首页 工具
登录
购物车

搜索结果

Search Results for " mink "

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T8730 BMS986260

TGF-beta/Smad Stem Cells
BMS986260是一种口服有活力的选择性TGFβR1抑制剂,是免疫肿瘤学药物。它能够抑制 MINK 和 NHLF 细胞系中 TGFβ 介导的 pSMAD2/3 核转位,IC50值分别为 350 nM 和 190 nM。它对 TGFβR1 的选择比 TGFβR2 同功酶高。
T69851 Riminkefon

Riminkefon 是κ 阿片受体的激动剂。
T0860L Mefloquine

Ro215998,WR 142490,Ro-215998,氟甲喹羟哌啶,Lariam,Ro 215998

Others Others
Mefloquine (Ro 215998) 是一种喹啉抗疟药,是一种抗 SARS-CoV-2 进入抑制剂。 Mefloquine 也是一种 K+ 通道 (KvQT1/minK) 拮抗剂,IC50 为 ~1 μM。它可用于疟疾、系统性红斑狼疮和癌症研究。
T0860 Mefloquine hydrochloride

Mefloquin hydrochloride,Mefloquine HCl,盐酸甲氟喹

Potassium Channel; SARS-CoV; Reactive Oxygen Species; Parasite; Autophagy Autophagy; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; NF-κB
Mefloquine hydrochloride (Mefloquin hydrochloride) 是喹啉抗疟药,是抗 SARS-CoV-2进入抑制剂,可研究疟疾、系统性红斑狼疮和癌症。它也是 K+通道(KvQT1/minK) 拮抗剂,IC50约为 1 μM。
T33945 PF-06260933 HCl

PF06260933 dihydrochloride,PF-06260933 dihydrochloride,PF 06260933 dihydrochloride

PF-06260933 Dihydrochloride is a MAP4K4 (HGK) inhibitor (IC50 = 140 nM). It can improve the fasting hyperglycemia in mice. In addition, it inhibited Mink and Tnik (IC50 values of 8 and 13 nM, respectively).
T36016 PF 06260933 dihydrochloride

MAP4K4 (HGK) inhibitor (IC50 = 140 nM). Also inhibits MINK and TNIK (IC50 values are 8 and 13 nM, respectively). Improves fasting hyperglycemia in mice. Orally active. Ammirati et al (2015) Discovery of an in vivo tool to establish proof-of-concept for MAP4K4-based antidiabetic treatment. ACS Med.Chem.Lett. 6 1128 PMID:26617966

化合物

BMS986260
Cat.No: T8730
Synonym:
Target: TGF-beta/Smad
Riminkefon
Cat.No: T69851
Synonym:
Target:
Mefloquine
Cat.No: T0860L
Synonym: Ro215998,WR 142490,Ro-215998,氟甲喹羟哌啶,Lariam,Ro 215998
Target: Others
Mefloquine hydrochloride
Cat.No: T0860
Synonym: Mefloquin hydrochloride,Mefloquine HCl,盐酸甲氟喹
Target: Potassium Channel, SARS-CoV, Reactive Oxygen Species, Parasite, Autophagy
PF-06260933 HCl
Cat.No: T33945
Synonym: PF06260933 dihydrochloride,PF-06260933 dihydrochloride,PF 06260933 dihydrochloride
Target:
PF 06260933 dihydrochloride
Cat.No: T36016
Synonym:
Target:
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼