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抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T2319 Acotiamide monohydrochloride trihydrate

Acotiamide hydrochloride,YM-443 HCl,盐酸阿考替胺,Z-338 HCl

AChE Neuroscience
Acotiamide monohydrochloride trihydrate (Z-338 HCl) 是一种首创的、具有口服活性的胃肠动力药。它通过促毒蕈碱受体拮抗作用和乙酰胆碱酯酶(AChE)抑制作用增强肠神经元释放的乙酰胆碱,从而增强胃排空和胃部适应性,有潜力用于功能性消化不良的研究。
T63237 Acotiamide hydrochloride

Acotiamide hydrochloride 是选择性的、口服具有活力的、可逆的乙酰胆酶碱酯 (AChE) 抑制剂 (IC50: 1.79 μM),能够提高胃收缩性,加速胃排空延迟,能够用于研究胃动力障碍的功能性消化不良及肠道炎症。
T70122 Acotiamide Methyl Ether

Acotiamide Methyl Ether is a metabolite of Acotiamide -- an acetylcholinesterase inhibitor which has been shown to stimulate gastric motility and improve gastric motility dysfunction in rats. Acotiamide Hydrochloride has also been shown to improve meal-related symptoms of functional dyspepsia.
T22230 Acotiamide

Acotiamide 是一种具有口服活性、选择性和可逆性的乙酰胆酶碱酯 (AChE) 抑制剂,IC50值为1.79 μM。Acotiamide 是一种胃促动力剂,可增强胃收缩性并加速胃排空延迟。Acotiamide 可用于胃动力障碍的功能性消化不良及肠道炎症的研究。

化合物

Acotiamide monohydrochloride trihydrate
Cat.No: T2319
Synonym: Acotiamide hydrochloride,YM-443 HCl,盐酸阿考替胺,Z-338 HCl
Target: AChE
Acotiamide hydrochloride
Cat.No: T63237
Synonym:
Target:
Acotiamide Methyl Ether
Cat.No: T70122
Synonym:
Target:
Acotiamide
Cat.No: T22230
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN2215 Taurochenodeoxycholic acid sodium

牛磺鹅去氧胆酸钠盐,Sodium taurochenodeoxycholate,牛磺鹅去氧胆酸钠

Apoptosis; Endogenous Metabolite Apoptosis; Metabolism
Taurochenodeoxycholic acid sodium (Sodium taurochenodeoxycholate) 是动物胆汁酸的主要生物活性物质之一。它可诱导细胞凋亡,具有抗炎和免疫调节作用。
T2A2481 Taurochenodeoxycholic Acid

Chenodeoxycholyltaurine,TCDCA,Chenyltaurine,Taurochenodeoxycholate,12-Deoxycholyltaurine,牛磺鹅去氧胆酸

Apoptosis; TNF; Caspase; Endogenous Metabolite Apoptosis; Metabolism; Proteases/Proteasome
Taurochenodeoxycholic Acid (12-Deoxycholyltaurine) 是动物胆汁酸的主要生物活性物质之一,可诱导细胞凋亡,具有明显的抗炎和免疫调节作用。

天然产物

Taurochenodeoxycholic acid sodium
Cat.No: TN2215
Synonym: 牛磺鹅去氧胆酸钠盐,Sodium taurochenodeoxycholate,牛磺鹅去氧胆酸钠
Target: Apoptosis, Endogenous Metabolite
Taurochenodeoxycholic Acid
Cat.No: T2A2481
Synonym: Chenodeoxycholyltaurine,TCDCA,Chenyltaurine,Taurochenodeoxycholate,12-Deoxycholyltaurine,牛磺鹅去氧胆酸
Target: Apoptosis, TNF, Caspase, Endogenous Metabolite
TargetMol Loading
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