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Cat. No. Product Name Target Signaling Pathways
T2350 MALT1 inhibitor MI-2

MALT1 inhibitor,MI 2,MI 2 (MALT1 inhibitor)

MALT Immunology/Inflammation
MI 2 (MALT1 inhibitor) 是一种MALT1抑制剂 (IC50=5.84 μM),对动物无毒性。它能够直接与 MALT1 结合,不可逆地抑制蛋白酶功能,并伴有 NF-κB 报告子活性抑制、c-REL 核定位抑制和 NF-κB 靶基因下调。
T2649 Menin-MLL inhibitor MI-2

Menin-MLL Inhibitor,MI2,MI-2,Menin-MLL inhibitor 2,MI 2

Apoptosis; Epigenetic Reader Domain; Histone Methyltransferase Apoptosis; Chromatin/Epigenetic
Menin-MLL inhibitor MI-2 (MI2) 抑制Menin-MLL 相互作用,IC50为 446±28 nM。
T22978 MI-2 (hydrochloride)

Others Others
MI-2 (Menin-MLL Inhibitor) is an effective menin-MLL interaction inhibitor (IC50: 446 ± 28 nM).

化合物

MALT1 inhibitor MI-2
Cat.No: T2350
Synonym: MALT1 inhibitor,MI 2,MI 2 (MALT1 inhibitor)
Target: MALT
Menin-MLL inhibitor MI-2
Cat.No: T2649
Synonym: Menin-MLL Inhibitor,MI2,MI-2,Menin-MLL inhibitor 2,MI 2
Target: Apoptosis, Epigenetic Reader Domain, Histone Methyltransferase
MI-2 (hydrochloride)
Cat.No: T22978
Synonym:
Target: Others
TargetMol Loading
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