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7

抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T33577 NADA-green

NADA green

NADA-green is a fluorescent D-amino acid for labeling peptidoglycans in live bacteria.
T62530 N-Arachidonyldopamine

NADA

Cannabinoid Receptor GPCR/G Protein
N-Arachidonyldopamine (NADA) 是一种选择性的、强效的内源性 CB1 受体激动剂 (Ki: 250 nM)。N-Arachidonyldopamine 也是一种有效的、选择性 TRPV1 激动剂,其 EC50 值 ~50 nM。
T2189 Sodium orthovanadate

Sodium vanadate,钒酸钠,Trisodium vanadate,Sodium pervanadate

ATPase; Phosphatase Membrane transporter/Ion channel; Metabolism
Sodium orthovanadate 是一种蛋白酪氨酸磷酸酶,碱性磷酸酶和一些ATP 酶的抑制剂,有可能充当磷酸盐类似物。它具有胰岛素样作用、对心室肌的正性肌力作用和其他代谢作用。
T9430 Venadaparib

NOV140101,IDX-1197

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
Venadaparib (NOV140101) 是一种选择性和具有口服活性的 PARP 抑制剂,对 PARP1和 PARP2的 IC50分别为 1.4 和 1.0 nM。它可防止 DNA 单链断裂 (SSB) 的修复,可研究实体瘤。
T39147 Venadaparib hydrochloride

IDX-1197 hydrochloride

Venadaparib hydrochloride (IDX-1197) is a potent and selective PARP inhibitor that exhibits significant anticancer properties. It is particularly effective in solid tumor research.
T23399 STEARDA

Others Others
STEARDA potentiates TRPV1-mediated effects of NADA.
T23118 PALDA

Others Others
PALDA potentiates TRPV1-mediated effects of NADA.

化合物

NADA-green
Cat.No: T33577
Synonym: NADA green
Target:
N-Arachidonyldopamine
Cat.No: T62530
Synonym: NADA
Target: Cannabinoid Receptor
Sodium orthovanadate
Cat.No: T2189
Synonym: Sodium vanadate,钒酸钠,Trisodium vanadate,Sodium pervanadate
Target: ATPase, Phosphatase
Venadaparib
Cat.No: T9430
Synonym: NOV140101,IDX-1197
Target: PARP
Venadaparib hydrochloride
Cat.No: T39147
Synonym: IDX-1197 hydrochloride
Target:
STEARDA
Cat.No: T23399
Synonym:
Target: Others
PALDA
Cat.No: T23118
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T40158 N-acetyldopamine

NADA,N-乙酰多巴胺

N-acetyldopamine (NADA) is a catecholamine utilized by insects as a precursor for sclerotization, a process that strengthens their cuticle.

天然产物

N-acetyldopamine
Cat.No: T40158
Synonym: NADA,N-乙酰多巴胺
Target:
TargetMol Loading
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