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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T3097 Mycophenolic Acid Impurity

马替麦考酚酸杂质,5,7-dihydroxy-4-methylphthalide

Others Others
Mycophenolic Acid Impurity (5,7-dihydroxy-4-methylphthalide) 是一种免疫抑制药物和有效的抗增殖剂,可用于代替旧的抗增殖剂 azathioprine。它通常用作三联疗法的一部分,包括钙调神经磷酸酶抑制剂(ciclosporin 或 tacrolimus)和prednisolone。它还可用于研究选择表达编码 XGPRT(黄嘌呤鸟嘌呤磷酸核糖基转移酶)的大肠杆菌基因的动物细胞。
T12135 Mycophenolic acid-d3

Mycophenolate-d3,Mycophenolate D3

Others; Antibacterial Microbiology/Virology; Others
Mycophenolic acid-d3 (Mycophenolate-d3) 是 Mycophenolic acid 的衍生物。Mycophenolic acid 是一种降低GTP 水平和损害RNA 聚合酶II (RNAP II)转录延伸的化合物,促进了近端位点的使用,能够逆转虫草素对选择性聚腺苷化的作用。
T61099 Mycophenolic acid sodium

Mycophenolic acid sodium is a potent uncompetitive inhibitor of inosine monophosphate dehydrogenase (IMPDH), exhibiting an EC50 of 0.24 μM. It has broad antiviral activity against RNA viruses, including influenza. Additionally, mycophenolic acid sodium possesses immunosuppressive properties and exerts antiangiogenic and antitumor effects [1][2].
T124275 Mycophenolic acid IV

Mycophenolic acid IV 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124275,CAS号为 74838-16-7。
T19303 (E/Z)-Methyl mycophenolate

Others Others
Methyl mycophenolate can be used to synthesize mycophenolic acid β-D-glucuronide and phenolic glycosides. (E/Z)-Methyl mycophenolate is a racemic compound of (Z)-Methyl mycophenolate and (E)-Methyl mycophenolate isomers. Methyl mycophenolate is a methyl e

化合物

Mycophenolic Acid Impurity
Cat.No: T3097
Synonym: 马替麦考酚酸杂质,5,7-dihydroxy-4-methylphthalide
Target: Others
Mycophenolic acid-d3
Cat.No: T12135
Synonym: Mycophenolate-d3,Mycophenolate D3
Target: Others, Antibacterial
Mycophenolic acid sodium
Cat.No: T61099
Synonym:
Target:
Mycophenolic acid IV
Cat.No: T124275
Synonym:
Target:
(E/Z)-Methyl mycophenolate
Cat.No: T19303
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T1335 Mycophenolic acid

霉酚酸,Mycophenolate,RS-61443

Apoptosis; Dehydrogenase; Endogenous Metabolite; Antibacterial; Antibiotic; UGT; Antifungal Apoptosis; Metabolism; Microbiology/Virology
Mycophenolic acid (Mycophenolate) 是一种有效的非竞争性肌苷单磷酸脱氢酶 (IMPDH) 抑制剂,EC50为 0.24 µM。它对多种 RNA 病毒具有抗病毒作用。它也是一种免疫抑制剂,具有抗血管生成和抗肿瘤作用。
T19424 Methyl mycophenolate

Mycophenolic Acid Methyl Ester,霉酚酸酯杂质E

Others Others
Methyl mycophenolate (Mycophenolic Acid Methyl Ester) 是一种霉酚酸的甲酯,存在于海洋真菌Phaeosphaeria spartinae 中。
T60104 Mycophenolic acid-β-D-glucuronide solution

Others Others
Mycophenolic acid glucuronide 是人血浆中mycophenolic acid 的葡糖甙代谢产物。
T6293 Mycophenolate Mofetil

TM-MMF,吗替麦考酚酯,RS 61443

Apoptosis; Dehydrogenase; Drug Metabolite Apoptosis; Metabolism
Mycophenolate Mofetil (TM-MMF) 是 Mycophenolic acid 的吗啉乙酯前药。它通过抑制肌苷一磷酸脱氢酶抑制从头嘌呤合成,显示出选择性淋巴细胞抗增殖作用。

天然产物

Mycophenolic acid
Cat.No: T1335
Synonym: 霉酚酸,Mycophenolate,RS-61443
Target: Apoptosis, Dehydrogenase, Endogenous Metabolite, Antibacterial, Antibiotic, UGT, Antifungal
Methyl mycophenolate
Cat.No: T19424
Synonym: Mycophenolic Acid Methyl Ester,霉酚酸酯杂质E
Target: Others
Mycophenolic acid-β-D-glucuronide solution
Cat.No: T60104
Synonym:
Target: Others
Mycophenolate Mofetil
Cat.No: T6293
Synonym: TM-MMF,吗替麦考酚酯,RS 61443
Target: Apoptosis, Dehydrogenase, Drug Metabolite
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