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1

抑制剂 & 化合物

9

天然产物

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Cat. No. Product Name Target Signaling Pathways
T81970 Kuwanon T

Kuwanon T为一种源自桑树根皮的异戊二烯黄酮类化合物,能抵御t-BHP诱导的氧化应激,其EC50值为30.32 μM。

化合物

Kuwanon T
Cat.No: T81970
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TQ0301 Kuwanon A

NO Synthase Immunology/Inflammation
Kuwanon A 抑制一氧化氮的产生 (IC50: 10.5 μM)。Kuwanon A 是从桑树 (Morus alba L.) 中分离出来的黄酮衍生物。
T81972 Kuwanon K

Kuwanon K为从Morus Lhou分离得到的天然化合物。
T81971 Kuwanon O

Kuwanon O, 黄酮类衍生物, 包含融合的二氢查尔酮部分,可从Morus lhou (set.) Koidz根皮中提取。
T81969 Kuwanon W

Kuwanon W为从Morus lhou根中分离的天然化合物。
TN1849 Kuwanon H

GPR; Bombesin Receptor Endocrinology/Hormones; GPCR/G Protein
Kuwanon H 是分离自桑白皮的黄酮类化合物,具有拮抗非肽类蛙皮素受体的活性。Kuwanon H 特异性抑制细胞内胃泌激素释放肽 CRP 与GRP-preferring 受体的结合,Ki 为 290 nM。
T3S1612 kuwanon G

桑黄酮G,Moracenin B,桑黄酮 G,Kuwanone G

Phosphatase; Antibacterial; Bombesin Receptor; AChR; AChE; Glucosidase GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience
Kuwanon G (Moracenin B) 是一种从桑树中得到的黄酮类蛙皮素受体拮抗剂,具有杀菌作用。
TN2445 Kuwanon B

Others Others
Kuwanon B belongs to the class of organic compounds known as 3-prenylated flavones. Within the cell, kuwanon B is primarily located in the membrane (predicted from logP). Outside of the human body, kuwanon b can be found in fruits. This makes kuwanon b a
TN1848 Kuwanon E

桑黄酮 E,桑皮酮 E,5'-[(E)-3,7-二甲基-2,6-辛二烯基]-2',4',5,7-四羟基黄烷酮

AChR Neuroscience
Kuwanon E inhibited cholinesterase enzyme in a dose-dependent manner with K i values ranging between 3.1 and 37.5 μM and between 1.7 and 19.1 μM against acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) enzymes, respectively. Kuwanon E also inh
TN3744 Cyclomorusin

NOS; AChR Immunology/Inflammation; Neuroscience
Cyclomorusin exhibits competitive inhibition toward monophenolase activity of mushroom tyrosinase, the IC50 value of 0.092 microM. It evokes the stimulation of superoxide anion generation in fMLP-stimulated rat neutrophils. Cyclomorusin , neocyclomorusin

天然产物

Kuwanon A
Cat.No: TQ0301
Synonym:
Target: NO Synthase
Kuwanon K
Cat.No: T81972
Synonym:
Target:
Kuwanon O
Cat.No: T81971
Synonym:
Target:
Kuwanon W
Cat.No: T81969
Synonym:
Target:
Kuwanon H
Cat.No: TN1849
Synonym:
Target: GPR, Bombesin Receptor
kuwanon G
Cat.No: T3S1612
Synonym: 桑黄酮G,Moracenin B,桑黄酮 G,Kuwanone G
Target: Phosphatase, Antibacterial, Bombesin Receptor, AChR, AChE, Glucosidase
Kuwanon B
Cat.No: TN2445
Synonym:
Target: Others
Kuwanon E
Cat.No: TN1848
Synonym: 桑黄酮 E,桑皮酮 E,5'-[(E)-3,7-二甲基-2,6-辛二烯基]-2',4',5,7-四羟基黄烷酮
Target: AChR
Cyclomorusin
Cat.No: TN3744
Synonym:
Target: NOS, AChR
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