
|
SARS-CoV | Microbiology/Virology |
SARS-CoV-2-IN-13 (compound 6) 是氯硝柳胺的类似物。在人血浆和肝S9酶测定中,SARS-CoV-2-IN-13 比氯硝柳胺更稳定。SARS-CoV-2-IN-13 口服给药时可以提高生物利用度和半衰期。SARS-CoV-2-IN-13 是SARS-CoV-2的有效抑制剂,IC50值为 0.057 μM。 | |||
T60538 |
SARS-CoV-2-IN-14
3',5-Dichlorosalicylanilide |
SARS-CoV | Microbiology/Virology |
SARS-CoV-2-IN-14 是一种有效的、可口服的 SARS-CoV-2 抑制剂(IC50 :0.39 μM),是一种氯硝柳胺类似物。SARS-CoV-2-IN-14在人血浆和肝 S9 酶测定中比氯硝柳胺稳定性更强。SARS-CoV-2-IN-14以口服的方式给药可以提高其生物利用度和半衰期。 | |||
T69250 |
JMX0312
|
||
JMX0312 is a salicylamide derivative used as a potent inhibitor of HAdV infection. JMX0312 showed significantly improved anti-HAdV activities with nanomolar to submicromolar IC50 values and high selectivity indexes (SI > 100), indicating better safety windows, compared to those of the lead compound niclosamide. | |||
T60818 |
SARS-CoV-2-IN-15
|
||
SARS-CoV-2-IN-15 (compound 11) 是一种氯硝柳胺类似物,其在人血浆和肝 S9 酶测定中比氯硝柳胺具有更高的稳定性。当口服给药时,它可以提高生物利用度和半衰期。SARS-CoV-2-IN-15 是SARS-CoV-2的有效抑制剂,IC50值为 0.49 μM。 | |||
T37632 |
TFM
|
||
TFM is a piscicide.1It is toxic to sea lamprey (P. marinus) with LC50values ranging from 1.97 to 2.11 and 2.05 to 2.21 mg/L for sac and swim-up fry, respectively, 1.6 to 2.45 mg/L for juveniles, and 1.6 to 1.63 mg/L for adults. It is also toxic to juvenile lake sturgeon (A. fulvescens) less than 100 mm in size but not to a variety of other fish species. TFM (50 μM) uncouples oxidative phosphorylation by 22 and 28% in isolated sea lamprey and rainbow trout (O. mykiss) liver, respectively.2Formula... |