7
1
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T33577 |
NADA-green
NADA green |
||
NADA-green is a fluorescent D-amino acid for labeling peptidoglycans in live bacteria. | |||
T62530 |
N-Arachidonyldopamine
NADA |
Cannabinoid Receptor | GPCR/G Protein |
N-Arachidonyldopamine (NADA) 是一种选择性的、强效的内源性 CB1 受体激动剂 (Ki: 250 nM)。N-Arachidonyldopamine 也是一种有效的、选择性 TRPV1 激动剂,其 EC50 值 ~50 nM。 | |||
T2189 |
Sodium orthovanadate
Sodium vanadate,钒酸钠,Trisodium vanadate,Sodium pervanadate |
ATPase; Phosphatase | Membrane transporter/Ion channel; Metabolism |
Sodium orthovanadate 是一种蛋白酪氨酸磷酸酶,碱性磷酸酶和一些ATP 酶的抑制剂,有可能充当磷酸盐类似物。它具有胰岛素样作用、对心室肌的正性肌力作用和其他代谢作用。 | |||
T9430 |
Venadaparib
NOV140101,IDX-1197 |
PARP | Chromatin/Epigenetic; DNA Damage/DNA Repair |
Venadaparib (NOV140101) 是一种选择性和具有口服活性的 PARP 抑制剂,对 PARP1和 PARP2的 IC50分别为 1.4 和 1.0 nM。它可防止 DNA 单链断裂 (SSB) 的修复,可研究实体瘤。 | |||
T39147 |
Venadaparib hydrochloride
IDX-1197 hydrochloride |
||
Venadaparib hydrochloride (IDX-1197) is a potent and selective PARP inhibitor that exhibits significant anticancer properties. It is particularly effective in solid tumor research. | |||
T23399 |
STEARDA
|
Others | Others |
STEARDA potentiates TRPV1-mediated effects of NADA. | |||
T23118 |
PALDA
|
Others | Others |
PALDA potentiates TRPV1-mediated effects of NADA. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T40158 |
N-acetyldopamine
NADA,N-乙酰多巴胺 |
||
N-acetyldopamine (NADA) is a catecholamine utilized by insects as a precursor for sclerotization, a process that strengthens their cuticle. |